Small Molecule HMS LINCS ID	Small Molecule Name	Protein HMS LINCS ID	Protein Name	Kd	Conc unit
10024-999-3	NVP-TAE684	200001	AAK1	470.0	nM
10024-999-3	NVP-TAE684	200004	ABL1(E255K)-phosphorylated	190.0	nM
10024-999-3	NVP-TAE684	200006	ABL1(F317I)-nonphosphorylated	93.0	nM
10024-999-3	NVP-TAE684	200007	ABL1(F317I)-phosphorylated	14.0	nM
10024-999-3	NVP-TAE684	200009	ABL1(F317L)-nonphosphorylated	54.0	nM
10024-999-3	NVP-TAE684	200010	ABL1(F317L)-phosphorylated	19.0	nM
10024-999-3	NVP-TAE684	200012	ABL1(H396P)-nonphosphorylated	73.0	nM
10024-999-3	NVP-TAE684	200013	ABL1(H396P)-phosphorylated	160.0	nM
10024-999-3	NVP-TAE684	200015	ABL1(M351T)-phosphorylated	95.0	nM
10024-999-3	NVP-TAE684	200017	ABL1(Q252H)-nonphosphorylated	39.0	nM
10024-999-3	NVP-TAE684	200018	ABL1(Q252H)-phosphorylated	70.0	nM
10024-999-3	NVP-TAE684	200020	ABL1(T315I)-nonphosphorylated	52.0	nM
10024-999-3	NVP-TAE684	200021	ABL1(T315I)-phosphorylated	5.4	nM
10024-999-3	NVP-TAE684	200023	ABL1(Y253F)-phosphorylated	100.0	nM
10024-999-3	NVP-TAE684	200024	ABL1-nonphosphorylated	200.0	nM
10024-999-3	NVP-TAE684	200025	ABL1-phosphorylated	170.0	nM
10024-999-3	NVP-TAE684	200026	ABL2	380.0	nM
10024-999-3	NVP-TAE684	200027	ACVR1	29.0	nM
10024-999-3	NVP-TAE684	200028	ACVR1B	97.0	nM
10024-999-3	NVP-TAE684	200029	ACVR2A	2200.0	nM
10024-999-3	NVP-TAE684	200030	ACVR2B	4300.0	nM
10024-999-3	NVP-TAE684	200031	ACVRL1	57.0	nM
10024-999-3	NVP-TAE684	200032	ADCK3	1700.0	nM
10024-999-3	NVP-TAE684	200033	ADCK4	92.0	nM
10024-999-3	NVP-TAE684	200034	AKT1		nM
10024-999-3	NVP-TAE684	200035	AKT2		nM
10024-999-3	NVP-TAE684	200036	AKT3		nM
10024-999-3	NVP-TAE684	200037	ALK	1.1	nM
10024-999-3	NVP-TAE684	200038	AMPK-alpha1	27.0	nM
10024-999-3	NVP-TAE684	200039	AMPK-alpha2	49.0	nM
10024-999-3	NVP-TAE684	200040	ANKK1	9400.0	nM
10024-999-3	NVP-TAE684	200041	NUAK1	13.0	nM
10024-999-3	NVP-TAE684	200042	M3K5		nM
10024-999-3	NVP-TAE684	200043	M3K6	1800.0	nM
10024-999-3	NVP-TAE684	200044	AURKA	44.0	nM
10024-999-3	NVP-TAE684	200045	AURKB	150.0	nM
10024-999-3	NVP-TAE684	200046	AURKC	33.0	nM
10024-999-3	NVP-TAE684	200047	AXL	12.0	nM
10024-999-3	NVP-TAE684	200048	BIKE	1900.0	nM
10024-999-3	NVP-TAE684	200049	BLK	130.0	nM
10024-999-3	NVP-TAE684	200050	BMPR1A	170.0	nM
10024-999-3	NVP-TAE684	200051	BMPR1B	0.9	nM
10024-999-3	NVP-TAE684	200052	BMPR2	3900.0	nM
10024-999-3	NVP-TAE684	200053	BMX	1100.0	nM
10024-999-3	NVP-TAE684	200054	BRAF		nM
10024-999-3	NVP-TAE684	200055	BRAF(V600E)		nM
10024-999-3	NVP-TAE684	200056	PTK6	36.0	nM
10024-999-3	NVP-TAE684	200057	BRSK1	310.0	nM
10024-999-3	NVP-TAE684	200058	BRSK2	190.0	nM
10024-999-3	NVP-TAE684	200059	BTK	23.0	nM
10024-999-3	NVP-TAE684	200060	CAMK1	1100.0	nM
10024-999-3	NVP-TAE684	200061	CAMK1D	230.0	nM
10024-999-3	NVP-TAE684	200062	CAMK1G	3000.0	nM
10024-999-3	NVP-TAE684	200063	CAMK2A	980.0	nM
10024-999-3	NVP-TAE684	200064	CAMK2B	1900.0	nM
10024-999-3	NVP-TAE684	200065	KCC2D	570.0	nM
10024-999-3	NVP-TAE684	200066	CAMK2G	780.0	nM
10024-999-3	NVP-TAE684	200067	KCC4	30.0	nM
10024-999-3	NVP-TAE684	200068	KKCC1	50.0	nM
10024-999-3	NVP-TAE684	200069	CAMKK2	11.0	nM
10024-999-3	NVP-TAE684	200070	CASK	920.0	nM
10024-999-3	NVP-TAE684	200071	CDC2L1		nM
10024-999-3	NVP-TAE684	200072	CDC2L2		nM
10024-999-3	NVP-TAE684	200073	CDC2L5		nM
10024-999-3	NVP-TAE684	200074	CDK11		nM
10024-999-3	NVP-TAE684	200075	CDK2	5200.0	nM
10024-999-3	NVP-TAE684	200076	CDK3		nM
10024-999-3	NVP-TAE684	200077	CDK4-cyclinD1	1400.0	nM
10024-999-3	NVP-TAE684	200078	CDK4-cyclinD3	400.0	nM
10024-999-3	NVP-TAE684	200079	CDK5	1600.0	nM
10024-999-3	NVP-TAE684	200080	CDK7	190.0	nM
10024-999-3	NVP-TAE684	200081	CDK8		nM
10024-999-3	NVP-TAE684	200082	CDK9		nM
10024-999-3	NVP-TAE684	200083	CDKL1		nM
10024-999-3	NVP-TAE684	200084	CDKL2		nM
10024-999-3	NVP-TAE684	200085	CDKL3		nM
10024-999-3	NVP-TAE684	200086	CDKL5		nM
10024-999-3	NVP-TAE684	200087	CHEK1	44.0	nM
10024-999-3	NVP-TAE684	200088	CHK2	72.0	nM
10024-999-3	NVP-TAE684	200089	CIT		nM
10024-999-3	NVP-TAE684	200090	CLK1	12.0	nM
10024-999-3	NVP-TAE684	200091	CLK2	82.0	nM
10024-999-3	NVP-TAE684	200092	CLK3	210.0	nM
10024-999-3	NVP-TAE684	200093	CLK4	110.0	nM
10024-999-3	NVP-TAE684	200094	CSF1R	48.0	nM
10024-999-3	NVP-TAE684	200095	CSK	1800.0	nM
10024-999-3	NVP-TAE684	200096	CSNK1A1		nM
10024-999-3	NVP-TAE684	200097	CSNK1A1L	5200.0	nM
10024-999-3	NVP-TAE684	200098	CSNK1D		nM
10024-999-3	NVP-TAE684	200099	CSNK1E		nM
10024-999-3	NVP-TAE684	200100	KC1G1		nM
10024-999-3	NVP-TAE684	200101	KC1G2		nM
10024-999-3	NVP-TAE684	200102	CSNK1G3		nM
10024-999-3	NVP-TAE684	200103	CSNK2A1		nM
10024-999-3	NVP-TAE684	200104	CSNK2A2	9600.0	nM
10024-999-3	NVP-TAE684	200105	CTK	2800.0	nM
10024-999-3	NVP-TAE684	200106	DAPK1	1800.0	nM
10024-999-3	NVP-TAE684	200107	DAPK2	870.0	nM
10024-999-3	NVP-TAE684	200108	DAPK3	2200.0	nM
10024-999-3	NVP-TAE684	200109	DCLK1	4.9	nM
10024-999-3	NVP-TAE684	200110	DCAMKL2	16.0	nM
10024-999-3	NVP-TAE684	200111	DCAMKL3	14.0	nM
10024-999-3	NVP-TAE684	200112	DDR1	140.0	nM
10024-999-3	NVP-TAE684	200113	DDR2	4100.0	nM
10024-999-3	NVP-TAE684	200114	M3K12	42.0	nM
10024-999-3	NVP-TAE684	200115	DMPK	2100.0	nM
10024-999-3	NVP-TAE684	200116	DMPK2	9500.0	nM
10024-999-3	NVP-TAE684	200117	DRAK1	2900.0	nM
10024-999-3	NVP-TAE684	200118	DRAK2	7100.0	nM
10024-999-3	NVP-TAE684	200119	DYRK1A	2900.0	nM
10024-999-3	NVP-TAE684	200120	DYRK1B	4500.0	nM
10024-999-3	NVP-TAE684	200121	DYRK2		nM
10024-999-3	NVP-TAE684	200122	EGFR	180.0	nM
10024-999-3	NVP-TAE684	200123	EGFR(E746-A750del)	81.0	nM
10024-999-3	NVP-TAE684	200124	EGFR(G719C)	2000.0	nM
10024-999-3	NVP-TAE684	200125	EGFR(G719S)	1600.0	nM
10024-999-3	NVP-TAE684	200126	EGFR(L747-E749del, A750P)	72.0	nM
10024-999-3	NVP-TAE684	200127	EGFR(L747-S752del, P753S)	110.0	nM
10024-999-3	NVP-TAE684	200128	EGFR(L747-T751del,Sins)	79.0	nM
10024-999-3	NVP-TAE684	200129	EGFR(L858R)	46.0	nM
10024-999-3	NVP-TAE684	200130	EGFR(L858R,T790M)	3.4	nM
10024-999-3	NVP-TAE684	200131	EGFR(L861Q)	98.0	nM
10024-999-3	NVP-TAE684	200132	EGFR(S752-I759del)	400.0	nM
10024-999-3	NVP-TAE684	200133	EGFR(T790M)	7.1	nM
10024-999-3	NVP-TAE684	200134	EIF2AK1		nM
10024-999-3	NVP-TAE684	200135	EPHA1	39.0	nM
10024-999-3	NVP-TAE684	200136	EPHA2	890.0	nM
10024-999-3	NVP-TAE684	200137	EPHA3	4000.0	nM
10024-999-3	NVP-TAE684	200138	EPHA4	910.0	nM
10024-999-3	NVP-TAE684	200139	EPHA5	3700.0	nM
10024-999-3	NVP-TAE684	200140	EPHA6	120.0	nM
10024-999-3	NVP-TAE684	200141	EPHA7	200.0	nM
10024-999-3	NVP-TAE684	200142	EPHA8		nM
10024-999-3	NVP-TAE684	200143	EPHB1	340.0	nM
10024-999-3	NVP-TAE684	200144	EPHB2	1500.0	nM
10024-999-3	NVP-TAE684	200145	EPHB3	1900.0	nM
10024-999-3	NVP-TAE684	200146	EPHB4	750.0	nM
10024-999-3	NVP-TAE684	200147	EPHB6	350.0	nM
10024-999-3	NVP-TAE684	200148	ERBB2	540.0	nM
10024-999-3	NVP-TAE684	200149	ERBB3		nM
10024-999-3	NVP-TAE684	200150	ERBB4	280.0	nM
10024-999-3	NVP-TAE684	200151	MK03	430.0	nM
10024-999-3	NVP-TAE684	200152	MK01	300.0	nM
10024-999-3	NVP-TAE684	200153	ERK3		nM
10024-999-3	NVP-TAE684	200154	ERK4		nM
10024-999-3	NVP-TAE684	200155	ERK5	48.0	nM
10024-999-3	NVP-TAE684	200156	ERK8	210.0	nM
10024-999-3	NVP-TAE684	200157	ERN1	180.0	nM
10024-999-3	NVP-TAE684	200158	FAK1	1.1	nM
10024-999-3	NVP-TAE684	200159	FER	1.4	nM
10024-999-3	NVP-TAE684	200160	FES	4.8	nM
10024-999-3	NVP-TAE684	200161	FGFR1	47.0	nM
10024-999-3	NVP-TAE684	200162	FGFR2	250.0	nM
10024-999-3	NVP-TAE684	200163	FGFR3	95.0	nM
10024-999-3	NVP-TAE684	200164	FGFR3(G697C)	120.0	nM
10024-999-3	NVP-TAE684	200165	FGFR4	110.0	nM
10024-999-3	NVP-TAE684	200166	FGR	120.0	nM
10024-999-3	NVP-TAE684	200167	VGFR1	550.0	nM
10024-999-3	NVP-TAE684	200168	FLT3	15.0	nM
10024-999-3	NVP-TAE684	200169	FLT3(D835H)	4.9	nM
10024-999-3	NVP-TAE684	200170	FLT3(D835Y)	2.0	nM
10024-999-3	NVP-TAE684	200171	FLT3(ITD)	8.6	nM
10024-999-3	NVP-TAE684	200172	FLT3(K663Q)	8.2	nM
10024-999-3	NVP-TAE684	200173	FLT3(N841I)	11.0	nM
10024-999-3	NVP-TAE684	200174	FLT3(R834Q)	34.0	nM
10024-999-3	NVP-TAE684	200175	FLT4	170.0	nM
10024-999-3	NVP-TAE684	200176	FRK	27.0	nM
10024-999-3	NVP-TAE684	200177	FYN	1400.0	nM
10024-999-3	NVP-TAE684	200178	GAK	5.3	nM
10024-999-3	NVP-TAE684	200179	GCN2(Kin.Dom.2,S808G)	1100.0	nM
10024-999-3	NVP-TAE684	200180	GRK1	410.0	nM
10024-999-3	NVP-TAE684	200181	GRK4	3500.0	nM
10024-999-3	NVP-TAE684	200182	GRK7	360.0	nM
10024-999-3	NVP-TAE684	200183	GSK3A		nM
10024-999-3	NVP-TAE684	200184	GSK3B		nM
10024-999-3	NVP-TAE684	200185	HCK	410.0	nM
10024-999-3	NVP-TAE684	200186	HIPK1	4400.0	nM
10024-999-3	NVP-TAE684	200187	HIPK2	4400.0	nM
10024-999-3	NVP-TAE684	200188	HIPK3	6900.0	nM
10024-999-3	NVP-TAE684	200189	HIPK4	350.0	nM
10024-999-3	NVP-TAE684	200190	M4K1	140.0	nM
10024-999-3	NVP-TAE684	200191	HUNK	350.0	nM
10024-999-3	NVP-TAE684	200192	ICK	4000.0	nM
10024-999-3	NVP-TAE684	200193	IGF1R	2.7	nM
10024-999-3	NVP-TAE684	200194	IKKA		nM
10024-999-3	NVP-TAE684	200195	IKKB		nM
10024-999-3	NVP-TAE684	200196	IKKE	1100.0	nM
10024-999-3	NVP-TAE684	200197	INSR	2.4	nM
10024-999-3	NVP-TAE684	200198	INSRR	6.2	nM
10024-999-3	NVP-TAE684	200199	IRAK1	45.0	nM
10024-999-3	NVP-TAE684	200200	IRAK3	160.0	nM
10024-999-3	NVP-TAE684	200201	IRAK4	77.0	nM
10024-999-3	NVP-TAE684	200202	ITK	34.0	nM
10024-999-3	NVP-TAE684	200203	JAK1(JH1domain-catalytic)	410.0	nM
10024-999-3	NVP-TAE684	200204	JAK1(JH2domain-pseudokinase)	300.0	nM
10024-999-3	NVP-TAE684	200207	JAK2(JH1domain-catalytic)	16.0	nM
10024-999-3	NVP-TAE684	200209	JAK3(JH1domain-catalytic)	17.0	nM
10024-999-3	NVP-TAE684	200211	JNK1	160.0	nM
10024-999-3	NVP-TAE684	200212	MK09	280.0	nM
10024-999-3	NVP-TAE684	200213	JNK3	67.0	nM
10024-999-3	NVP-TAE684	200214	KIT	110.0	nM
10024-999-3	NVP-TAE684	200215	KIT(A829P)	220.0	nM
10024-999-3	NVP-TAE684	200216	KIT(D816H)	140.0	nM
10024-999-3	NVP-TAE684	200217	KIT(D816V)	26.0	nM
10024-999-3	NVP-TAE684	200218	KIT(L576P)	49.0	nM
10024-999-3	NVP-TAE684	200219	KIT(V559D)	81.0	nM
10024-999-3	NVP-TAE684	200220	KIT(V559D,T670I)	130.0	nM
10024-999-3	NVP-TAE684	200221	KIT(V559D,V654A)	1200.0	nM
10024-999-3	NVP-TAE684	200222	LATS1	1600.0	nM
10024-999-3	NVP-TAE684	200223	LATS2	2000.0	nM
10024-999-3	NVP-TAE684	200224	LCK	49.0	nM
10024-999-3	NVP-TAE684	200225	LIMK1	1100.0	nM
10024-999-3	NVP-TAE684	200226	LIMK2	1100.0	nM
10024-999-3	NVP-TAE684	200227	LKB1		nM
10024-999-3	NVP-TAE684	200228	LOK	82.0	nM
10024-999-3	NVP-TAE684	200229	LRRK2	1.4	nM
10024-999-3	NVP-TAE684	200230	LRRK2(G2019S)	0.9	nM
10024-999-3	NVP-TAE684	200231	LTK	1.0	nM
10024-999-3	NVP-TAE684	200232	LYN	280.0	nM
10024-999-3	NVP-TAE684	200233	M3K13	57.0	nM
10024-999-3	NVP-TAE684	200234	MAK		nM
10024-999-3	NVP-TAE684	200235	MAP3K1	4300.0	nM
10024-999-3	NVP-TAE684	200236	MAP3K15	800.0	nM
10024-999-3	NVP-TAE684	200237	M3K2	110.0	nM
10024-999-3	NVP-TAE684	200238	MAP3K3	320.0	nM
10024-999-3	NVP-TAE684	200239	MAP3K4	2000.0	nM
10024-999-3	NVP-TAE684	200240	MAP4K2	190.0	nM
10024-999-3	NVP-TAE684	200241	M4K3	65.0	nM
10024-999-3	NVP-TAE684	200242	MAP4K4	970.0	nM
10024-999-3	NVP-TAE684	200243	MAP4K5	190.0	nM
10024-999-3	NVP-TAE684	200244	MAPKAPK2		nM
10024-999-3	NVP-TAE684	200245	MAPKAPK5		nM
10024-999-3	NVP-TAE684	200246	MARK1	31.0	nM
10024-999-3	NVP-TAE684	200247	MARK2	44.0	nM
10024-999-3	NVP-TAE684	200248	MARK3	12.0	nM
10024-999-3	NVP-TAE684	200249	MARK4	12.0	nM
10024-999-3	NVP-TAE684	200250	MAST1	3300.0	nM
10024-999-3	NVP-TAE684	200251	MP2K1	550.0	nM
10024-999-3	NVP-TAE684	200252	MP2K2	630.0	nM
10024-999-3	NVP-TAE684	200253	MP2K3	170.0	nM
10024-999-3	NVP-TAE684	200254	MP2K4	150.0	nM
10024-999-3	NVP-TAE684	200255	MP2K5	200.0	nM
10024-999-3	NVP-TAE684	200256	MP2K6	2000.0	nM
10024-999-3	NVP-TAE684	200257	MELK	99.0	nM
10024-999-3	NVP-TAE684	200258	MERTK	19.0	nM
10024-999-3	NVP-TAE684	200259	MET	170.0	nM
10024-999-3	NVP-TAE684	200260	MET(M1250T)	64.0	nM
10024-999-3	NVP-TAE684	200261	MET(Y1235D)	180.0	nM
10024-999-3	NVP-TAE684	200262	MINK	330.0	nM
10024-999-3	NVP-TAE684	200263	MP2K7		nM
10024-999-3	NVP-TAE684	200264	MKNK1		nM
10024-999-3	NVP-TAE684	200265	MKNK2	44.0	nM
10024-999-3	NVP-TAE684	200266	MLCK		nM
10024-999-3	NVP-TAE684	200267	MLK1	410.0	nM
10024-999-3	NVP-TAE684	200268	MLK2	1100.0	nM
10024-999-3	NVP-TAE684	200269	MLK3	420.0	nM
10024-999-3	NVP-TAE684	200270	MRCKA		nM
10024-999-3	NVP-TAE684	200271	MRCKB	4800.0	nM
10024-999-3	NVP-TAE684	200272	MST1	330.0	nM
10024-999-3	NVP-TAE684	200273	MST1R	610.0	nM
10024-999-3	NVP-TAE684	200274	MST2	310.0	nM
10024-999-3	NVP-TAE684	200275	MST3	2900.0	nM
10024-999-3	NVP-TAE684	200276	MST4	510.0	nM
10024-999-3	NVP-TAE684	200277	MTOR		nM
10024-999-3	NVP-TAE684	200278	MUSK	260.0	nM
10024-999-3	NVP-TAE684	200279	MYLK	220.0	nM
10024-999-3	NVP-TAE684	200280	MYLK2		nM
10024-999-3	NVP-TAE684	200281	MYLK4		nM
10024-999-3	NVP-TAE684	200282	MYO3A	67.0	nM
10024-999-3	NVP-TAE684	200283	MYO3B	81.0	nM
10024-999-3	NVP-TAE684	200284	NDR1	440.0	nM
10024-999-3	NVP-TAE684	200285	NDR2	580.0	nM
10024-999-3	NVP-TAE684	200286	NEK1		nM
10024-999-3	NVP-TAE684	200287	NEK11		nM
10024-999-3	NVP-TAE684	200288	NEK2	1800.0	nM
10024-999-3	NVP-TAE684	200289	NEK3	8800.0	nM
10024-999-3	NVP-TAE684	200290	NEK4		nM
10024-999-3	NVP-TAE684	200291	NEK5		nM
10024-999-3	NVP-TAE684	200292	NEK6	1300.0	nM
10024-999-3	NVP-TAE684	200293	NEK7	2300.0	nM
10024-999-3	NVP-TAE684	200294	NEK9	800.0	nM
10024-999-3	NVP-TAE684	200295	NIM1	2600.0	nM
10024-999-3	NVP-TAE684	200296	NLK		nM
10024-999-3	NVP-TAE684	200297	OSR1	48.0	nM
10024-999-3	NVP-TAE684	200298	MK14		nM
10024-999-3	NVP-TAE684	200299	MK11		nM
10024-999-3	NVP-TAE684	200300	MK13		nM
10024-999-3	NVP-TAE684	200301	MK12	9400.0	nM
10024-999-3	NVP-TAE684	200302	PAK1	650.0	nM
10024-999-3	NVP-TAE684	200303	PAK2	5800.0	nM
10024-999-3	NVP-TAE684	200304	PAK3	29.0	nM
10024-999-3	NVP-TAE684	200305	PAK4	2000.0	nM
10024-999-3	NVP-TAE684	200306	PAK6	3500.0	nM
10024-999-3	NVP-TAE684	200307	PAK7	390.0	nM
10024-999-3	NVP-TAE684	200309	CDK16	560.0	nM
10024-999-3	NVP-TAE684	200310	PCTK2	810.0	nM
10024-999-3	NVP-TAE684	200311	PCTK3		nM
10024-999-3	NVP-TAE684	200312	PGFRA	840.0	nM
10024-999-3	NVP-TAE684	200313	PGFRB	150.0	nM
10024-999-3	NVP-TAE684	200314	PDPK1		nM
10024-999-3	NVP-TAE684	200315	PFCDPK1(P.falciparum)	710.0	nM
10024-999-3	NVP-TAE684	200316	PFPK5(P.falciparum)		nM
10024-999-3	NVP-TAE684	200317	CDK15	2100.0	nM
10024-999-3	NVP-TAE684	200318	CDK14		nM
10024-999-3	NVP-TAE684	200319	PHKG1	17.0	nM
10024-999-3	NVP-TAE684	200320	PHKG2	13.0	nM
10024-999-3	NVP-TAE684	200321	PIK3C2B		nM
10024-999-3	NVP-TAE684	200322	PIK3C2G		nM
10024-999-3	NVP-TAE684	200323	PIK3CA		nM
10024-999-3	NVP-TAE684	200324	PIK3CA(C420R)		nM
10024-999-3	NVP-TAE684	200325	PIK3CA(E542K)		nM
10024-999-3	NVP-TAE684	200326	PIK3CA(E545A)		nM
10024-999-3	NVP-TAE684	200327	PIK3CA(E545K)		nM
10024-999-3	NVP-TAE684	200328	PIK3CA(H1047L)		nM
10024-999-3	NVP-TAE684	200329	PIK3CA(H1047Y)		nM
10024-999-3	NVP-TAE684	200330	PIK3CA(I800L)		nM
10024-999-3	NVP-TAE684	200331	PIK3CA(M1043I)		nM
10024-999-3	NVP-TAE684	200332	PIK3CA(Q546K)		nM
10024-999-3	NVP-TAE684	200333	PIK3CB		nM
10024-999-3	NVP-TAE684	200334	PIK3CD		nM
10024-999-3	NVP-TAE684	200335	PIK3CG		nM
10024-999-3	NVP-TAE684	200336	PIK4CB	780.0	nM
10024-999-3	NVP-TAE684	200337	PIM1		nM
10024-999-3	NVP-TAE684	200338	PIM2		nM
10024-999-3	NVP-TAE684	200339	PIM3		nM
10024-999-3	NVP-TAE684	200340	PIP5K1A	9700.0	nM
10024-999-3	NVP-TAE684	200341	PIP5K1C		nM
10024-999-3	NVP-TAE684	200342	PIP5K2B		nM
10024-999-3	NVP-TAE684	200343	PI42C	2300.0	nM
10024-999-3	NVP-TAE684	200344	PKAC-alpha	4000.0	nM
10024-999-3	NVP-TAE684	200345	PKAC-beta	4100.0	nM
10024-999-3	NVP-TAE684	200346	PKMYT1		nM
10024-999-3	NVP-TAE684	200347	PKN1	340.0	nM
10024-999-3	NVP-TAE684	200348	PKN2	680.0	nM
10024-999-3	NVP-TAE684	200349	PKNB(M.tuberculosis)	1200.0	nM
10024-999-3	NVP-TAE684	200350	PLK1	20.0	nM
10024-999-3	NVP-TAE684	200351	PLK2	1200.0	nM
10024-999-3	NVP-TAE684	200352	PLK3	210.0	nM
10024-999-3	NVP-TAE684	200353	PLK4	0.9	nM
10024-999-3	NVP-TAE684	200354	KPCD	3500.0	nM
10024-999-3	NVP-TAE684	200355	KPCE	2000.0	nM
10024-999-3	NVP-TAE684	200356	KPCL		nM
10024-999-3	NVP-TAE684	200357	KPCI		nM
10024-999-3	NVP-TAE684	200358	KPCT	1500.0	nM
10024-999-3	NVP-TAE684	200359	KPCD1	80.0	nM
10024-999-3	NVP-TAE684	200360	KPCD2	160.0	nM
10024-999-3	NVP-TAE684	200361	KPCD3	90.0	nM
10024-999-3	NVP-TAE684	200362	KGP1	430.0	nM
10024-999-3	NVP-TAE684	200363	KGP2	240.0	nM
10024-999-3	NVP-TAE684	200364	PRKR		nM
10024-999-3	NVP-TAE684	200365	PRKX	5800.0	nM
10024-999-3	NVP-TAE684	200366	PRP4	7600.0	nM
10024-999-3	NVP-TAE684	200367	FAK2	1.1	nM
10024-999-3	NVP-TAE684	200368	SIK3	1300.0	nM
10024-999-3	NVP-TAE684	200369	RAF1		nM
10024-999-3	NVP-TAE684	200370	RET	150.0	nM
10024-999-3	NVP-TAE684	200371	RET(M918T)	140.0	nM
10024-999-3	NVP-TAE684	200372	RET(V804L)	120.0	nM
10024-999-3	NVP-TAE684	200373	RET(V804M)	140.0	nM
10024-999-3	NVP-TAE684	200374	RIOK1		nM
10024-999-3	NVP-TAE684	200375	RIOK2		nM
10024-999-3	NVP-TAE684	200376	RIOK3	3500.0	nM
10024-999-3	NVP-TAE684	200377	RIPK1		nM
10024-999-3	NVP-TAE684	200378	RIPK2	9600.0	nM
10024-999-3	NVP-TAE684	200379	RIPK4	3200.0	nM
10024-999-3	NVP-TAE684	200380	RIPK5	57.0	nM
10024-999-3	NVP-TAE684	200381	ROCK1	37.0	nM
10024-999-3	NVP-TAE684	200382	ROCK2	130.0	nM
10024-999-3	NVP-TAE684	200383	ROS1	0.5	nM
10024-999-3	NVP-TAE684	200390	RPS6KA4(Kin.Dom.1-N-terminal)	2500.0	nM
10024-999-3	NVP-TAE684	200392	RPS6KA4(Kin.Dom.2-C-terminal)		nM
10024-999-3	NVP-TAE684	200394	RPS6KA5(Kin.Dom.1-N-terminal)		nM
10024-999-3	NVP-TAE684	200396	RPS6KA5(Kin.Dom.2-C-terminal)		nM
10024-999-3	NVP-TAE684	200399	RSK1(Kin.Dom.1-N-terminal)	160.0	nM
10024-999-3	NVP-TAE684	200400	RSK1(Kin.Dom.2-C-terminal)	650.0	nM
10024-999-3	NVP-TAE684	200401	RSK2(Kin.Dom.1-N-terminal)	17.0	nM
10024-999-3	NVP-TAE684	200402	RSK3(Kin.Dom.1-N-terminal)	33.0	nM
10024-999-3	NVP-TAE684	200403	RSK3(Kin.Dom.2-C-terminal)	160.0	nM
10024-999-3	NVP-TAE684	200404	RSK4(Kin.Dom.1-N-terminal)	27.0	nM
10024-999-3	NVP-TAE684	200405	RSK4(Kin.Dom.2-C-terminal)	160.0	nM
10024-999-3	NVP-TAE684	200406	S6K1	2700.0	nM
10024-999-3	NVP-TAE684	200407	SBK1	21.0	nM
10024-999-3	NVP-TAE684	200408	SgK110	54.0	nM
10024-999-3	NVP-TAE684	200409	SGK3		nM
10024-999-3	NVP-TAE684	200410	SIK1	15.0	nM
10024-999-3	NVP-TAE684	200411	SIK2	17.0	nM
10024-999-3	NVP-TAE684	200412	SLK	21.0	nM
10024-999-3	NVP-TAE684	200413	SNARK	1.2	nM
10024-999-3	NVP-TAE684	200414	SNRK	300.0	nM
10024-999-3	NVP-TAE684	200415	SRC	280.0	nM
10024-999-3	NVP-TAE684	200416	SRMS	160.0	nM
10024-999-3	NVP-TAE684	200417	SRPK1	4800.0	nM
10024-999-3	NVP-TAE684	200418	SRPK2		nM
10024-999-3	NVP-TAE684	200419	SRPK3	2900.0	nM
10024-999-3	NVP-TAE684	200420	STK16	800.0	nM
10024-999-3	NVP-TAE684	200421	STK33	3.2	nM
10024-999-3	NVP-TAE684	200422	STK35	260.0	nM
10024-999-3	NVP-TAE684	200423	STK36	1400.0	nM
10024-999-3	NVP-TAE684	200424	STK39	150.0	nM
10024-999-3	NVP-TAE684	200425	SYK	1300.0	nM
10024-999-3	NVP-TAE684	200426	TAK1	160.0	nM
10024-999-3	NVP-TAE684	200427	TAOK1	25.0	nM
10024-999-3	NVP-TAE684	200428	TAOK2	740.0	nM
10024-999-3	NVP-TAE684	200429	TAOK3	44.0	nM
10024-999-3	NVP-TAE684	200430	TBK1	470.0	nM
10024-999-3	NVP-TAE684	200431	TEC	180.0	nM
10024-999-3	NVP-TAE684	200432	TESK1		nM
10024-999-3	NVP-TAE684	200433	TGFBR1	190.0	nM
10024-999-3	NVP-TAE684	200434	TGFBR2	250.0	nM
10024-999-3	NVP-TAE684	200435	TIE1	15.0	nM
10024-999-3	NVP-TAE684	200436	TIE2	46.0	nM
10024-999-3	NVP-TAE684	200437	TLK1		nM
10024-999-3	NVP-TAE684	200438	TLK2		nM
10024-999-3	NVP-TAE684	200439	TNIK	1200.0	nM
10024-999-3	NVP-TAE684	200440	TNK1	1.8	nM
10024-999-3	NVP-TAE684	200441	TNK2	2.0	nM
10024-999-3	NVP-TAE684	200442	TNNI3K	2000.0	nM
10024-999-3	NVP-TAE684	200443	TRKA	460.0	nM
10024-999-3	NVP-TAE684	200444	TRKB	130.0	nM
10024-999-3	NVP-TAE684	200445	TRKC		nM
10024-999-3	NVP-TAE684	200446	TRPM6		nM
10024-999-3	NVP-TAE684	200447	TSSK1	25.0	nM
10024-999-3	NVP-TAE684	200448	TTK	50.0	nM
10024-999-3	NVP-TAE684	200449	TXK	480.0	nM
10024-999-3	NVP-TAE684	200450	TYK2(JH1domain-catalytic)	77.0	nM
10024-999-3	NVP-TAE684	200451	TYK2(JH2domain-pseudokinase)	1900.0	nM
10024-999-3	NVP-TAE684	200454	TYRO3	7200.0	nM
10024-999-3	NVP-TAE684	200455	ULK1	0.8	nM
10024-999-3	NVP-TAE684	200456	ULK2	1.8	nM
10024-999-3	NVP-TAE684	200457	ULK3	11.0	nM
10024-999-3	NVP-TAE684	200458	VGFR2	940.0	nM
10024-999-3	NVP-TAE684	200459	VRK2		nM
10024-999-3	NVP-TAE684	200460	WEE1	3000.0	nM
10024-999-3	NVP-TAE684	200461	WEE2		nM
10024-999-3	NVP-TAE684	200462	YANK1	13.0	nM
10024-999-3	NVP-TAE684	200463	YANK2	24.0	nM
10024-999-3	NVP-TAE684	200464	YANK3	55.0	nM
10024-999-3	NVP-TAE684	200465	YES	23.0	nM
10024-999-3	NVP-TAE684	200466	YSK1	7700.0	nM
10024-999-3	NVP-TAE684	200467	YSK4	2800.0	nM
10024-999-3	NVP-TAE684	200468	MLTK		nM
10024-999-3	NVP-TAE684	200469	ZAP70	1600.0	nM
