Small Molecule HMS LINCS ID	Small Molecule Name	Protein HMS LINCS ID	Protein Name	% Control	Assay compound conc	Conc unit
10047-101-3	Pictilisib	200001	AAK1	89.0	100	nM
10047-101-3	Pictilisib	200001	AAK1	93.0	1000	nM
10047-101-3	Pictilisib	200004	ABL1(E255K)-phosphorylated	73.0	100	nM
10047-101-3	Pictilisib	200004	ABL1(E255K)-phosphorylated	85.0	1000	nM
10047-101-3	Pictilisib	200006	ABL1(F317I)-nonphosphorylated	100.0	100	nM
10047-101-3	Pictilisib	200006	ABL1(F317I)-nonphosphorylated	100.0	1000	nM
10047-101-3	Pictilisib	200007	ABL1(F317I)-phosphorylated	100.0	100	nM
10047-101-3	Pictilisib	200007	ABL1(F317I)-phosphorylated	100.0	1000	nM
10047-101-3	Pictilisib	200009	ABL1(F317L)-nonphosphorylated	100.0	100	nM
10047-101-3	Pictilisib	200009	ABL1(F317L)-nonphosphorylated	100.0	1000	nM
10047-101-3	Pictilisib	200010	ABL1(F317L)-phosphorylated	100.0	100	nM
10047-101-3	Pictilisib	200010	ABL1(F317L)-phosphorylated	100.0	1000	nM
10047-101-3	Pictilisib	200012	ABL1(H396P)-nonphosphorylated	82.0	100	nM
10047-101-3	Pictilisib	200012	ABL1(H396P)-nonphosphorylated	81.0	1000	nM
10047-101-3	Pictilisib	200013	ABL1(H396P)-phosphorylated	100.0	100	nM
10047-101-3	Pictilisib	200013	ABL1(H396P)-phosphorylated	100.0	1000	nM
10047-101-3	Pictilisib	200015	ABL1(M351T)-phosphorylated	100.0	100	nM
10047-101-3	Pictilisib	200015	ABL1(M351T)-phosphorylated	100.0	1000	nM
10047-101-3	Pictilisib	200017	ABL1(Q252H)-nonphosphorylated	69.0	100	nM
10047-101-3	Pictilisib	200017	ABL1(Q252H)-nonphosphorylated	80.0	1000	nM
10047-101-3	Pictilisib	200018	ABL1(Q252H)-phosphorylated	100.0	100	nM
10047-101-3	Pictilisib	200018	ABL1(Q252H)-phosphorylated	100.0	1000	nM
10047-101-3	Pictilisib	200020	ABL1(T315I)-nonphosphorylated	100.0	100	nM
10047-101-3	Pictilisib	200020	ABL1(T315I)-nonphosphorylated	96.0	1000	nM
10047-101-3	Pictilisib	200021	ABL1(T315I)-phosphorylated	100.0	100	nM
10047-101-3	Pictilisib	200021	ABL1(T315I)-phosphorylated	100.0	1000	nM
10047-101-3	Pictilisib	200023	ABL1(Y253F)-phosphorylated	100.0	100	nM
10047-101-3	Pictilisib	200023	ABL1(Y253F)-phosphorylated	100.0	1000	nM
10047-101-3	Pictilisib	200024	ABL1-nonphosphorylated	83.0	100	nM
10047-101-3	Pictilisib	200024	ABL1-nonphosphorylated	85.0	1000	nM
10047-101-3	Pictilisib	200025	ABL1-phosphorylated	97.0	100	nM
10047-101-3	Pictilisib	200025	ABL1-phosphorylated	99.0	1000	nM
10047-101-3	Pictilisib	200026	ABL2	100.0	100	nM
10047-101-3	Pictilisib	200026	ABL2	99.0	1000	nM
10047-101-3	Pictilisib	200027	ACVR1	100.0	100	nM
10047-101-3	Pictilisib	200027	ACVR1	100.0	1000	nM
10047-101-3	Pictilisib	200028	ACVR1B	100.0	100	nM
10047-101-3	Pictilisib	200028	ACVR1B	100.0	1000	nM
10047-101-3	Pictilisib	200029	ACVR2A	81.0	100	nM
10047-101-3	Pictilisib	200029	ACVR2A	88.0	1000	nM
10047-101-3	Pictilisib	200030	ACVR2B	90.0	100	nM
10047-101-3	Pictilisib	200030	ACVR2B	100.0	1000	nM
10047-101-3	Pictilisib	200031	ACVRL1	100.0	100	nM
10047-101-3	Pictilisib	200031	ACVRL1	100.0	1000	nM
10047-101-3	Pictilisib	200032	ADCK3	95.0	100	nM
10047-101-3	Pictilisib	200032	ADCK3	91.0	1000	nM
10047-101-3	Pictilisib	200033	ADCK4	100.0	100	nM
10047-101-3	Pictilisib	200033	ADCK4	87.0	1000	nM
10047-101-3	Pictilisib	200034	AKT1	83.0	100	nM
10047-101-3	Pictilisib	200034	AKT1	100.0	1000	nM
10047-101-3	Pictilisib	200035	AKT2	95.0	100	nM
10047-101-3	Pictilisib	200035	AKT2	100.0	1000	nM
10047-101-3	Pictilisib	200036	AKT3	97.0	100	nM
10047-101-3	Pictilisib	200036	AKT3	96.0	1000	nM
10047-101-3	Pictilisib	200037	ALK	73.0	100	nM
10047-101-3	Pictilisib	200037	ALK	96.0	1000	nM
10047-101-3	Pictilisib	200479	ALK(C1156Y)	100.0	100	nM
10047-101-3	Pictilisib	200479	ALK(C1156Y)	100.0	1000	nM
10047-101-3	Pictilisib	200480	ALK(L1196M)	81.0	100	nM
10047-101-3	Pictilisib	200480	ALK(L1196M)	100.0	1000	nM
10047-101-3	Pictilisib	200038	AMPK-alpha1	94.0	100	nM
10047-101-3	Pictilisib	200038	AMPK-alpha1	88.0	1000	nM
10047-101-3	Pictilisib	200039	AMPK-alpha2	100.0	100	nM
10047-101-3	Pictilisib	200039	AMPK-alpha2	100.0	1000	nM
10047-101-3	Pictilisib	200040	ANKK1	100.0	100	nM
10047-101-3	Pictilisib	200040	ANKK1	100.0	1000	nM
10047-101-3	Pictilisib	200041	NUAK1	100.0	100	nM
10047-101-3	Pictilisib	200041	NUAK1	97.0	1000	nM
10047-101-3	Pictilisib	200042	M3K5	100.0	100	nM
10047-101-3	Pictilisib	200042	M3K5	100.0	1000	nM
10047-101-3	Pictilisib	200043	M3K6	100.0	100	nM
10047-101-3	Pictilisib	200043	M3K6	100.0	1000	nM
10047-101-3	Pictilisib	200044	AURKA	96.0	100	nM
10047-101-3	Pictilisib	200044	AURKA	100.0	1000	nM
10047-101-3	Pictilisib	200045	AURKB	96.0	100	nM
10047-101-3	Pictilisib	200045	AURKB	100.0	1000	nM
10047-101-3	Pictilisib	200046	AURKC	97.0	100	nM
10047-101-3	Pictilisib	200046	AURKC	100.0	1000	nM
10047-101-3	Pictilisib	200047	AXL	100.0	100	nM
10047-101-3	Pictilisib	200047	AXL	93.0	1000	nM
10047-101-3	Pictilisib	200048	BIKE	88.0	100	nM
10047-101-3	Pictilisib	200048	BIKE	85.0	1000	nM
10047-101-3	Pictilisib	200049	BLK	100.0	100	nM
10047-101-3	Pictilisib	200049	BLK	100.0	1000	nM
10047-101-3	Pictilisib	200050	BMPR1A	100.0	100	nM
10047-101-3	Pictilisib	200050	BMPR1A	100.0	1000	nM
10047-101-3	Pictilisib	200051	BMPR1B	100.0	100	nM
10047-101-3	Pictilisib	200051	BMPR1B	100.0	1000	nM
10047-101-3	Pictilisib	200052	BMPR2	100.0	100	nM
10047-101-3	Pictilisib	200052	BMPR2	100.0	1000	nM
10047-101-3	Pictilisib	200053	BMX	100.0	100	nM
10047-101-3	Pictilisib	200053	BMX	100.0	1000	nM
10047-101-3	Pictilisib	200054	BRAF	78.0	100	nM
10047-101-3	Pictilisib	200054	BRAF	92.0	1000	nM
10047-101-3	Pictilisib	200055	BRAF(V600E)	96.0	100	nM
10047-101-3	Pictilisib	200055	BRAF(V600E)	99.0	1000	nM
10047-101-3	Pictilisib	200056	PTK6	100.0	100	nM
10047-101-3	Pictilisib	200056	PTK6	100.0	1000	nM
10047-101-3	Pictilisib	200057	BRSK1	91.0	100	nM
10047-101-3	Pictilisib	200057	BRSK1	100.0	1000	nM
10047-101-3	Pictilisib	200058	BRSK2	100.0	100	nM
10047-101-3	Pictilisib	200058	BRSK2	88.0	1000	nM
10047-101-3	Pictilisib	200059	BTK	80.0	100	nM
10047-101-3	Pictilisib	200059	BTK	97.0	1000	nM
10047-101-3	Pictilisib	200470	BUB1	100.0	100	nM
10047-101-3	Pictilisib	200470	BUB1	100.0	1000	nM
10047-101-3	Pictilisib	200060	CAMK1	100.0	100	nM
10047-101-3	Pictilisib	200060	CAMK1	100.0	1000	nM
10047-101-3	Pictilisib	201324	CAMK1B	100.0	100	nM
10047-101-3	Pictilisib	201324	CAMK1B	100.0	1000	nM
10047-101-3	Pictilisib	200061	CAMK1D	100.0	100	nM
10047-101-3	Pictilisib	200061	CAMK1D	99.0	1000	nM
10047-101-3	Pictilisib	200062	CAMK1G	80.0	100	nM
10047-101-3	Pictilisib	200062	CAMK1G	100.0	1000	nM
10047-101-3	Pictilisib	200063	CAMK2A	97.0	100	nM
10047-101-3	Pictilisib	200063	CAMK2A	89.0	1000	nM
10047-101-3	Pictilisib	200064	CAMK2B	99.0	100	nM
10047-101-3	Pictilisib	200064	CAMK2B	87.0	1000	nM
10047-101-3	Pictilisib	200065	KCC2D	86.0	100	nM
10047-101-3	Pictilisib	200065	KCC2D	99.0	1000	nM
10047-101-3	Pictilisib	200066	CAMK2G	95.0	100	nM
10047-101-3	Pictilisib	200066	CAMK2G	100.0	1000	nM
10047-101-3	Pictilisib	200067	KCC4	100.0	100	nM
10047-101-3	Pictilisib	200067	KCC4	94.0	1000	nM
10047-101-3	Pictilisib	200068	KKCC1	96.0	100	nM
10047-101-3	Pictilisib	200068	KKCC1	84.0	1000	nM
10047-101-3	Pictilisib	200069	CAMKK2	91.0	100	nM
10047-101-3	Pictilisib	200069	CAMKK2	97.0	1000	nM
10047-101-3	Pictilisib	200070	CASK	68.0	100	nM
10047-101-3	Pictilisib	200070	CASK	78.0	1000	nM
10047-101-3	Pictilisib	200071	CDC2L1	100.0	100	nM
10047-101-3	Pictilisib	200071	CDC2L1	100.0	1000	nM
10047-101-3	Pictilisib	200072	CDC2L2	100.0	100	nM
10047-101-3	Pictilisib	200072	CDC2L2	100.0	1000	nM
10047-101-3	Pictilisib	200073	CDC2L5	63.0	100	nM
10047-101-3	Pictilisib	200073	CDC2L5	99.0	1000	nM
10047-101-3	Pictilisib	200074	CDK11	100.0	100	nM
10047-101-3	Pictilisib	200074	CDK11	99.0	1000	nM
10047-101-3	Pictilisib	200075	CDK2	100.0	100	nM
10047-101-3	Pictilisib	200075	CDK2	98.0	1000	nM
10047-101-3	Pictilisib	200076	CDK3	100.0	100	nM
10047-101-3	Pictilisib	200076	CDK3	100.0	1000	nM
10047-101-3	Pictilisib	200077	CDK4-cyclinD1	100.0	100	nM
10047-101-3	Pictilisib	200077	CDK4-cyclinD1	100.0	1000	nM
10047-101-3	Pictilisib	200077	CDK4-cyclinD1	94.0	100	nM
10047-101-3	Pictilisib	200077	CDK4-cyclinD1	98.0	1000	nM
10047-101-3	Pictilisib	200078	CDK4-cyclinD3	100.0	100	nM
10047-101-3	Pictilisib	200078	CDK4-cyclinD3	100.0	1000	nM
10047-101-3	Pictilisib	200079	CDK5	88.0	100	nM
10047-101-3	Pictilisib	200079	CDK5	94.0	1000	nM
10047-101-3	Pictilisib	200080	CDK7	100.0	100	nM
10047-101-3	Pictilisib	200080	CDK7	100.0	1000	nM
10047-101-3	Pictilisib	200081	CDK8	90.0	100	nM
10047-101-3	Pictilisib	200081	CDK8	92.0	1000	nM
10047-101-3	Pictilisib	200082	CDK9	100.0	100	nM
10047-101-3	Pictilisib	200082	CDK9	100.0	1000	nM
10047-101-3	Pictilisib	200083	CDKL1	75.0	100	nM
10047-101-3	Pictilisib	200083	CDKL1	84.0	1000	nM
10047-101-3	Pictilisib	200084	CDKL2	95.0	100	nM
10047-101-3	Pictilisib	200084	CDKL2	92.0	1000	nM
10047-101-3	Pictilisib	200085	CDKL3	95.0	100	nM
10047-101-3	Pictilisib	200085	CDKL3	100.0	1000	nM
10047-101-3	Pictilisib	200086	CDKL5	100.0	100	nM
10047-101-3	Pictilisib	200086	CDKL5	100.0	1000	nM
10047-101-3	Pictilisib	200087	CHEK1	100.0	100	nM
10047-101-3	Pictilisib	200087	CHEK1	100.0	1000	nM
10047-101-3	Pictilisib	200088	CHK2	100.0	100	nM
10047-101-3	Pictilisib	200088	CHK2	100.0	1000	nM
10047-101-3	Pictilisib	200089	CIT	97.0	100	nM
10047-101-3	Pictilisib	200089	CIT	98.0	1000	nM
10047-101-3	Pictilisib	200090	CLK1	86.0	100	nM
10047-101-3	Pictilisib	200090	CLK1	59.0	1000	nM
10047-101-3	Pictilisib	200091	CLK2	99.0	100	nM
10047-101-3	Pictilisib	200091	CLK2	55.0	1000	nM
10047-101-3	Pictilisib	200092	CLK3	100.0	100	nM
10047-101-3	Pictilisib	200092	CLK3	100.0	1000	nM
10047-101-3	Pictilisib	200093	CLK4	69.0	100	nM
10047-101-3	Pictilisib	200093	CLK4	56.0	1000	nM
10047-101-3	Pictilisib	200094	CSF1R	100.0	100	nM
10047-101-3	Pictilisib	200094	CSF1R	100.0	1000	nM
10047-101-3	Pictilisib	200471	CSF1R-autoinhibited	82.0	100	nM
10047-101-3	Pictilisib	200471	CSF1R-autoinhibited	96.0	1000	nM
10047-101-3	Pictilisib	200095	CSK	99.0	100	nM
10047-101-3	Pictilisib	200095	CSK	100.0	1000	nM
10047-101-3	Pictilisib	200096	CSNK1A1	84.0	100	nM
10047-101-3	Pictilisib	200096	CSNK1A1	88.0	1000	nM
10047-101-3	Pictilisib	200097	CSNK1A1L	100.0	100	nM
10047-101-3	Pictilisib	200097	CSNK1A1L	98.0	1000	nM
10047-101-3	Pictilisib	200098	CSNK1D	82.0	100	nM
10047-101-3	Pictilisib	200098	CSNK1D	66.0	1000	nM
10047-101-3	Pictilisib	200099	CSNK1E	100.0	100	nM
10047-101-3	Pictilisib	200099	CSNK1E	75.0	1000	nM
10047-101-3	Pictilisib	200100	KC1G1	100.0	100	nM
10047-101-3	Pictilisib	200100	KC1G1	100.0	1000	nM
10047-101-3	Pictilisib	200101	KC1G2	92.0	100	nM
10047-101-3	Pictilisib	200101	KC1G2	95.0	1000	nM
10047-101-3	Pictilisib	200102	CSNK1G3	100.0	100	nM
10047-101-3	Pictilisib	200102	CSNK1G3	99.0	1000	nM
10047-101-3	Pictilisib	200103	CSNK2A1	100.0	100	nM
10047-101-3	Pictilisib	200103	CSNK2A1	97.0	1000	nM
10047-101-3	Pictilisib	200104	CSNK2A2	91.0	100	nM
10047-101-3	Pictilisib	200104	CSNK2A2	95.0	1000	nM
10047-101-3	Pictilisib	200105	CTK	100.0	100	nM
10047-101-3	Pictilisib	200105	CTK	100.0	1000	nM
10047-101-3	Pictilisib	200106	DAPK1	78.0	100	nM
10047-101-3	Pictilisib	200106	DAPK1	77.0	1000	nM
10047-101-3	Pictilisib	200107	DAPK2	96.0	100	nM
10047-101-3	Pictilisib	200107	DAPK2	100.0	1000	nM
10047-101-3	Pictilisib	200108	DAPK3	91.0	100	nM
10047-101-3	Pictilisib	200108	DAPK3	82.0	1000	nM
10047-101-3	Pictilisib	200109	DCLK1	83.0	100	nM
10047-101-3	Pictilisib	200109	DCLK1	100.0	1000	nM
10047-101-3	Pictilisib	200110	DCAMKL2	99.0	100	nM
10047-101-3	Pictilisib	200110	DCAMKL2	100.0	1000	nM
10047-101-3	Pictilisib	200111	DCAMKL3	100.0	100	nM
10047-101-3	Pictilisib	200111	DCAMKL3	96.0	1000	nM
10047-101-3	Pictilisib	200112	DDR1	96.0	100	nM
10047-101-3	Pictilisib	200112	DDR1	100.0	1000	nM
10047-101-3	Pictilisib	200113	DDR2	93.0	100	nM
10047-101-3	Pictilisib	200113	DDR2	80.0	1000	nM
10047-101-3	Pictilisib	200114	M3K12	100.0	100	nM
10047-101-3	Pictilisib	200114	M3K12	100.0	1000	nM
10047-101-3	Pictilisib	200115	DMPK	100.0	100	nM
10047-101-3	Pictilisib	200115	DMPK	100.0	1000	nM
10047-101-3	Pictilisib	200116	DMPK2	100.0	100	nM
10047-101-3	Pictilisib	200116	DMPK2	100.0	1000	nM
10047-101-3	Pictilisib	200117	DRAK1	96.0	100	nM
10047-101-3	Pictilisib	200117	DRAK1	98.0	1000	nM
10047-101-3	Pictilisib	200118	DRAK2	90.0	100	nM
10047-101-3	Pictilisib	200118	DRAK2	100.0	1000	nM
10047-101-3	Pictilisib	200119	DYRK1A	100.0	100	nM
10047-101-3	Pictilisib	200119	DYRK1A	100.0	1000	nM
10047-101-3	Pictilisib	200120	DYRK1B	100.0	100	nM
10047-101-3	Pictilisib	200120	DYRK1B	99.0	1000	nM
10047-101-3	Pictilisib	200121	DYRK2	100.0	100	nM
10047-101-3	Pictilisib	200121	DYRK2	100.0	1000	nM
10047-101-3	Pictilisib	200122	EGFR	99.0	100	nM
10047-101-3	Pictilisib	200122	EGFR	100.0	1000	nM
10047-101-3	Pictilisib	200123	EGFR(E746-A750del)	91.0	100	nM
10047-101-3	Pictilisib	200123	EGFR(E746-A750del)	82.0	1000	nM
10047-101-3	Pictilisib	200124	EGFR(G719C)	100.0	100	nM
10047-101-3	Pictilisib	200124	EGFR(G719C)	100.0	1000	nM
10047-101-3	Pictilisib	200125	EGFR(G719S)	99.0	100	nM
10047-101-3	Pictilisib	200125	EGFR(G719S)	93.0	1000	nM
10047-101-3	Pictilisib	200126	EGFR(L747-E749del, A750P)	100.0	100	nM
10047-101-3	Pictilisib	200126	EGFR(L747-E749del, A750P)	100.0	1000	nM
10047-101-3	Pictilisib	200127	EGFR(L747-S752del, P753S)	64.0	100	nM
10047-101-3	Pictilisib	200127	EGFR(L747-S752del, P753S)	66.0	1000	nM
10047-101-3	Pictilisib	200128	EGFR(L747-T751del,Sins)	89.0	100	nM
10047-101-3	Pictilisib	200128	EGFR(L747-T751del,Sins)	98.0	1000	nM
10047-101-3	Pictilisib	200129	EGFR(L858R)	100.0	100	nM
10047-101-3	Pictilisib	200129	EGFR(L858R)	100.0	1000	nM
10047-101-3	Pictilisib	200130	EGFR(L858R,T790M)	98.0	100	nM
10047-101-3	Pictilisib	200130	EGFR(L858R,T790M)	100.0	1000	nM
10047-101-3	Pictilisib	200131	EGFR(L861Q)	88.0	100	nM
10047-101-3	Pictilisib	200131	EGFR(L861Q)	77.0	1000	nM
10047-101-3	Pictilisib	200132	EGFR(S752-I759del)	91.0	100	nM
10047-101-3	Pictilisib	200132	EGFR(S752-I759del)	94.0	1000	nM
10047-101-3	Pictilisib	200133	EGFR(T790M)	100.0	100	nM
10047-101-3	Pictilisib	200133	EGFR(T790M)	100.0	1000	nM
10047-101-3	Pictilisib	200134	EIF2AK1	100.0	100	nM
10047-101-3	Pictilisib	200134	EIF2AK1	100.0	1000	nM
10047-101-3	Pictilisib	200135	EPHA1	100.0	100	nM
10047-101-3	Pictilisib	200135	EPHA1	100.0	1000	nM
10047-101-3	Pictilisib	200136	EPHA2	77.0	100	nM
10047-101-3	Pictilisib	200136	EPHA2	83.0	1000	nM
10047-101-3	Pictilisib	200137	EPHA3	100.0	100	nM
10047-101-3	Pictilisib	200137	EPHA3	100.0	1000	nM
10047-101-3	Pictilisib	200138	EPHA4	100.0	100	nM
10047-101-3	Pictilisib	200138	EPHA4	100.0	1000	nM
10047-101-3	Pictilisib	200139	EPHA5	83.0	100	nM
10047-101-3	Pictilisib	200139	EPHA5	97.0	1000	nM
10047-101-3	Pictilisib	200140	EPHA6	100.0	100	nM
10047-101-3	Pictilisib	200140	EPHA6	100.0	1000	nM
10047-101-3	Pictilisib	200141	EPHA7	100.0	100	nM
10047-101-3	Pictilisib	200141	EPHA7	100.0	1000	nM
10047-101-3	Pictilisib	200142	EPHA8	100.0	100	nM
10047-101-3	Pictilisib	200142	EPHA8	100.0	1000	nM
10047-101-3	Pictilisib	200143	EPHB1	100.0	100	nM
10047-101-3	Pictilisib	200143	EPHB1	100.0	1000	nM
10047-101-3	Pictilisib	200144	EPHB2	100.0	100	nM
10047-101-3	Pictilisib	200144	EPHB2	98.0	1000	nM
10047-101-3	Pictilisib	200145	EPHB3	97.0	100	nM
10047-101-3	Pictilisib	200145	EPHB3	100.0	1000	nM
10047-101-3	Pictilisib	200146	EPHB4	98.0	100	nM
10047-101-3	Pictilisib	200146	EPHB4	96.0	1000	nM
10047-101-3	Pictilisib	200147	EPHB6	97.0	100	nM
10047-101-3	Pictilisib	200147	EPHB6	57.0	1000	nM
10047-101-3	Pictilisib	200148	ERBB2	99.0	100	nM
10047-101-3	Pictilisib	200148	ERBB2	92.0	1000	nM
10047-101-3	Pictilisib	200149	ERBB3	100.0	100	nM
10047-101-3	Pictilisib	200149	ERBB3	100.0	1000	nM
10047-101-3	Pictilisib	200150	ERBB4	93.0	100	nM
10047-101-3	Pictilisib	200150	ERBB4	97.0	1000	nM
10047-101-3	Pictilisib	200151	MK03	99.0	100	nM
10047-101-3	Pictilisib	200151	MK03	100.0	1000	nM
10047-101-3	Pictilisib	200152	MK01	89.0	100	nM
10047-101-3	Pictilisib	200152	MK01	98.0	1000	nM
10047-101-3	Pictilisib	200153	ERK3	100.0	100	nM
10047-101-3	Pictilisib	200153	ERK3	100.0	1000	nM
10047-101-3	Pictilisib	200154	ERK4	100.0	100	nM
10047-101-3	Pictilisib	200154	ERK4	100.0	1000	nM
10047-101-3	Pictilisib	200155	ERK5	93.0	100	nM
10047-101-3	Pictilisib	200155	ERK5	93.0	1000	nM
10047-101-3	Pictilisib	200156	ERK8	80.0	100	nM
10047-101-3	Pictilisib	200156	ERK8	99.0	1000	nM
10047-101-3	Pictilisib	200157	ERN1	100.0	100	nM
10047-101-3	Pictilisib	200157	ERN1	100.0	1000	nM
10047-101-3	Pictilisib	200158	FAK1	96.0	100	nM
10047-101-3	Pictilisib	200158	FAK1	95.0	1000	nM
10047-101-3	Pictilisib	200159	FER	75.0	100	nM
10047-101-3	Pictilisib	200159	FER	83.0	1000	nM
10047-101-3	Pictilisib	200160	FES	100.0	100	nM
10047-101-3	Pictilisib	200160	FES	100.0	1000	nM
10047-101-3	Pictilisib	200161	FGFR1	100.0	100	nM
10047-101-3	Pictilisib	200161	FGFR1	78.0	1000	nM
10047-101-3	Pictilisib	200162	FGFR2	89.0	100	nM
10047-101-3	Pictilisib	200162	FGFR2	100.0	1000	nM
10047-101-3	Pictilisib	200163	FGFR3	94.0	100	nM
10047-101-3	Pictilisib	200163	FGFR3	100.0	1000	nM
10047-101-3	Pictilisib	200164	FGFR3(G697C)	100.0	100	nM
10047-101-3	Pictilisib	200164	FGFR3(G697C)	100.0	1000	nM
10047-101-3	Pictilisib	200165	FGFR4	100.0	100	nM
10047-101-3	Pictilisib	200165	FGFR4	100.0	1000	nM
10047-101-3	Pictilisib	200166	FGR	100.0	100	nM
10047-101-3	Pictilisib	200166	FGR	100.0	1000	nM
10047-101-3	Pictilisib	200167	VGFR1	96.0	100	nM
10047-101-3	Pictilisib	200167	VGFR1	100.0	1000	nM
10047-101-3	Pictilisib	200168	FLT3	91.0	100	nM
10047-101-3	Pictilisib	200168	FLT3	67.0	1000	nM
10047-101-3	Pictilisib	200169	FLT3(D835H)	99.0	100	nM
10047-101-3	Pictilisib	200169	FLT3(D835H)	79.0	1000	nM
10047-101-3	Pictilisib	201325	FLT3(D835V)	86.0	100	nM
10047-101-3	Pictilisib	201325	FLT3(D835V)	62.0	1000	nM
10047-101-3	Pictilisib	200170	FLT3(D835Y)	100.0	100	nM
10047-101-3	Pictilisib	200170	FLT3(D835Y)	89.0	1000	nM
10047-101-3	Pictilisib	200171	FLT3(ITD)	100.0	100	nM
10047-101-3	Pictilisib	200171	FLT3(ITD)	79.0	1000	nM
10047-101-3	Pictilisib	201326	FLT3(ITD,D835V)	78.0	100	nM
10047-101-3	Pictilisib	201326	FLT3(ITD,D835V)	67.0	1000	nM
10047-101-3	Pictilisib	201327	FLT3(ITD,F691L)	92.0	100	nM
10047-101-3	Pictilisib	201327	FLT3(ITD,F691L)	71.0	1000	nM
10047-101-3	Pictilisib	200172	FLT3(K663Q)	100.0	100	nM
10047-101-3	Pictilisib	200172	FLT3(K663Q)	100.0	1000	nM
10047-101-3	Pictilisib	200173	FLT3(N841I)	100.0	100	nM
10047-101-3	Pictilisib	200173	FLT3(N841I)	100.0	1000	nM
10047-101-3	Pictilisib	200174	FLT3(R834Q)	100.0	100	nM
10047-101-3	Pictilisib	200174	FLT3(R834Q)	100.0	1000	nM
10047-101-3	Pictilisib	200472	FLT3-autoinhibited	97.0	100	nM
10047-101-3	Pictilisib	200472	FLT3-autoinhibited	100.0	1000	nM
10047-101-3	Pictilisib	200175	FLT4	100.0	100	nM
10047-101-3	Pictilisib	200175	FLT4	99.0	1000	nM
10047-101-3	Pictilisib	200176	FRK	96.0	100	nM
10047-101-3	Pictilisib	200176	FRK	95.0	1000	nM
10047-101-3	Pictilisib	200177	FYN	82.0	100	nM
10047-101-3	Pictilisib	200177	FYN	91.0	1000	nM
10047-101-3	Pictilisib	200178	GAK	100.0	100	nM
10047-101-3	Pictilisib	200178	GAK	100.0	1000	nM
10047-101-3	Pictilisib	200179	GCN2(Kin.Dom.2,S808G)	100.0	100	nM
10047-101-3	Pictilisib	200179	GCN2(Kin.Dom.2,S808G)	94.0	1000	nM
10047-101-3	Pictilisib	200180	GRK1	83.0	100	nM
10047-101-3	Pictilisib	200180	GRK1	100.0	1000	nM
10047-101-3	Pictilisib	201328	BARK1	100.0	100	nM
10047-101-3	Pictilisib	201328	BARK1	100.0	1000	nM
10047-101-3	Pictilisib	201329	BARK2	100.0	100	nM
10047-101-3	Pictilisib	201329	BARK2	100.0	1000	nM
10047-101-3	Pictilisib	200181	GRK4	93.0	100	nM
10047-101-3	Pictilisib	200181	GRK4	100.0	1000	nM
10047-101-3	Pictilisib	200182	GRK7	100.0	100	nM
10047-101-3	Pictilisib	200182	GRK7	100.0	1000	nM
10047-101-3	Pictilisib	200183	GSK3A	89.0	100	nM
10047-101-3	Pictilisib	200183	GSK3A	72.0	1000	nM
10047-101-3	Pictilisib	200184	GSK3B	100.0	100	nM
10047-101-3	Pictilisib	200184	GSK3B	100.0	1000	nM
10047-101-3	Pictilisib	200473	HASP	87.0	100	nM
10047-101-3	Pictilisib	200473	HASP	59.0	1000	nM
10047-101-3	Pictilisib	200185	HCK	96.0	100	nM
10047-101-3	Pictilisib	200185	HCK	99.0	1000	nM
10047-101-3	Pictilisib	200186	HIPK1	89.0	100	nM
10047-101-3	Pictilisib	200186	HIPK1	79.0	1000	nM
10047-101-3	Pictilisib	200187	HIPK2	100.0	100	nM
10047-101-3	Pictilisib	200187	HIPK2	61.0	1000	nM
10047-101-3	Pictilisib	200188	HIPK3	100.0	100	nM
10047-101-3	Pictilisib	200188	HIPK3	79.0	1000	nM
10047-101-3	Pictilisib	200189	HIPK4	95.0	100	nM
10047-101-3	Pictilisib	200189	HIPK4	87.0	1000	nM
10047-101-3	Pictilisib	200190	M4K1	85.0	100	nM
10047-101-3	Pictilisib	200190	M4K1	85.0	1000	nM
10047-101-3	Pictilisib	200191	HUNK	72.0	100	nM
10047-101-3	Pictilisib	200191	HUNK	100.0	1000	nM
10047-101-3	Pictilisib	200192	ICK	100.0	100	nM
10047-101-3	Pictilisib	200192	ICK	100.0	1000	nM
10047-101-3	Pictilisib	200193	IGF1R	100.0	100	nM
10047-101-3	Pictilisib	200193	IGF1R	100.0	1000	nM
10047-101-3	Pictilisib	200194	IKKA	100.0	100	nM
10047-101-3	Pictilisib	200194	IKKA	100.0	1000	nM
10047-101-3	Pictilisib	200195	IKKB	97.0	100	nM
10047-101-3	Pictilisib	200195	IKKB	100.0	1000	nM
10047-101-3	Pictilisib	200196	IKKE	100.0	100	nM
10047-101-3	Pictilisib	200196	IKKE	95.0	1000	nM
10047-101-3	Pictilisib	200197	INSR	100.0	100	nM
10047-101-3	Pictilisib	200197	INSR	100.0	1000	nM
10047-101-3	Pictilisib	200198	INSRR	100.0	100	nM
10047-101-3	Pictilisib	200198	INSRR	100.0	1000	nM
10047-101-3	Pictilisib	200199	IRAK1	100.0	100	nM
10047-101-3	Pictilisib	200199	IRAK1	100.0	1000	nM
10047-101-3	Pictilisib	200200	IRAK3	100.0	100	nM
10047-101-3	Pictilisib	200200	IRAK3	97.0	1000	nM
10047-101-3	Pictilisib	200201	IRAK4	100.0	100	nM
10047-101-3	Pictilisib	200201	IRAK4	100.0	1000	nM
10047-101-3	Pictilisib	200202	ITK	97.0	100	nM
10047-101-3	Pictilisib	200202	ITK	95.0	1000	nM
10047-101-3	Pictilisib	200203	JAK1(JH1domain-catalytic)	97.0	100	nM
10047-101-3	Pictilisib	200203	JAK1(JH1domain-catalytic)	92.0	1000	nM
10047-101-3	Pictilisib	200204	JAK1(JH2domain-pseudokinase)	76.0	100	nM
10047-101-3	Pictilisib	200204	JAK1(JH2domain-pseudokinase)	18.0	1000	nM
10047-101-3	Pictilisib	200207	JAK2(JH1domain-catalytic)	100.0	100	nM
10047-101-3	Pictilisib	200207	JAK2(JH1domain-catalytic)	88.0	1000	nM
10047-101-3	Pictilisib	200209	JAK3(JH1domain-catalytic)	92.0	100	nM
10047-101-3	Pictilisib	200209	JAK3(JH1domain-catalytic)	84.0	1000	nM
10047-101-3	Pictilisib	200211	JNK1	100.0	100	nM
10047-101-3	Pictilisib	200211	JNK1	71.0	1000	nM
10047-101-3	Pictilisib	200212	MK09	100.0	100	nM
10047-101-3	Pictilisib	200212	MK09	98.0	1000	nM
10047-101-3	Pictilisib	200213	JNK3	100.0	100	nM
10047-101-3	Pictilisib	200213	JNK3	93.0	1000	nM
10047-101-3	Pictilisib	200214	KIT	100.0	100	nM
10047-101-3	Pictilisib	200214	KIT	99.0	1000	nM
10047-101-3	Pictilisib	200215	KIT(A829P)	71.0	100	nM
10047-101-3	Pictilisib	200215	KIT(A829P)	100.0	1000	nM
10047-101-3	Pictilisib	200216	KIT(D816H)	88.0	100	nM
10047-101-3	Pictilisib	200216	KIT(D816H)	83.0	1000	nM
10047-101-3	Pictilisib	200217	KIT(D816V)	96.0	100	nM
10047-101-3	Pictilisib	200217	KIT(D816V)	97.0	1000	nM
10047-101-3	Pictilisib	200218	KIT(L576P)	100.0	100	nM
10047-101-3	Pictilisib	200218	KIT(L576P)	95.0	1000	nM
10047-101-3	Pictilisib	200219	KIT(V559D)	100.0	100	nM
10047-101-3	Pictilisib	200219	KIT(V559D)	100.0	1000	nM
10047-101-3	Pictilisib	200220	KIT(V559D,T670I)	100.0	100	nM
10047-101-3	Pictilisib	200220	KIT(V559D,T670I)	99.0	1000	nM
10047-101-3	Pictilisib	200221	KIT(V559D,V654A)	94.0	100	nM
10047-101-3	Pictilisib	200221	KIT(V559D,V654A)	100.0	1000	nM
10047-101-3	Pictilisib	200474	KIT-autoinhibited	72.0	100	nM
10047-101-3	Pictilisib	200474	KIT-autoinhibited	82.0	1000	nM
10047-101-3	Pictilisib	200222	LATS1	100.0	100	nM
10047-101-3	Pictilisib	200222	LATS1	100.0	1000	nM
10047-101-3	Pictilisib	200223	LATS2	100.0	100	nM
10047-101-3	Pictilisib	200223	LATS2	85.0	1000	nM
10047-101-3	Pictilisib	200224	LCK	82.0	100	nM
10047-101-3	Pictilisib	200224	LCK	85.0	1000	nM
10047-101-3	Pictilisib	200225	LIMK1	100.0	100	nM
10047-101-3	Pictilisib	200225	LIMK1	100.0	1000	nM
10047-101-3	Pictilisib	200226	LIMK2	100.0	100	nM
10047-101-3	Pictilisib	200226	LIMK2	99.0	1000	nM
10047-101-3	Pictilisib	200227	LKB1	92.0	100	nM
10047-101-3	Pictilisib	200227	LKB1	100.0	1000	nM
10047-101-3	Pictilisib	200228	LOK	95.0	100	nM
10047-101-3	Pictilisib	200228	LOK	93.0	1000	nM
10047-101-3	Pictilisib	200229	LRRK2	100.0	100	nM
10047-101-3	Pictilisib	200229	LRRK2	100.0	1000	nM
10047-101-3	Pictilisib	200230	LRRK2(G2019S)	100.0	100	nM
10047-101-3	Pictilisib	200230	LRRK2(G2019S)	100.0	1000	nM
10047-101-3	Pictilisib	200231	LTK	100.0	100	nM
10047-101-3	Pictilisib	200231	LTK	100.0	1000	nM
10047-101-3	Pictilisib	200232	LYN	100.0	100	nM
10047-101-3	Pictilisib	200232	LYN	100.0	1000	nM
10047-101-3	Pictilisib	200233	M3K13	100.0	100	nM
10047-101-3	Pictilisib	200233	M3K13	100.0	1000	nM
10047-101-3	Pictilisib	200234	MAK	100.0	100	nM
10047-101-3	Pictilisib	200234	MAK	90.0	1000	nM
10047-101-3	Pictilisib	200235	MAP3K1	100.0	100	nM
10047-101-3	Pictilisib	200235	MAP3K1	100.0	1000	nM
10047-101-3	Pictilisib	200236	MAP3K15	100.0	100	nM
10047-101-3	Pictilisib	200236	MAP3K15	100.0	1000	nM
10047-101-3	Pictilisib	200237	M3K2	98.0	100	nM
10047-101-3	Pictilisib	200237	M3K2	99.0	1000	nM
10047-101-3	Pictilisib	200238	MAP3K3	100.0	100	nM
10047-101-3	Pictilisib	200238	MAP3K3	100.0	1000	nM
10047-101-3	Pictilisib	200239	MAP3K4	100.0	100	nM
10047-101-3	Pictilisib	200239	MAP3K4	100.0	1000	nM
10047-101-3	Pictilisib	200240	MAP4K2	100.0	100	nM
10047-101-3	Pictilisib	200240	MAP4K2	100.0	1000	nM
10047-101-3	Pictilisib	200241	M4K3	98.0	100	nM
10047-101-3	Pictilisib	200241	M4K3	100.0	1000	nM
10047-101-3	Pictilisib	200242	MAP4K4	86.0	100	nM
10047-101-3	Pictilisib	200242	MAP4K4	88.0	1000	nM
10047-101-3	Pictilisib	200243	MAP4K5	91.0	100	nM
10047-101-3	Pictilisib	200243	MAP4K5	90.0	1000	nM
10047-101-3	Pictilisib	200244	MAPKAPK2	96.0	100	nM
10047-101-3	Pictilisib	200244	MAPKAPK2	100.0	1000	nM
10047-101-3	Pictilisib	200245	MAPKAPK5	100.0	100	nM
10047-101-3	Pictilisib	200245	MAPKAPK5	100.0	1000	nM
10047-101-3	Pictilisib	200246	MARK1	100.0	100	nM
10047-101-3	Pictilisib	200246	MARK1	86.0	1000	nM
10047-101-3	Pictilisib	200247	MARK2	100.0	100	nM
10047-101-3	Pictilisib	200247	MARK2	100.0	1000	nM
10047-101-3	Pictilisib	200248	MARK3	100.0	100	nM
10047-101-3	Pictilisib	200248	MARK3	100.0	1000	nM
10047-101-3	Pictilisib	200249	MARK4	100.0	100	nM
10047-101-3	Pictilisib	200249	MARK4	84.0	1000	nM
10047-101-3	Pictilisib	200250	MAST1	100.0	100	nM
10047-101-3	Pictilisib	200250	MAST1	100.0	1000	nM
10047-101-3	Pictilisib	200251	MP2K1	68.0	100	nM
10047-101-3	Pictilisib	200251	MP2K1	75.0	1000	nM
10047-101-3	Pictilisib	200252	MP2K2	81.0	100	nM
10047-101-3	Pictilisib	200252	MP2K2	96.0	1000	nM
10047-101-3	Pictilisib	200253	MP2K3	80.0	100	nM
10047-101-3	Pictilisib	200253	MP2K3	79.0	1000	nM
10047-101-3	Pictilisib	200254	MP2K4	100.0	100	nM
10047-101-3	Pictilisib	200254	MP2K4	100.0	1000	nM
10047-101-3	Pictilisib	200255	MP2K5	85.0	100	nM
10047-101-3	Pictilisib	200255	MP2K5	72.0	1000	nM
10047-101-3	Pictilisib	200256	MP2K6	100.0	100	nM
10047-101-3	Pictilisib	200256	MP2K6	100.0	1000	nM
10047-101-3	Pictilisib	200257	MELK	100.0	100	nM
10047-101-3	Pictilisib	200257	MELK	100.0	1000	nM
10047-101-3	Pictilisib	200258	MERTK	100.0	100	nM
10047-101-3	Pictilisib	200258	MERTK	100.0	1000	nM
10047-101-3	Pictilisib	200259	MET	98.0	100	nM
10047-101-3	Pictilisib	200259	MET	95.0	1000	nM
10047-101-3	Pictilisib	200260	MET(M1250T)	94.0	100	nM
10047-101-3	Pictilisib	200260	MET(M1250T)	100.0	1000	nM
10047-101-3	Pictilisib	200261	MET(Y1235D)	92.0	100	nM
10047-101-3	Pictilisib	200261	MET(Y1235D)	85.0	1000	nM
10047-101-3	Pictilisib	200262	MINK	69.0	100	nM
10047-101-3	Pictilisib	200262	MINK	72.0	1000	nM
10047-101-3	Pictilisib	200263	MP2K7	93.0	100	nM
10047-101-3	Pictilisib	200263	MP2K7	97.0	1000	nM
10047-101-3	Pictilisib	200264	MKNK1	60.0	100	nM
10047-101-3	Pictilisib	200264	MKNK1	86.0	1000	nM
10047-101-3	Pictilisib	200265	MKNK2	100.0	100	nM
10047-101-3	Pictilisib	200265	MKNK2	100.0	1000	nM
10047-101-3	Pictilisib	200266	MLCK	90.0	100	nM
10047-101-3	Pictilisib	200266	MLCK	79.0	1000	nM
10047-101-3	Pictilisib	200267	MLK1	66.0	100	nM
10047-101-3	Pictilisib	200267	MLK1	100.0	1000	nM
10047-101-3	Pictilisib	200268	MLK2	97.0	100	nM
10047-101-3	Pictilisib	200268	MLK2	75.0	1000	nM
10047-101-3	Pictilisib	200269	MLK3	64.0	100	nM
10047-101-3	Pictilisib	200269	MLK3	66.0	1000	nM
10047-101-3	Pictilisib	200270	MRCKA	100.0	100	nM
10047-101-3	Pictilisib	200270	MRCKA	100.0	1000	nM
10047-101-3	Pictilisib	200271	MRCKB	97.0	100	nM
10047-101-3	Pictilisib	200271	MRCKB	100.0	1000	nM
10047-101-3	Pictilisib	200272	MST1	97.0	100	nM
10047-101-3	Pictilisib	200272	MST1	99.0	1000	nM
10047-101-3	Pictilisib	200273	MST1R	100.0	100	nM
10047-101-3	Pictilisib	200273	MST1R	100.0	1000	nM
10047-101-3	Pictilisib	200274	MST2	90.0	100	nM
10047-101-3	Pictilisib	200274	MST2	100.0	1000	nM
10047-101-3	Pictilisib	200275	MST3	100.0	100	nM
10047-101-3	Pictilisib	200275	MST3	100.0	1000	nM
10047-101-3	Pictilisib	200276	MST4	100.0	100	nM
10047-101-3	Pictilisib	200276	MST4	100.0	1000	nM
10047-101-3	Pictilisib	200277	MTOR	66.0	100	nM
10047-101-3	Pictilisib	200277	MTOR	13.0	1000	nM
10047-101-3	Pictilisib	200278	MUSK	100.0	100	nM
10047-101-3	Pictilisib	200278	MUSK	100.0	1000	nM
10047-101-3	Pictilisib	200279	MYLK	87.0	100	nM
10047-101-3	Pictilisib	200279	MYLK	86.0	1000	nM
10047-101-3	Pictilisib	200280	MYLK2	100.0	100	nM
10047-101-3	Pictilisib	200280	MYLK2	100.0	1000	nM
10047-101-3	Pictilisib	200281	MYLK4	100.0	100	nM
10047-101-3	Pictilisib	200281	MYLK4	52.0	1000	nM
10047-101-3	Pictilisib	200282	MYO3A	100.0	100	nM
10047-101-3	Pictilisib	200282	MYO3A	100.0	1000	nM
10047-101-3	Pictilisib	200283	MYO3B	93.0	100	nM
10047-101-3	Pictilisib	200283	MYO3B	100.0	1000	nM
10047-101-3	Pictilisib	200284	NDR1	91.0	100	nM
10047-101-3	Pictilisib	200284	NDR1	90.0	1000	nM
10047-101-3	Pictilisib	200285	NDR2	100.0	100	nM
10047-101-3	Pictilisib	200285	NDR2	100.0	1000	nM
10047-101-3	Pictilisib	200286	NEK1	100.0	100	nM
10047-101-3	Pictilisib	200286	NEK1	92.0	1000	nM
10047-101-3	Pictilisib	200481	NEK10	93.0	100	nM
10047-101-3	Pictilisib	200481	NEK10	85.0	1000	nM
10047-101-3	Pictilisib	200287	NEK11	100.0	100	nM
10047-101-3	Pictilisib	200287	NEK11	100.0	1000	nM
10047-101-3	Pictilisib	200288	NEK2	100.0	100	nM
10047-101-3	Pictilisib	200288	NEK2	100.0	1000	nM
10047-101-3	Pictilisib	200289	NEK3	79.0	100	nM
10047-101-3	Pictilisib	200289	NEK3	81.0	1000	nM
10047-101-3	Pictilisib	200290	NEK4	100.0	100	nM
10047-101-3	Pictilisib	200290	NEK4	100.0	1000	nM
10047-101-3	Pictilisib	200291	NEK5	100.0	100	nM
10047-101-3	Pictilisib	200291	NEK5	99.0	1000	nM
10047-101-3	Pictilisib	200292	NEK6	95.0	100	nM
10047-101-3	Pictilisib	200292	NEK6	98.0	1000	nM
10047-101-3	Pictilisib	200293	NEK7	100.0	100	nM
10047-101-3	Pictilisib	200293	NEK7	100.0	1000	nM
10047-101-3	Pictilisib	200294	NEK9	100.0	100	nM
10047-101-3	Pictilisib	200294	NEK9	100.0	1000	nM
10047-101-3	Pictilisib	201107	MAP3K14	98.0	100	nM
10047-101-3	Pictilisib	201107	MAP3K14	100.0	1000	nM
10047-101-3	Pictilisib	200295	NIM1	100.0	100	nM
10047-101-3	Pictilisib	200295	NIM1	100.0	1000	nM
10047-101-3	Pictilisib	200296	NLK	98.0	100	nM
10047-101-3	Pictilisib	200296	NLK	100.0	1000	nM
10047-101-3	Pictilisib	200297	OSR1	100.0	100	nM
10047-101-3	Pictilisib	200297	OSR1	100.0	1000	nM
10047-101-3	Pictilisib	200298	MK14	100.0	100	nM
10047-101-3	Pictilisib	200298	MK14	100.0	1000	nM
10047-101-3	Pictilisib	200299	MK11	97.0	100	nM
10047-101-3	Pictilisib	200299	MK11	100.0	1000	nM
10047-101-3	Pictilisib	200300	MK13	99.0	100	nM
10047-101-3	Pictilisib	200300	MK13	99.0	1000	nM
10047-101-3	Pictilisib	200301	MK12	77.0	100	nM
10047-101-3	Pictilisib	200301	MK12	59.0	1000	nM
10047-101-3	Pictilisib	200302	PAK1	91.0	100	nM
10047-101-3	Pictilisib	200302	PAK1	100.0	1000	nM
10047-101-3	Pictilisib	200303	PAK2	78.0	100	nM
10047-101-3	Pictilisib	200303	PAK2	87.0	1000	nM
10047-101-3	Pictilisib	200304	PAK3	100.0	100	nM
10047-101-3	Pictilisib	200304	PAK3	100.0	1000	nM
10047-101-3	Pictilisib	200305	PAK4	96.0	100	nM
10047-101-3	Pictilisib	200305	PAK4	100.0	1000	nM
10047-101-3	Pictilisib	200306	PAK6	94.0	100	nM
10047-101-3	Pictilisib	200306	PAK6	90.0	1000	nM
10047-101-3	Pictilisib	200307	PAK7	99.0	100	nM
10047-101-3	Pictilisib	200307	PAK7	100.0	1000	nM
10047-101-3	Pictilisib	200309	CDK16	100.0	100	nM
10047-101-3	Pictilisib	200309	CDK16	100.0	1000	nM
10047-101-3	Pictilisib	200310	PCTK2	100.0	100	nM
10047-101-3	Pictilisib	200310	PCTK2	100.0	1000	nM
10047-101-3	Pictilisib	200311	PCTK3	95.0	100	nM
10047-101-3	Pictilisib	200311	PCTK3	94.0	1000	nM
10047-101-3	Pictilisib	200312	PGFRA	100.0	100	nM
10047-101-3	Pictilisib	200312	PGFRA	100.0	1000	nM
10047-101-3	Pictilisib	200313	PGFRB	100.0	100	nM
10047-101-3	Pictilisib	200313	PGFRB	100.0	1000	nM
10047-101-3	Pictilisib	200314	PDPK1	65.0	100	nM
10047-101-3	Pictilisib	200314	PDPK1	73.0	1000	nM
10047-101-3	Pictilisib	200315	PFCDPK1(P.falciparum)	98.0	100	nM
10047-101-3	Pictilisib	200315	PFCDPK1(P.falciparum)	90.0	1000	nM
10047-101-3	Pictilisib	200316	PFPK5(P.falciparum)	97.0	100	nM
10047-101-3	Pictilisib	200316	PFPK5(P.falciparum)	95.0	1000	nM
10047-101-3	Pictilisib	200317	CDK15	100.0	100	nM
10047-101-3	Pictilisib	200317	CDK15	100.0	1000	nM
10047-101-3	Pictilisib	200318	CDK14	86.0	100	nM
10047-101-3	Pictilisib	200318	CDK14	96.0	1000	nM
10047-101-3	Pictilisib	200319	PHKG1	100.0	100	nM
10047-101-3	Pictilisib	200319	PHKG1	100.0	1000	nM
10047-101-3	Pictilisib	200320	PHKG2	97.0	100	nM
10047-101-3	Pictilisib	200320	PHKG2	100.0	1000	nM
10047-101-3	Pictilisib	200321	PIK3C2B	100.0	100	nM
10047-101-3	Pictilisib	200321	PIK3C2B	18.0	1000	nM
10047-101-3	Pictilisib	200322	PIK3C2G	66.0	100	nM
10047-101-3	Pictilisib	200322	PIK3C2G	17.0	1000	nM
10047-101-3	Pictilisib	200323	PIK3CA	3.5	100	nM
10047-101-3	Pictilisib	200323	PIK3CA	0.2	1000	nM
10047-101-3	Pictilisib	200324	PIK3CA(C420R)	1.9	100	nM
10047-101-3	Pictilisib	200324	PIK3CA(C420R)	0.0	1000	nM
10047-101-3	Pictilisib	200325	PIK3CA(E542K)	1.2	100	nM
10047-101-3	Pictilisib	200325	PIK3CA(E542K)	0.0	1000	nM
10047-101-3	Pictilisib	200326	PIK3CA(E545A)	1.6	100	nM
10047-101-3	Pictilisib	200326	PIK3CA(E545A)	0.0	1000	nM
10047-101-3	Pictilisib	200327	PIK3CA(E545K)	0.8	100	nM
10047-101-3	Pictilisib	200327	PIK3CA(E545K)	0.0	1000	nM
10047-101-3	Pictilisib	200328	PIK3CA(H1047L)	17.0	100	nM
10047-101-3	Pictilisib	200328	PIK3CA(H1047L)	0.8	1000	nM
10047-101-3	Pictilisib	200329	PIK3CA(H1047Y)	1.0	100	nM
10047-101-3	Pictilisib	200329	PIK3CA(H1047Y)	0.0	1000	nM
10047-101-3	Pictilisib	200330	PIK3CA(I800L)	7.0	100	nM
10047-101-3	Pictilisib	200330	PIK3CA(I800L)	0.0	1000	nM
10047-101-3	Pictilisib	200331	PIK3CA(M1043I)	0.0	100	nM
10047-101-3	Pictilisib	200331	PIK3CA(M1043I)	0.4	1000	nM
10047-101-3	Pictilisib	200332	PIK3CA(Q546K)	4.0	100	nM
10047-101-3	Pictilisib	200332	PIK3CA(Q546K)	0.1	1000	nM
10047-101-3	Pictilisib	200333	PIK3CB	15.0	100	nM
10047-101-3	Pictilisib	200333	PIK3CB	0.0	1000	nM
10047-101-3	Pictilisib	200334	PIK3CD	7.0	100	nM
10047-101-3	Pictilisib	200334	PIK3CD	0.0	1000	nM
10047-101-3	Pictilisib	200335	PIK3CG	48.0	100	nM
10047-101-3	Pictilisib	200335	PIK3CG	3.5	1000	nM
10047-101-3	Pictilisib	200336	PIK4CB	100.0	100	nM
10047-101-3	Pictilisib	200336	PIK4CB	100.0	1000	nM
10047-101-3	Pictilisib	201330	FYV1	59.0	100	nM
10047-101-3	Pictilisib	201330	FYV1	4.5	1000	nM
10047-101-3	Pictilisib	200337	PIM1	89.0	100	nM
10047-101-3	Pictilisib	200337	PIM1	100.0	1000	nM
10047-101-3	Pictilisib	200338	PIM2	83.0	100	nM
10047-101-3	Pictilisib	200338	PIM2	100.0	1000	nM
10047-101-3	Pictilisib	200339	PIM3	88.0	100	nM
10047-101-3	Pictilisib	200339	PIM3	100.0	1000	nM
10047-101-3	Pictilisib	200340	PIP5K1A	99.0	100	nM
10047-101-3	Pictilisib	200340	PIP5K1A	100.0	1000	nM
10047-101-3	Pictilisib	200341	PIP5K1C	51.0	100	nM
10047-101-3	Pictilisib	200341	PIP5K1C	71.0	1000	nM
10047-101-3	Pictilisib	200342	PIP5K2B	100.0	100	nM
10047-101-3	Pictilisib	200342	PIP5K2B	100.0	1000	nM
10047-101-3	Pictilisib	200343	PI42C	78.0	100	nM
10047-101-3	Pictilisib	200343	PI42C	70.0	1000	nM
10047-101-3	Pictilisib	200344	PKAC-alpha	74.0	100	nM
10047-101-3	Pictilisib	200344	PKAC-alpha	93.0	1000	nM
10047-101-3	Pictilisib	200345	PKAC-beta	95.0	100	nM
10047-101-3	Pictilisib	200345	PKAC-beta	100.0	1000	nM
10047-101-3	Pictilisib	200346	PKMYT1	94.0	100	nM
10047-101-3	Pictilisib	200346	PKMYT1	97.0	1000	nM
10047-101-3	Pictilisib	200347	PKN1	100.0	100	nM
10047-101-3	Pictilisib	200347	PKN1	100.0	1000	nM
10047-101-3	Pictilisib	200348	PKN2	100.0	100	nM
10047-101-3	Pictilisib	200348	PKN2	100.0	1000	nM
10047-101-3	Pictilisib	200349	PKNB(M.tuberculosis)	100.0	100	nM
10047-101-3	Pictilisib	200349	PKNB(M.tuberculosis)	100.0	1000	nM
10047-101-3	Pictilisib	200350	PLK1	91.0	100	nM
10047-101-3	Pictilisib	200350	PLK1	91.0	1000	nM
10047-101-3	Pictilisib	200351	PLK2	99.0	100	nM
10047-101-3	Pictilisib	200351	PLK2	100.0	1000	nM
10047-101-3	Pictilisib	200352	PLK3	65.0	100	nM
10047-101-3	Pictilisib	200352	PLK3	81.0	1000	nM
10047-101-3	Pictilisib	200353	PLK4	97.0	100	nM
10047-101-3	Pictilisib	200353	PLK4	95.0	1000	nM
10047-101-3	Pictilisib	200354	KPCD	96.0	100	nM
10047-101-3	Pictilisib	200354	KPCD	83.0	1000	nM
10047-101-3	Pictilisib	200355	KPCE	73.0	100	nM
10047-101-3	Pictilisib	200355	KPCE	76.0	1000	nM
10047-101-3	Pictilisib	200356	KPCL	100.0	100	nM
10047-101-3	Pictilisib	200356	KPCL	100.0	1000	nM
10047-101-3	Pictilisib	200357	KPCI	75.0	100	nM
10047-101-3	Pictilisib	200357	KPCI	85.0	1000	nM
10047-101-3	Pictilisib	200358	KPCT	94.0	100	nM
10047-101-3	Pictilisib	200358	KPCT	85.0	1000	nM
10047-101-3	Pictilisib	200359	KPCD1	100.0	100	nM
10047-101-3	Pictilisib	200359	KPCD1	86.0	1000	nM
10047-101-3	Pictilisib	200360	KPCD2	97.0	100	nM
10047-101-3	Pictilisib	200360	KPCD2	95.0	1000	nM
10047-101-3	Pictilisib	200361	KPCD3	100.0	100	nM
10047-101-3	Pictilisib	200361	KPCD3	100.0	1000	nM
10047-101-3	Pictilisib	200362	KGP1	92.0	100	nM
10047-101-3	Pictilisib	200362	KGP1	65.0	1000	nM
10047-101-3	Pictilisib	200363	KGP2	93.0	100	nM
10047-101-3	Pictilisib	200363	KGP2	99.0	1000	nM
10047-101-3	Pictilisib	200364	PRKR	98.0	100	nM
10047-101-3	Pictilisib	200364	PRKR	100.0	1000	nM
10047-101-3	Pictilisib	200365	PRKX	100.0	100	nM
10047-101-3	Pictilisib	200365	PRKX	100.0	1000	nM
10047-101-3	Pictilisib	200366	PRP4	91.0	100	nM
10047-101-3	Pictilisib	200366	PRP4	83.0	1000	nM
10047-101-3	Pictilisib	200367	FAK2	100.0	100	nM
10047-101-3	Pictilisib	200367	FAK2	100.0	1000	nM
10047-101-3	Pictilisib	200368	SIK3	86.0	100	nM
10047-101-3	Pictilisib	200368	SIK3	100.0	1000	nM
10047-101-3	Pictilisib	200369	RAF1	100.0	100	nM
10047-101-3	Pictilisib	200369	RAF1	100.0	1000	nM
10047-101-3	Pictilisib	200370	RET	99.0	100	nM
10047-101-3	Pictilisib	200370	RET	91.0	1000	nM
10047-101-3	Pictilisib	200371	RET(M918T)	100.0	100	nM
10047-101-3	Pictilisib	200371	RET(M918T)	100.0	1000	nM
10047-101-3	Pictilisib	200372	RET(V804L)	100.0	100	nM
10047-101-3	Pictilisib	200372	RET(V804L)	100.0	1000	nM
10047-101-3	Pictilisib	200373	RET(V804M)	100.0	100	nM
10047-101-3	Pictilisib	200373	RET(V804M)	100.0	1000	nM
10047-101-3	Pictilisib	200374	RIOK1	85.0	100	nM
10047-101-3	Pictilisib	200374	RIOK1	98.0	1000	nM
10047-101-3	Pictilisib	200375	RIOK2	100.0	100	nM
10047-101-3	Pictilisib	200375	RIOK2	67.0	1000	nM
10047-101-3	Pictilisib	200376	RIOK3	98.0	100	nM
10047-101-3	Pictilisib	200376	RIOK3	95.0	1000	nM
10047-101-3	Pictilisib	200377	RIPK1	94.0	100	nM
10047-101-3	Pictilisib	200377	RIPK1	91.0	1000	nM
10047-101-3	Pictilisib	200378	RIPK2	100.0	100	nM
10047-101-3	Pictilisib	200378	RIPK2	98.0	1000	nM
10047-101-3	Pictilisib	200379	RIPK4	100.0	100	nM
10047-101-3	Pictilisib	200379	RIPK4	100.0	1000	nM
10047-101-3	Pictilisib	200380	RIPK5	100.0	100	nM
10047-101-3	Pictilisib	200380	RIPK5	100.0	1000	nM
10047-101-3	Pictilisib	200381	ROCK1	100.0	100	nM
10047-101-3	Pictilisib	200381	ROCK1	100.0	1000	nM
10047-101-3	Pictilisib	200382	ROCK2	100.0	100	nM
10047-101-3	Pictilisib	200382	ROCK2	100.0	1000	nM
10047-101-3	Pictilisib	200383	ROS1	74.0	100	nM
10047-101-3	Pictilisib	200383	ROS1	77.0	1000	nM
10047-101-3	Pictilisib	200390	RPS6KA4(Kin.Dom.1-N-terminal)	93.0	100	nM
10047-101-3	Pictilisib	200390	RPS6KA4(Kin.Dom.1-N-terminal)	93.0	1000	nM
10047-101-3	Pictilisib	200392	RPS6KA4(Kin.Dom.2-C-terminal)	98.0	100	nM
10047-101-3	Pictilisib	200392	RPS6KA4(Kin.Dom.2-C-terminal)	100.0	1000	nM
10047-101-3	Pictilisib	200394	RPS6KA5(Kin.Dom.1-N-terminal)	100.0	100	nM
10047-101-3	Pictilisib	200394	RPS6KA5(Kin.Dom.1-N-terminal)	100.0	1000	nM
10047-101-3	Pictilisib	200396	RPS6KA5(Kin.Dom.2-C-terminal)	100.0	100	nM
10047-101-3	Pictilisib	200396	RPS6KA5(Kin.Dom.2-C-terminal)	100.0	1000	nM
10047-101-3	Pictilisib	200399	RSK1(Kin.Dom.1-N-terminal)	100.0	100	nM
10047-101-3	Pictilisib	200399	RSK1(Kin.Dom.1-N-terminal)	94.0	1000	nM
10047-101-3	Pictilisib	200400	RSK1(Kin.Dom.2-C-terminal)	67.0	100	nM
10047-101-3	Pictilisib	200400	RSK1(Kin.Dom.2-C-terminal)	71.0	1000	nM
10047-101-3	Pictilisib	200401	RSK2(Kin.Dom.1-N-terminal)	87.0	100	nM
10047-101-3	Pictilisib	200401	RSK2(Kin.Dom.1-N-terminal)	80.0	1000	nM
10047-101-3	Pictilisib	200475	RSK2(Kin.Dom.2-C-terminal)	48.0	100	nM
10047-101-3	Pictilisib	200475	RSK2(Kin.Dom.2-C-terminal)	79.0	1000	nM
10047-101-3	Pictilisib	200402	RSK3(Kin.Dom.1-N-terminal)	86.0	100	nM
10047-101-3	Pictilisib	200402	RSK3(Kin.Dom.1-N-terminal)	84.0	1000	nM
10047-101-3	Pictilisib	200403	RSK3(Kin.Dom.2-C-terminal)	77.0	100	nM
10047-101-3	Pictilisib	200403	RSK3(Kin.Dom.2-C-terminal)	79.0	1000	nM
10047-101-3	Pictilisib	200404	RSK4(Kin.Dom.1-N-terminal)	100.0	100	nM
10047-101-3	Pictilisib	200404	RSK4(Kin.Dom.1-N-terminal)	100.0	1000	nM
10047-101-3	Pictilisib	200405	RSK4(Kin.Dom.2-C-terminal)	70.0	100	nM
10047-101-3	Pictilisib	200405	RSK4(Kin.Dom.2-C-terminal)	93.0	1000	nM
10047-101-3	Pictilisib	200406	S6K1	80.0	100	nM
10047-101-3	Pictilisib	200406	S6K1	93.0	1000	nM
10047-101-3	Pictilisib	200407	SBK1	100.0	100	nM
10047-101-3	Pictilisib	200407	SBK1	100.0	1000	nM
10047-101-3	Pictilisib	200476	SGK1	100.0	100	nM
10047-101-3	Pictilisib	200476	SGK1	100.0	1000	nM
10047-101-3	Pictilisib	200408	SgK110	93.0	100	nM
10047-101-3	Pictilisib	200408	SgK110	99.0	1000	nM
10047-101-3	Pictilisib	201108	SGK2	100.0	100	nM
10047-101-3	Pictilisib	201108	SGK2	100.0	1000	nM
10047-101-3	Pictilisib	200409	SGK3	100.0	100	nM
10047-101-3	Pictilisib	200409	SGK3	100.0	1000	nM
10047-101-3	Pictilisib	200410	SIK1	83.0	100	nM
10047-101-3	Pictilisib	200410	SIK1	100.0	1000	nM
10047-101-3	Pictilisib	200411	SIK2	100.0	100	nM
10047-101-3	Pictilisib	200411	SIK2	99.0	1000	nM
10047-101-3	Pictilisib	200412	SLK	84.0	100	nM
10047-101-3	Pictilisib	200412	SLK	87.0	1000	nM
10047-101-3	Pictilisib	200413	SNARK	100.0	100	nM
10047-101-3	Pictilisib	200413	SNARK	100.0	1000	nM
10047-101-3	Pictilisib	200414	SNRK	100.0	100	nM
10047-101-3	Pictilisib	200414	SNRK	100.0	1000	nM
10047-101-3	Pictilisib	200415	SRC	80.0	100	nM
10047-101-3	Pictilisib	200415	SRC	90.0	1000	nM
10047-101-3	Pictilisib	200416	SRMS	69.0	100	nM
10047-101-3	Pictilisib	200416	SRMS	83.0	1000	nM
10047-101-3	Pictilisib	200417	SRPK1	100.0	100	nM
10047-101-3	Pictilisib	200417	SRPK1	100.0	1000	nM
10047-101-3	Pictilisib	200418	SRPK2	91.0	100	nM
10047-101-3	Pictilisib	200418	SRPK2	90.0	1000	nM
10047-101-3	Pictilisib	200419	SRPK3	94.0	100	nM
10047-101-3	Pictilisib	200419	SRPK3	94.0	1000	nM
10047-101-3	Pictilisib	200420	STK16	100.0	100	nM
10047-101-3	Pictilisib	200420	STK16	81.0	1000	nM
10047-101-3	Pictilisib	200421	STK33	89.0	100	nM
10047-101-3	Pictilisib	200421	STK33	93.0	1000	nM
10047-101-3	Pictilisib	200422	STK35	100.0	100	nM
10047-101-3	Pictilisib	200422	STK35	100.0	1000	nM
10047-101-3	Pictilisib	200423	STK36	100.0	100	nM
10047-101-3	Pictilisib	200423	STK36	100.0	1000	nM
10047-101-3	Pictilisib	200424	STK39	100.0	100	nM
10047-101-3	Pictilisib	200424	STK39	98.0	1000	nM
10047-101-3	Pictilisib	200425	SYK	85.0	100	nM
10047-101-3	Pictilisib	200425	SYK	97.0	1000	nM
10047-101-3	Pictilisib	200426	TAK1	100.0	100	nM
10047-101-3	Pictilisib	200426	TAK1	100.0	1000	nM
10047-101-3	Pictilisib	200427	TAOK1	100.0	100	nM
10047-101-3	Pictilisib	200427	TAOK1	100.0	1000	nM
10047-101-3	Pictilisib	200428	TAOK2	68.0	100	nM
10047-101-3	Pictilisib	200428	TAOK2	100.0	1000	nM
10047-101-3	Pictilisib	200429	TAOK3	100.0	100	nM
10047-101-3	Pictilisib	200429	TAOK3	100.0	1000	nM
10047-101-3	Pictilisib	200430	TBK1	86.0	100	nM
10047-101-3	Pictilisib	200430	TBK1	79.0	1000	nM
10047-101-3	Pictilisib	200431	TEC	100.0	100	nM
10047-101-3	Pictilisib	200431	TEC	100.0	1000	nM
10047-101-3	Pictilisib	200432	TESK1	99.0	100	nM
10047-101-3	Pictilisib	200432	TESK1	100.0	1000	nM
10047-101-3	Pictilisib	200433	TGFBR1	100.0	100	nM
10047-101-3	Pictilisib	200433	TGFBR1	99.0	1000	nM
10047-101-3	Pictilisib	200434	TGFBR2	100.0	100	nM
10047-101-3	Pictilisib	200434	TGFBR2	100.0	1000	nM
10047-101-3	Pictilisib	200435	TIE1	100.0	100	nM
10047-101-3	Pictilisib	200435	TIE1	100.0	1000	nM
10047-101-3	Pictilisib	200436	TIE2	97.0	100	nM
10047-101-3	Pictilisib	200436	TIE2	100.0	1000	nM
10047-101-3	Pictilisib	200437	TLK1	73.0	100	nM
10047-101-3	Pictilisib	200437	TLK1	71.0	1000	nM
10047-101-3	Pictilisib	200438	TLK2	100.0	100	nM
10047-101-3	Pictilisib	200438	TLK2	100.0	1000	nM
10047-101-3	Pictilisib	200439	TNIK	64.0	100	nM
10047-101-3	Pictilisib	200439	TNIK	73.0	1000	nM
10047-101-3	Pictilisib	200440	TNK1	100.0	100	nM
10047-101-3	Pictilisib	200440	TNK1	75.0	1000	nM
10047-101-3	Pictilisib	200441	TNK2	100.0	100	nM
10047-101-3	Pictilisib	200441	TNK2	100.0	1000	nM
10047-101-3	Pictilisib	200442	TNNI3K	100.0	100	nM
10047-101-3	Pictilisib	200442	TNNI3K	100.0	1000	nM
10047-101-3	Pictilisib	200443	TRKA	100.0	100	nM
10047-101-3	Pictilisib	200443	TRKA	81.0	1000	nM
10047-101-3	Pictilisib	200444	TRKB	100.0	100	nM
10047-101-3	Pictilisib	200444	TRKB	100.0	1000	nM
10047-101-3	Pictilisib	200445	TRKC	100.0	100	nM
10047-101-3	Pictilisib	200445	TRKC	100.0	1000	nM
10047-101-3	Pictilisib	200446	TRPM6	100.0	100	nM
10047-101-3	Pictilisib	200446	TRPM6	100.0	1000	nM
10047-101-3	Pictilisib	200447	TSSK1	100.0	100	nM
10047-101-3	Pictilisib	200447	TSSK1	100.0	1000	nM
10047-101-3	Pictilisib	201331	TSSK3	100.0	100	nM
10047-101-3	Pictilisib	201331	TSSK3	100.0	1000	nM
10047-101-3	Pictilisib	200448	TTK	95.0	100	nM
10047-101-3	Pictilisib	200448	TTK	93.0	1000	nM
10047-101-3	Pictilisib	200449	TXK	100.0	100	nM
10047-101-3	Pictilisib	200449	TXK	100.0	1000	nM
10047-101-3	Pictilisib	200450	TYK2(JH1domain-catalytic)	100.0	100	nM
10047-101-3	Pictilisib	200450	TYK2(JH1domain-catalytic)	100.0	1000	nM
10047-101-3	Pictilisib	200451	TYK2(JH2domain-pseudokinase)	100.0	100	nM
10047-101-3	Pictilisib	200451	TYK2(JH2domain-pseudokinase)	96.0	1000	nM
10047-101-3	Pictilisib	200454	TYRO3	67.0	100	nM
10047-101-3	Pictilisib	200454	TYRO3	95.0	1000	nM
10047-101-3	Pictilisib	200455	ULK1	100.0	100	nM
10047-101-3	Pictilisib	200455	ULK1	100.0	1000	nM
10047-101-3	Pictilisib	200456	ULK2	100.0	100	nM
10047-101-3	Pictilisib	200456	ULK2	100.0	1000	nM
10047-101-3	Pictilisib	200457	ULK3	100.0	100	nM
10047-101-3	Pictilisib	200457	ULK3	100.0	1000	nM
10047-101-3	Pictilisib	200458	VGFR2	95.0	100	nM
10047-101-3	Pictilisib	200458	VGFR2	100.0	1000	nM
10047-101-3	Pictilisib	201332	PIK3C3	100.0	100	nM
10047-101-3	Pictilisib	201332	PIK3C3	84.0	1000	nM
10047-101-3	Pictilisib	200459	VRK2	74.0	100	nM
10047-101-3	Pictilisib	200459	VRK2	54.0	1000	nM
10047-101-3	Pictilisib	200460	WEE1	88.0	100	nM
10047-101-3	Pictilisib	200460	WEE1	99.0	1000	nM
10047-101-3	Pictilisib	200461	WEE2	98.0	100	nM
10047-101-3	Pictilisib	200461	WEE2	100.0	1000	nM
10047-101-3	Pictilisib	200477	WNK1	90.0	100	nM
10047-101-3	Pictilisib	200477	WNK1	100.0	1000	nM
10047-101-3	Pictilisib	201333	WNK2	100.0	100	nM
10047-101-3	Pictilisib	201333	WNK2	100.0	1000	nM
10047-101-3	Pictilisib	200478	WNK3	100.0	100	nM
10047-101-3	Pictilisib	200478	WNK3	100.0	1000	nM
10047-101-3	Pictilisib	201334	WNK4	100.0	100	nM
10047-101-3	Pictilisib	201334	WNK4	100.0	1000	nM
10047-101-3	Pictilisib	200462	YANK1	100.0	100	nM
10047-101-3	Pictilisib	200462	YANK1	100.0	1000	nM
10047-101-3	Pictilisib	200463	YANK2	98.0	100	nM
10047-101-3	Pictilisib	200463	YANK2	100.0	1000	nM
10047-101-3	Pictilisib	200464	YANK3	100.0	100	nM
10047-101-3	Pictilisib	200464	YANK3	100.0	1000	nM
10047-101-3	Pictilisib	200465	YES	100.0	100	nM
10047-101-3	Pictilisib	200465	YES	100.0	1000	nM
10047-101-3	Pictilisib	200466	YSK1	100.0	100	nM
10047-101-3	Pictilisib	200466	YSK1	100.0	1000	nM
10047-101-3	Pictilisib	200467	YSK4	100.0	100	nM
10047-101-3	Pictilisib	200467	YSK4	95.0	1000	nM
10047-101-3	Pictilisib	200468	MLTK	100.0	100	nM
10047-101-3	Pictilisib	200468	MLTK	100.0	1000	nM
10047-101-3	Pictilisib	200469	ZAP70	86.0	100	nM
10047-101-3	Pictilisib	200469	ZAP70	100.0	1000	nM
