Small Molecule HMS LINCS ID	Small Molecule Name	Protein HMS LINCS ID	Protein Name	Kd	Conc unit
10226-999-4	Tofacitinib	200001	AAK1		nM
10226-999-4	Tofacitinib	200004	ABL1(E255K)-phosphorylated		nM
10226-999-4	Tofacitinib	200006	ABL1(F317I)-nonphosphorylated		nM
10226-999-4	Tofacitinib	200007	ABL1(F317I)-phosphorylated		nM
10226-999-4	Tofacitinib	200009	ABL1(F317L)-nonphosphorylated		nM
10226-999-4	Tofacitinib	200010	ABL1(F317L)-phosphorylated		nM
10226-999-4	Tofacitinib	200012	ABL1(H396P)-nonphosphorylated	4500.0	nM
10226-999-4	Tofacitinib	200013	ABL1(H396P)-phosphorylated	6700.0	nM
10226-999-4	Tofacitinib	200015	ABL1(M351T)-phosphorylated		nM
10226-999-4	Tofacitinib	200017	ABL1(Q252H)-nonphosphorylated		nM
10226-999-4	Tofacitinib	200018	ABL1(Q252H)-phosphorylated		nM
10226-999-4	Tofacitinib	200020	ABL1(T315I)-nonphosphorylated		nM
10226-999-4	Tofacitinib	200021	ABL1(T315I)-phosphorylated	2200.0	nM
10226-999-4	Tofacitinib	200023	ABL1(Y253F)-phosphorylated		nM
10226-999-4	Tofacitinib	200024	ABL1-nonphosphorylated		nM
10226-999-4	Tofacitinib	200025	ABL1-phosphorylated		nM
10226-999-4	Tofacitinib	200026	ABL2		nM
10226-999-4	Tofacitinib	200027	ACVR1		nM
10226-999-4	Tofacitinib	200028	ACVR1B		nM
10226-999-4	Tofacitinib	200029	ACVR2A		nM
10226-999-4	Tofacitinib	200030	ACVR2B		nM
10226-999-4	Tofacitinib	200031	ACVRL1		nM
10226-999-4	Tofacitinib	200032	ADCK3		nM
10226-999-4	Tofacitinib	200033	ADCK4		nM
10226-999-4	Tofacitinib	200034	AKT1		nM
10226-999-4	Tofacitinib	200035	AKT2		nM
10226-999-4	Tofacitinib	200036	AKT3		nM
10226-999-4	Tofacitinib	200037	ALK		nM
10226-999-4	Tofacitinib	200038	AMPK-alpha1		nM
10226-999-4	Tofacitinib	200039	AMPK-alpha2		nM
10226-999-4	Tofacitinib	200040	ANKK1		nM
10226-999-4	Tofacitinib	200041	NUAK1		nM
10226-999-4	Tofacitinib	200042	M3K5		nM
10226-999-4	Tofacitinib	200043	M3K6		nM
10226-999-4	Tofacitinib	200044	AURKA		nM
10226-999-4	Tofacitinib	200045	AURKB		nM
10226-999-4	Tofacitinib	200046	AURKC		nM
10226-999-4	Tofacitinib	200047	AXL		nM
10226-999-4	Tofacitinib	200048	BIKE	7100.0	nM
10226-999-4	Tofacitinib	200049	BLK		nM
10226-999-4	Tofacitinib	200050	BMPR1A		nM
10226-999-4	Tofacitinib	200051	BMPR1B		nM
10226-999-4	Tofacitinib	200052	BMPR2		nM
10226-999-4	Tofacitinib	200053	BMX		nM
10226-999-4	Tofacitinib	200054	BRAF		nM
10226-999-4	Tofacitinib	200055	BRAF(V600E)		nM
10226-999-4	Tofacitinib	200056	PTK6		nM
10226-999-4	Tofacitinib	200057	BRSK1		nM
10226-999-4	Tofacitinib	200058	BRSK2		nM
10226-999-4	Tofacitinib	200059	BTK		nM
10226-999-4	Tofacitinib	200060	CAMK1	1200.0	nM
10226-999-4	Tofacitinib	200061	CAMK1D	1600.0	nM
10226-999-4	Tofacitinib	200062	CAMK1G		nM
10226-999-4	Tofacitinib	200063	CAMK2A	3500.0	nM
10226-999-4	Tofacitinib	200064	CAMK2B		nM
10226-999-4	Tofacitinib	200065	KCC2D	2700.0	nM
10226-999-4	Tofacitinib	200066	CAMK2G		nM
10226-999-4	Tofacitinib	200067	KCC4		nM
10226-999-4	Tofacitinib	200068	KKCC1		nM
10226-999-4	Tofacitinib	200069	CAMKK2		nM
10226-999-4	Tofacitinib	200070	CASK		nM
10226-999-4	Tofacitinib	200071	CDC2L1		nM
10226-999-4	Tofacitinib	200072	CDC2L2		nM
10226-999-4	Tofacitinib	200073	CDC2L5		nM
10226-999-4	Tofacitinib	200074	CDK11		nM
10226-999-4	Tofacitinib	200075	CDK2		nM
10226-999-4	Tofacitinib	200076	CDK3		nM
10226-999-4	Tofacitinib	200077	CDK4-cyclinD1		nM
10226-999-4	Tofacitinib	200078	CDK4-cyclinD3		nM
10226-999-4	Tofacitinib	200079	CDK5		nM
10226-999-4	Tofacitinib	200080	CDK7		nM
10226-999-4	Tofacitinib	200081	CDK8		nM
10226-999-4	Tofacitinib	200082	CDK9		nM
10226-999-4	Tofacitinib	200083	CDKL1		nM
10226-999-4	Tofacitinib	200084	CDKL2		nM
10226-999-4	Tofacitinib	200085	CDKL3		nM
10226-999-4	Tofacitinib	200086	CDKL5		nM
10226-999-4	Tofacitinib	200087	CHEK1		nM
10226-999-4	Tofacitinib	200088	CHK2		nM
10226-999-4	Tofacitinib	200089	CIT		nM
10226-999-4	Tofacitinib	200090	CLK1		nM
10226-999-4	Tofacitinib	200091	CLK2		nM
10226-999-4	Tofacitinib	200092	CLK3		nM
10226-999-4	Tofacitinib	200093	CLK4		nM
10226-999-4	Tofacitinib	200094	CSF1R		nM
10226-999-4	Tofacitinib	200095	CSK		nM
10226-999-4	Tofacitinib	200096	CSNK1A1		nM
10226-999-4	Tofacitinib	200097	CSNK1A1L		nM
10226-999-4	Tofacitinib	200098	CSNK1D		nM
10226-999-4	Tofacitinib	200099	CSNK1E		nM
10226-999-4	Tofacitinib	200100	KC1G1		nM
10226-999-4	Tofacitinib	200101	KC1G2		nM
10226-999-4	Tofacitinib	200102	CSNK1G3		nM
10226-999-4	Tofacitinib	200103	CSNK2A1		nM
10226-999-4	Tofacitinib	200104	CSNK2A2		nM
10226-999-4	Tofacitinib	200105	CTK		nM
10226-999-4	Tofacitinib	200106	DAPK1		nM
10226-999-4	Tofacitinib	200107	DAPK2		nM
10226-999-4	Tofacitinib	200108	DAPK3		nM
10226-999-4	Tofacitinib	200109	DCLK1	6700.0	nM
10226-999-4	Tofacitinib	200110	DCAMKL2		nM
10226-999-4	Tofacitinib	200111	DCAMKL3	12.0	nM
10226-999-4	Tofacitinib	200112	DDR1		nM
10226-999-4	Tofacitinib	200113	DDR2		nM
10226-999-4	Tofacitinib	200114	M3K12		nM
10226-999-4	Tofacitinib	200115	DMPK	1200.0	nM
10226-999-4	Tofacitinib	200116	DMPK2		nM
10226-999-4	Tofacitinib	200117	DRAK1		nM
10226-999-4	Tofacitinib	200118	DRAK2		nM
10226-999-4	Tofacitinib	200119	DYRK1A		nM
10226-999-4	Tofacitinib	200120	DYRK1B		nM
10226-999-4	Tofacitinib	200121	DYRK2		nM
10226-999-4	Tofacitinib	200122	EGFR		nM
10226-999-4	Tofacitinib	200123	EGFR(E746-A750del)		nM
10226-999-4	Tofacitinib	200124	EGFR(G719C)		nM
10226-999-4	Tofacitinib	200125	EGFR(G719S)		nM
10226-999-4	Tofacitinib	200126	EGFR(L747-E749del, A750P)		nM
10226-999-4	Tofacitinib	200127	EGFR(L747-S752del, P753S)		nM
10226-999-4	Tofacitinib	200128	EGFR(L747-T751del,Sins)		nM
10226-999-4	Tofacitinib	200129	EGFR(L858R)		nM
10226-999-4	Tofacitinib	200130	EGFR(L858R,T790M)		nM
10226-999-4	Tofacitinib	200131	EGFR(L861Q)		nM
10226-999-4	Tofacitinib	200132	EGFR(S752-I759del)		nM
10226-999-4	Tofacitinib	200133	EGFR(T790M)		nM
10226-999-4	Tofacitinib	200134	EIF2AK1		nM
10226-999-4	Tofacitinib	200135	EPHA1		nM
10226-999-4	Tofacitinib	200136	EPHA2		nM
10226-999-4	Tofacitinib	200137	EPHA3		nM
10226-999-4	Tofacitinib	200138	EPHA4		nM
10226-999-4	Tofacitinib	200139	EPHA5		nM
10226-999-4	Tofacitinib	200140	EPHA6		nM
10226-999-4	Tofacitinib	200141	EPHA7		nM
10226-999-4	Tofacitinib	200142	EPHA8		nM
10226-999-4	Tofacitinib	200143	EPHB1		nM
10226-999-4	Tofacitinib	200144	EPHB2		nM
10226-999-4	Tofacitinib	200145	EPHB3		nM
10226-999-4	Tofacitinib	200146	EPHB4		nM
10226-999-4	Tofacitinib	200147	EPHB6		nM
10226-999-4	Tofacitinib	200148	ERBB2		nM
10226-999-4	Tofacitinib	200149	ERBB3		nM
10226-999-4	Tofacitinib	200150	ERBB4		nM
10226-999-4	Tofacitinib	200151	MK03		nM
10226-999-4	Tofacitinib	200152	MK01		nM
10226-999-4	Tofacitinib	200153	ERK3		nM
10226-999-4	Tofacitinib	200154	ERK4		nM
10226-999-4	Tofacitinib	200155	ERK5		nM
10226-999-4	Tofacitinib	200156	ERK8		nM
10226-999-4	Tofacitinib	200157	ERN1		nM
10226-999-4	Tofacitinib	200158	FAK1		nM
10226-999-4	Tofacitinib	200159	FER		nM
10226-999-4	Tofacitinib	200160	FES		nM
10226-999-4	Tofacitinib	200161	FGFR1		nM
10226-999-4	Tofacitinib	200162	FGFR2		nM
10226-999-4	Tofacitinib	200163	FGFR3		nM
10226-999-4	Tofacitinib	200164	FGFR3(G697C)		nM
10226-999-4	Tofacitinib	200165	FGFR4		nM
10226-999-4	Tofacitinib	200166	FGR		nM
10226-999-4	Tofacitinib	200167	VGFR1		nM
10226-999-4	Tofacitinib	200168	FLT3		nM
10226-999-4	Tofacitinib	200169	FLT3(D835H)		nM
10226-999-4	Tofacitinib	200170	FLT3(D835Y)		nM
10226-999-4	Tofacitinib	200171	FLT3(ITD)		nM
10226-999-4	Tofacitinib	200172	FLT3(K663Q)		nM
10226-999-4	Tofacitinib	200173	FLT3(N841I)		nM
10226-999-4	Tofacitinib	200174	FLT3(R834Q)		nM
10226-999-4	Tofacitinib	200175	FLT4		nM
10226-999-4	Tofacitinib	200176	FRK		nM
10226-999-4	Tofacitinib	200177	FYN	1100.0	nM
10226-999-4	Tofacitinib	200178	GAK		nM
10226-999-4	Tofacitinib	200179	GCN2(Kin.Dom.2,S808G)		nM
10226-999-4	Tofacitinib	200180	GRK1		nM
10226-999-4	Tofacitinib	200181	GRK4		nM
10226-999-4	Tofacitinib	200182	GRK7	4300.0	nM
10226-999-4	Tofacitinib	200183	GSK3A		nM
10226-999-4	Tofacitinib	200184	GSK3B		nM
10226-999-4	Tofacitinib	200185	HCK		nM
10226-999-4	Tofacitinib	200186	HIPK1		nM
10226-999-4	Tofacitinib	200187	HIPK2		nM
10226-999-4	Tofacitinib	200188	HIPK3		nM
10226-999-4	Tofacitinib	200189	HIPK4		nM
10226-999-4	Tofacitinib	200190	M4K1		nM
10226-999-4	Tofacitinib	200191	HUNK		nM
10226-999-4	Tofacitinib	200192	ICK		nM
10226-999-4	Tofacitinib	200193	IGF1R		nM
10226-999-4	Tofacitinib	200194	IKKA		nM
10226-999-4	Tofacitinib	200195	IKKB		nM
10226-999-4	Tofacitinib	200196	IKKE		nM
10226-999-4	Tofacitinib	200197	INSR		nM
10226-999-4	Tofacitinib	200198	INSRR		nM
10226-999-4	Tofacitinib	200199	IRAK1		nM
10226-999-4	Tofacitinib	200200	IRAK3		nM
10226-999-4	Tofacitinib	200201	IRAK4		nM
10226-999-4	Tofacitinib	200202	ITK		nM
10226-999-4	Tofacitinib	200203	JAK1(JH1domain-catalytic)	1.6	nM
10226-999-4	Tofacitinib	200204	JAK1(JH2domain-pseudokinase)		nM
10226-999-4	Tofacitinib	200207	JAK2(JH1domain-catalytic)	0.6	nM
10226-999-4	Tofacitinib	200209	JAK3(JH1domain-catalytic)	0.2	nM
10226-999-4	Tofacitinib	200211	JNK1		nM
10226-999-4	Tofacitinib	200212	MK09		nM
10226-999-4	Tofacitinib	200213	JNK3		nM
10226-999-4	Tofacitinib	200214	KIT		nM
10226-999-4	Tofacitinib	200215	KIT(A829P)		nM
10226-999-4	Tofacitinib	200216	KIT(D816H)		nM
10226-999-4	Tofacitinib	200217	KIT(D816V)		nM
10226-999-4	Tofacitinib	200218	KIT(L576P)		nM
10226-999-4	Tofacitinib	200219	KIT(V559D)		nM
10226-999-4	Tofacitinib	200220	KIT(V559D,T670I)		nM
10226-999-4	Tofacitinib	200221	KIT(V559D,V654A)		nM
10226-999-4	Tofacitinib	200222	LATS1		nM
10226-999-4	Tofacitinib	200223	LATS2		nM
10226-999-4	Tofacitinib	200224	LCK	460.0	nM
10226-999-4	Tofacitinib	200225	LIMK1		nM
10226-999-4	Tofacitinib	200226	LIMK2		nM
10226-999-4	Tofacitinib	200227	LKB1		nM
10226-999-4	Tofacitinib	200228	LOK		nM
10226-999-4	Tofacitinib	200229	LRRK2	1300.0	nM
10226-999-4	Tofacitinib	200230	LRRK2(G2019S)	550.0	nM
10226-999-4	Tofacitinib	200231	LTK		nM
10226-999-4	Tofacitinib	200232	LYN		nM
10226-999-4	Tofacitinib	200233	M3K13		nM
10226-999-4	Tofacitinib	200234	MAK		nM
10226-999-4	Tofacitinib	200235	MAP3K1		nM
10226-999-4	Tofacitinib	200236	MAP3K15		nM
10226-999-4	Tofacitinib	200237	M3K2		nM
10226-999-4	Tofacitinib	200238	MAP3K3		nM
10226-999-4	Tofacitinib	200239	MAP3K4		nM
10226-999-4	Tofacitinib	200240	MAP4K2	4800.0	nM
10226-999-4	Tofacitinib	200241	M4K3		nM
10226-999-4	Tofacitinib	200242	MAP4K4		nM
10226-999-4	Tofacitinib	200243	MAP4K5		nM
10226-999-4	Tofacitinib	200244	MAPKAPK2		nM
10226-999-4	Tofacitinib	200245	MAPKAPK5		nM
10226-999-4	Tofacitinib	200246	MARK1		nM
10226-999-4	Tofacitinib	200247	MARK2		nM
10226-999-4	Tofacitinib	200248	MARK3		nM
10226-999-4	Tofacitinib	200249	MARK4		nM
10226-999-4	Tofacitinib	200250	MAST1		nM
10226-999-4	Tofacitinib	200251	MP2K1		nM
10226-999-4	Tofacitinib	200252	MP2K2		nM
10226-999-4	Tofacitinib	200253	MP2K3		nM
10226-999-4	Tofacitinib	200254	MP2K4		nM
10226-999-4	Tofacitinib	200255	MP2K5		nM
10226-999-4	Tofacitinib	200256	MP2K6		nM
10226-999-4	Tofacitinib	200257	MELK		nM
10226-999-4	Tofacitinib	200258	MERTK		nM
10226-999-4	Tofacitinib	200259	MET		nM
10226-999-4	Tofacitinib	200260	MET(M1250T)		nM
10226-999-4	Tofacitinib	200261	MET(Y1235D)		nM
10226-999-4	Tofacitinib	200262	MINK		nM
10226-999-4	Tofacitinib	200263	MP2K7		nM
10226-999-4	Tofacitinib	200264	MKNK1		nM
10226-999-4	Tofacitinib	200265	MKNK2	1600.0	nM
10226-999-4	Tofacitinib	200266	MLCK		nM
10226-999-4	Tofacitinib	200267	MLK1		nM
10226-999-4	Tofacitinib	200268	MLK2		nM
10226-999-4	Tofacitinib	200269	MLK3		nM
10226-999-4	Tofacitinib	200270	MRCKA		nM
10226-999-4	Tofacitinib	200271	MRCKB		nM
10226-999-4	Tofacitinib	200272	MST1		nM
10226-999-4	Tofacitinib	200273	MST1R		nM
10226-999-4	Tofacitinib	200274	MST2		nM
10226-999-4	Tofacitinib	200275	MST3		nM
10226-999-4	Tofacitinib	200276	MST4		nM
10226-999-4	Tofacitinib	200277	MTOR		nM
10226-999-4	Tofacitinib	200278	MUSK		nM
10226-999-4	Tofacitinib	200279	MYLK		nM
10226-999-4	Tofacitinib	200280	MYLK2		nM
10226-999-4	Tofacitinib	200281	MYLK4		nM
10226-999-4	Tofacitinib	200282	MYO3A		nM
10226-999-4	Tofacitinib	200283	MYO3B		nM
10226-999-4	Tofacitinib	200284	NDR1		nM
10226-999-4	Tofacitinib	200285	NDR2		nM
10226-999-4	Tofacitinib	200286	NEK1		nM
10226-999-4	Tofacitinib	200287	NEK11		nM
10226-999-4	Tofacitinib	200288	NEK2		nM
10226-999-4	Tofacitinib	200289	NEK3		nM
10226-999-4	Tofacitinib	200290	NEK4		nM
10226-999-4	Tofacitinib	200291	NEK5		nM
10226-999-4	Tofacitinib	200292	NEK6		nM
10226-999-4	Tofacitinib	200293	NEK7		nM
10226-999-4	Tofacitinib	200294	NEK9		nM
10226-999-4	Tofacitinib	200295	NIM1		nM
10226-999-4	Tofacitinib	200296	NLK		nM
10226-999-4	Tofacitinib	200297	OSR1		nM
10226-999-4	Tofacitinib	200298	MK14		nM
10226-999-4	Tofacitinib	200299	MK11		nM
10226-999-4	Tofacitinib	200300	MK13		nM
10226-999-4	Tofacitinib	200301	MK12		nM
10226-999-4	Tofacitinib	200302	PAK1		nM
10226-999-4	Tofacitinib	200303	PAK2		nM
10226-999-4	Tofacitinib	200304	PAK3		nM
10226-999-4	Tofacitinib	200305	PAK4		nM
10226-999-4	Tofacitinib	200306	PAK6		nM
10226-999-4	Tofacitinib	200307	PAK7		nM
10226-999-4	Tofacitinib	200309	CDK16		nM
10226-999-4	Tofacitinib	200310	PCTK2		nM
10226-999-4	Tofacitinib	200311	PCTK3		nM
10226-999-4	Tofacitinib	200312	PGFRA		nM
10226-999-4	Tofacitinib	200313	PGFRB		nM
10226-999-4	Tofacitinib	200314	PDPK1		nM
10226-999-4	Tofacitinib	200315	PFCDPK1(P.falciparum)		nM
10226-999-4	Tofacitinib	200316	PFPK5(P.falciparum)		nM
10226-999-4	Tofacitinib	200317	CDK15		nM
10226-999-4	Tofacitinib	200318	CDK14		nM
10226-999-4	Tofacitinib	200319	PHKG1		nM
10226-999-4	Tofacitinib	200320	PHKG2		nM
10226-999-4	Tofacitinib	200321	PIK3C2B		nM
10226-999-4	Tofacitinib	200322	PIK3C2G		nM
10226-999-4	Tofacitinib	200323	PIK3CA		nM
10226-999-4	Tofacitinib	200324	PIK3CA(C420R)		nM
10226-999-4	Tofacitinib	200325	PIK3CA(E542K)		nM
10226-999-4	Tofacitinib	200326	PIK3CA(E545A)		nM
10226-999-4	Tofacitinib	200327	PIK3CA(E545K)		nM
10226-999-4	Tofacitinib	200328	PIK3CA(H1047L)		nM
10226-999-4	Tofacitinib	200329	PIK3CA(H1047Y)		nM
10226-999-4	Tofacitinib	200330	PIK3CA(I800L)		nM
10226-999-4	Tofacitinib	200331	PIK3CA(M1043I)		nM
10226-999-4	Tofacitinib	200332	PIK3CA(Q546K)		nM
10226-999-4	Tofacitinib	200333	PIK3CB		nM
10226-999-4	Tofacitinib	200334	PIK3CD		nM
10226-999-4	Tofacitinib	200335	PIK3CG		nM
10226-999-4	Tofacitinib	200336	PIK4CB		nM
10226-999-4	Tofacitinib	200337	PIM1		nM
10226-999-4	Tofacitinib	200338	PIM2		nM
10226-999-4	Tofacitinib	200339	PIM3		nM
10226-999-4	Tofacitinib	200340	PIP5K1A		nM
10226-999-4	Tofacitinib	200341	PIP5K1C		nM
10226-999-4	Tofacitinib	200342	PIP5K2B		nM
10226-999-4	Tofacitinib	200343	PI42C		nM
10226-999-4	Tofacitinib	200344	PKAC-alpha		nM
10226-999-4	Tofacitinib	200345	PKAC-beta		nM
10226-999-4	Tofacitinib	200346	PKMYT1		nM
10226-999-4	Tofacitinib	200347	PKN1	170.0	nM
10226-999-4	Tofacitinib	200348	PKN2	1200.0	nM
10226-999-4	Tofacitinib	200349	PKNB(M.tuberculosis)	2000.0	nM
10226-999-4	Tofacitinib	200350	PLK1		nM
10226-999-4	Tofacitinib	200351	PLK2		nM
10226-999-4	Tofacitinib	200352	PLK3		nM
10226-999-4	Tofacitinib	200353	PLK4		nM
10226-999-4	Tofacitinib	200354	KPCD	2000.0	nM
10226-999-4	Tofacitinib	200355	KPCE		nM
10226-999-4	Tofacitinib	200356	KPCL		nM
10226-999-4	Tofacitinib	200357	KPCI		nM
10226-999-4	Tofacitinib	200358	KPCT		nM
10226-999-4	Tofacitinib	200359	KPCD1		nM
10226-999-4	Tofacitinib	200360	KPCD2		nM
10226-999-4	Tofacitinib	200361	KPCD3		nM
10226-999-4	Tofacitinib	200362	KGP1		nM
10226-999-4	Tofacitinib	200363	KGP2		nM
10226-999-4	Tofacitinib	200364	PRKR		nM
10226-999-4	Tofacitinib	200365	PRKX		nM
10226-999-4	Tofacitinib	200366	PRP4		nM
10226-999-4	Tofacitinib	200367	FAK2		nM
10226-999-4	Tofacitinib	200368	SIK3		nM
10226-999-4	Tofacitinib	200369	RAF1		nM
10226-999-4	Tofacitinib	200370	RET		nM
10226-999-4	Tofacitinib	200371	RET(M918T)	3300.0	nM
10226-999-4	Tofacitinib	200372	RET(V804L)		nM
10226-999-4	Tofacitinib	200373	RET(V804M)		nM
10226-999-4	Tofacitinib	200374	RIOK1		nM
10226-999-4	Tofacitinib	200375	RIOK2		nM
10226-999-4	Tofacitinib	200376	RIOK3		nM
10226-999-4	Tofacitinib	200377	RIPK1		nM
10226-999-4	Tofacitinib	200378	RIPK2		nM
10226-999-4	Tofacitinib	200379	RIPK4		nM
10226-999-4	Tofacitinib	200380	RIPK5		nM
10226-999-4	Tofacitinib	200381	ROCK1	470.0	nM
10226-999-4	Tofacitinib	200382	ROCK2	420.0	nM
10226-999-4	Tofacitinib	200383	ROS1		nM
10226-999-4	Tofacitinib	200390	RPS6KA4(Kin.Dom.1-N-terminal)		nM
10226-999-4	Tofacitinib	200392	RPS6KA4(Kin.Dom.2-C-terminal)		nM
10226-999-4	Tofacitinib	200394	RPS6KA5(Kin.Dom.1-N-terminal)		nM
10226-999-4	Tofacitinib	200396	RPS6KA5(Kin.Dom.2-C-terminal)		nM
10226-999-4	Tofacitinib	200399	RSK1(Kin.Dom.1-N-terminal)		nM
10226-999-4	Tofacitinib	200400	RSK1(Kin.Dom.2-C-terminal)	1400.0	nM
10226-999-4	Tofacitinib	200401	RSK2(Kin.Dom.1-N-terminal)		nM
10226-999-4	Tofacitinib	200402	RSK3(Kin.Dom.1-N-terminal)		nM
10226-999-4	Tofacitinib	200403	RSK3(Kin.Dom.2-C-terminal)	600.0	nM
10226-999-4	Tofacitinib	200404	RSK4(Kin.Dom.1-N-terminal)		nM
10226-999-4	Tofacitinib	200405	RSK4(Kin.Dom.2-C-terminal)	540.0	nM
10226-999-4	Tofacitinib	200406	S6K1		nM
10226-999-4	Tofacitinib	200407	SBK1		nM
10226-999-4	Tofacitinib	200408	SgK110		nM
10226-999-4	Tofacitinib	200409	SGK3		nM
10226-999-4	Tofacitinib	200410	SIK1		nM
10226-999-4	Tofacitinib	200411	SIK2		nM
10226-999-4	Tofacitinib	200412	SLK		nM
10226-999-4	Tofacitinib	200413	SNARK	240.0	nM
10226-999-4	Tofacitinib	200414	SNRK		nM
10226-999-4	Tofacitinib	200415	SRC		nM
10226-999-4	Tofacitinib	200416	SRMS		nM
10226-999-4	Tofacitinib	200417	SRPK1		nM
10226-999-4	Tofacitinib	200418	SRPK2		nM
10226-999-4	Tofacitinib	200419	SRPK3		nM
10226-999-4	Tofacitinib	200420	STK16		nM
10226-999-4	Tofacitinib	200421	STK33		nM
10226-999-4	Tofacitinib	200422	STK35		nM
10226-999-4	Tofacitinib	200423	STK36		nM
10226-999-4	Tofacitinib	200424	STK39		nM
10226-999-4	Tofacitinib	200425	SYK		nM
10226-999-4	Tofacitinib	200426	TAK1		nM
10226-999-4	Tofacitinib	200427	TAOK1		nM
10226-999-4	Tofacitinib	200428	TAOK2		nM
10226-999-4	Tofacitinib	200429	TAOK3		nM
10226-999-4	Tofacitinib	200430	TBK1		nM
10226-999-4	Tofacitinib	200431	TEC		nM
10226-999-4	Tofacitinib	200432	TESK1		nM
10226-999-4	Tofacitinib	200433	TGFBR1		nM
10226-999-4	Tofacitinib	200434	TGFBR2		nM
10226-999-4	Tofacitinib	200435	TIE1		nM
10226-999-4	Tofacitinib	200436	TIE2		nM
10226-999-4	Tofacitinib	200437	TLK1		nM
10226-999-4	Tofacitinib	200438	TLK2		nM
10226-999-4	Tofacitinib	200439	TNIK		nM
10226-999-4	Tofacitinib	200440	TNK1	120.0	nM
10226-999-4	Tofacitinib	200441	TNK2		nM
10226-999-4	Tofacitinib	200442	TNNI3K		nM
10226-999-4	Tofacitinib	200443	TRKA		nM
10226-999-4	Tofacitinib	200444	TRKB		nM
10226-999-4	Tofacitinib	200445	TRKC		nM
10226-999-4	Tofacitinib	200446	TRPM6		nM
10226-999-4	Tofacitinib	200447	TSSK1		nM
10226-999-4	Tofacitinib	200448	TTK		nM
10226-999-4	Tofacitinib	200449	TXK		nM
10226-999-4	Tofacitinib	200450	TYK2(JH1domain-catalytic)	4.8	nM
10226-999-4	Tofacitinib	200451	TYK2(JH2domain-pseudokinase)		nM
10226-999-4	Tofacitinib	200454	TYRO3		nM
10226-999-4	Tofacitinib	200455	ULK1		nM
10226-999-4	Tofacitinib	200456	ULK2		nM
10226-999-4	Tofacitinib	200457	ULK3	6400.0	nM
10226-999-4	Tofacitinib	200458	VGFR2		nM
10226-999-4	Tofacitinib	200459	VRK2		nM
10226-999-4	Tofacitinib	200460	WEE1		nM
10226-999-4	Tofacitinib	200461	WEE2		nM
10226-999-4	Tofacitinib	200462	YANK1		nM
10226-999-4	Tofacitinib	200463	YANK2		nM
10226-999-4	Tofacitinib	200464	YANK3		nM
10226-999-4	Tofacitinib	200465	YES		nM
10226-999-4	Tofacitinib	200466	YSK1		nM
10226-999-4	Tofacitinib	200467	YSK4		nM
10226-999-4	Tofacitinib	200468	MLTK		nM
10226-999-4	Tofacitinib	200469	ZAP70		nM
