Small Molecule HMS LINCS ID	Small Molecule Name	Cell Line HMS LINCS ID	Cell Line Name	Protein HMS LINCS ID	Protein Name	Sequence	Labeling Site	% Inhibition	Assay compound conc	Conc unit
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200633	ABL,ARG	LMTGDTYTAHAGAKFPIK	Activation Loop	>90	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200635	ACK	TVSVAVKCLKPDVLSQPEAMDDFIR	Lys1	-33.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200640	AMPKa1,AMPKa2	VAVKILNR	Lys1	9.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200643	ATR	FYIMMCKPK	ATP	21.3	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200644	AurA	DIKPENLLLGSAGELK	Lys2	-1.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201072	AurB	SHFIVALKVLFK	Lys1	-84.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200877	BARK1	DLKPANILLDEHGHVR	Lys2	10.8	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200647	BRAF	DLKSNNIFLHEDLTVK	Lys2	-17.0	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200880	BTK	GQYDVAIKMIK	Lys1	-31.3	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200881	BTK	YVLDDEYTSSVGSKFPVR	Activation Loop	-24.0	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200882	CAMK1D	LFAVKCIPK	Lys1	-9.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201047	CaMK2a,CaMK2b,CaMK2d,CaMK2g	DLKPENLLLASK	Lys2	8.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200654	CDC2	DLKPQNLLIDDKGTIK	Lys2	52.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200656	CDK11,CDK8	DLKPANILVMGEGPER	Lys2	52.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200658	CDK2	DLKPQNLLINTEGAIK	Lys2	61.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200890	CDK5	DLKPQNLLINR	Lys2	61.3	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200663	CDK7	DLKPNNLLLDENGVLK	Lys2	-0.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200666	CHK2	VAIKIISK	Lys1	-0.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200667	KC1A	DIKPDNFLMGIGR	Lys2	20.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200669	CSK	VSDFGLTKEASSTQDTGKLPVK	Activation Loop	8.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200674	DNAPK	EHPFLVKGGEDLR	ATP	34.0	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200677	eEF2K	YIKYNSNSGFVR	ATP	3.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200681	MK03	DLKPSNLLINTTCDLK	Lys2	2.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200686	FER	TSVAVKTCKEDLPQELK	Lys1	-21.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200918	FGR	LIKDDEYNPCQGSKFPIK	Activation Loop	26.8	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200921	FRAP1	IQSIAPSLQVITSKQRPR	ATP	-15.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200687	FYN,SRC,YES	QGAKFPIKWTAPEAALYGR	Activation Loop	39.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200690	GCK	DIKGANLLLTLQGDVK	Lys2	26.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200693	GSK3A	DIKPQNLLVDPDTAVLK	Lys2	5.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200694	GSK3B	DIKPQNLLLDPDTAVLK	Lys2	32.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200928	HPK1	DKVSGDLVALKMVK	Lys1	1.8	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200933	IKKE	SGELVAVKVFNTTSYLRPR	Lys1	-0.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200697	IKKE,TBK1	DIKPGNIMR	Lys2	7.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200698	ILK	ISMADVKFSFQCPGR	Protein Kinase Domain	-26.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200701	IRAK4	DIKSANILLDEAFTAK	Lys2	33.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200704	JAK1	QLASALSYLEDKDLVHGNVCTKNLLLAR	Protein Kinase Domain	29.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200705	JAK1_domain2	YDPEGDNTGEQVAVKSLKPESGGNHIADLKK	Lys1	19.3	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200707	JNK1,JNK2,JNK3	DLKPSNIVVK	Lys2	10.7	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200710	KHS1	NVHTGELAAVKIIK	Lys1	-13.0	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200712	LKB1	DIKPGNLLLTTGGTLK	Lys2	-2.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200714	LOK	DLKAGNVLMTLEGDIR	Lys2	63.0	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200940	LYN	VAVKTLKPGTMSVQAFLEEANLMK	Lys1	90.7	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200941	LYN	EGAKFPIKWTAPEAINFGCFTIK	Activation Loop	79.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200718	MAP2K1	IMHRDVKPSNILVNSR	Lys2	-11.8	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200719	MAP2K1,MAP2K2	DVKPSNILVNSR	Lys2	0.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200722	MAP2K3	DVKPSNVLINK	Lys2	-10.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200724	MAP2K4	DIKPSNILLDR	Lys2	-8.7	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200725	MAP2K5	DVKPSNMLVNTR	Lys2	4.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200726	MAP2K6	DVKPSNVLINALGQVK	Lys2	-2.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200729	MP2K7	DVKPSNILLDER	Lys2	-0.7	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200730	MAP3K1	DVKGANLLIDSTGQR	Lys2	88.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200732	M3K2,MAP3K3	DIKGANILR	Lys2	-16.8	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200734	MAP3K4	DIKGANIFLTSSGLIK	Lys2	4.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200944	MAP3K5	DIKGDNVLINTYSGVLK	Lys2	9.8	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200739	MARK2,MARK3	DLKAENLLLDADMNIK	Lys2	6.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200740	MARK3	EVAIKIIDKTQLNPTSLQK	Lys1	-11.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200743	MAST3	DLKPDNLLITSLGHIK	Lys2	26.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200950	MASTL	LYAVKVVK	Lys1	-2.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200751	MST1	ETGQIVAIKQVPVESDLQEIIK	Lys1	-2.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200755	MST2	ESGQVVAIKQVPVESDLQEIIK	Lys1	0.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200756	MST3	DIKAANVLLSEHGEVK	Lys2	8.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200759	MST4,YSK1	DIKAANVLLSEQGDVK	Lys2	19.0	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200760	NDR1	DTGHVYAMKILR	Lys1	-12.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200765	NDR2	DIKPDNLLLDAK	Lys2	-7.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200960	NEK3	SKNIFLTQNGK	Activation Loop	4.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200768	NEK6,NEK7	DIKPANVFITATGVVK	Lys2	13.0	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200770	NEK7	AACLLDGVPVALKK	Lys1	1.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200774	NEK9	DIKTLNIFLTK	Lys2	0.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200967	MK14	QELNKTIWEVPER	Protein Kinase Domain	69.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200777	p38d,p38g	DLKPGNLAVNEDCELK	Lys2	57.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200779	KS6B1	DLKPENIMLNHQGHVK	Lys2	-16.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200787	CDK14	LVALKVIR	Lys1	94.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200790	PI4KB	VPHTQAVVLNSKDK	ATP	-10.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200793	PIK3C3	TEDGGKYPVIFKHGDDLR	ATP	-6.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200976	PIK3CB	VFGEDSVGVIFKNGDDLR	ATP	1.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200977	PIK3CD	VNWLAHNVSKDNRQ	ATP	-3.3	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200797	PIP4K2A	AKELPTLKDNDFINEGQK	ATP	14.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200799	PI42C	TLVIKEVSSEDIADMHSNLSNYHQYIVK	ATP	-9.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200800	FYV1	GGKSGAAFYATEDDRFILK	ATP	16.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200801	PITSLRE	DLKTSNLLLSHAGILK	Lys2	9.8	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200805	PKD1,PKD2	NIVHCDLKPENVLLASADPFPQVK	Lys2	-4.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201064	PKD2	DVAVKVIDK	Lys1	-16.8	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200807	PKD3	NIVHCDLKPENVLLASAEPFPQVK	Lys2	13.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201094	PKN1	VLLSEFRPSGELFAIKALK	Lys1	-85.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200809	PKR	DLKPSNIFLVDTK	Lys2	-14.7	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200810	PLK1	CFEISDADTKEVFAGKIVPK	Lys1	-14.3	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200997	FAK2	YIEDEDYYKASVTR	Activation Loop	28.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200814	ROCK1,ROCK2	DVKPDNMLLDK	Lys2	-19.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201045	RSK1 domain1	DLKPENILLDEEGHIKLTDFGLSKEAIDHEK	Lys2	26.8	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200819	RSK1_domain2	DLKPSNILYVDESGNPECLR	Lys2	-7.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200821	RSK2_domain2	DLKPSNILYVDESGNPESIR	Lys2	1.7	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200826	SGK3	FYAVKVLQK	Lys1	-12.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200829	SLK	DLKAGNILFTLDGDIK	Lys2	-35.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200833	STLK5	YSVKVLPWLSPEVLQQNLQGYDAK	Activation Loop	5.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201099	STLK6	SIKASHILISGDGLVTLSGLSHLHSLVK	Lys2	-1.8	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201069	SYK	ISDFGLSKALR	Activation Loop	-12.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201017	SYK	TVAVKILK	Lys1	-31.7	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200834	TAO1,TAOK3	DIKAGNILLTEPGQVK	Lys2	25.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200835	TAOK2	DVKAGNILLSEPGLVK	Lys2	4.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201077	TEC	YVLDDQYTSSSGAKFPVK	Activation Loop	-13.7	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200837	TLK1	YLNEIKPPIIHYDLKPGNILLVDGTACGEIK	Lys2	18.5	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201022	TLK1/2	YLNEIKPPIIHYDLKPGNILLVNGTACGEIK	Lys2	-19.6	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201026	ULK3	EVVAIKCVAK	Lys1	-25.3	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200845	MLTK	WISQDKEVAVKK	Lys1	80.7	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	200847	ZC1/HGK,ZC2/TNIK,ZC3/MINK	DIKGQNVLLTENAEVK	Lys2	72.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201163	BLK	IIDSEYTAQEGAKFPIK	Activation Loop	76.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201210	KCC2D	IPTGQEYAAKIINTKK	Lys1	-4.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201208	KC1G1	DVKPENFLIGR	Lys2	8.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201209	KC1G2	DVKPENFLVGRPGTK	Lys2	20.1	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201217	LCK	EGAKFPIKWTAPEAINYGTFTIK	Activation Loop	75.4	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201231	MARK1,MARK2	EVAVKIIDK	Lys1	-16.2	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201213	KPCI	DLKLDNVLLDSEGHIK	Lys2	-16.0	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201282	ZAP70	ISDFGLSKALGADDSYYTAR	Activation Loop	3.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201167	KCC4	DLKPENLLYATPAPDAPLK	Lys2	33.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201192	MK01	DLKPSNLLLNTTCDLK	Lys2	-17.9	1	uM
10351-101-1	DCC-2036	50811-1	Ramos (RA 1)	201262	RSK2 domain1	DLKPENILLDEEGHIKLTDFGLSKESIDHEK	Lys2	30.4	1	uM
