Small Molecule HMS LINCS ID	Small Molecule Name	Protein HMS LINCS ID	Protein Name	Kd	Conc unit
10151-999-2	Nintedanib	200001	AAK1	63.0	nM
10151-999-2	Nintedanib	200004	ABL1(E255K)-phosphorylated	63.0	nM
10151-999-2	Nintedanib	200006	ABL1(F317I)-nonphosphorylated	6900.0	nM
10151-999-2	Nintedanib	200007	ABL1(F317I)-phosphorylated	2600.0	nM
10151-999-2	Nintedanib	200009	ABL1(F317L)-nonphosphorylated	2300.0	nM
10151-999-2	Nintedanib	200010	ABL1(F317L)-phosphorylated	640.0	nM
10151-999-2	Nintedanib	200012	ABL1(H396P)-nonphosphorylated	45.0	nM
10151-999-2	Nintedanib	200013	ABL1(H396P)-phosphorylated	49.0	nM
10151-999-2	Nintedanib	200015	ABL1(M351T)-phosphorylated	52.0	nM
10151-999-2	Nintedanib	200017	ABL1(Q252H)-nonphosphorylated	73.0	nM
10151-999-2	Nintedanib	200018	ABL1(Q252H)-phosphorylated	28.0	nM
10151-999-2	Nintedanib	200020	ABL1(T315I)-nonphosphorylated	66.0	nM
10151-999-2	Nintedanib	200021	ABL1(T315I)-phosphorylated	10.0	nM
10151-999-2	Nintedanib	200023	ABL1(Y253F)-phosphorylated	37.0	nM
10151-999-2	Nintedanib	200024	ABL1-nonphosphorylated	230.0	nM
10151-999-2	Nintedanib	200025	ABL1-phosphorylated	64.0	nM
10151-999-2	Nintedanib	200026	ABL2	2000.0	nM
10151-999-2	Nintedanib	200027	ACVR1	600.0	nM
10151-999-2	Nintedanib	200028	ACVR1B	4900.0	nM
10151-999-2	Nintedanib	200029	ACVR2A		nM
10151-999-2	Nintedanib	200030	ACVR2B		nM
10151-999-2	Nintedanib	200031	ACVRL1	4200.0	nM
10151-999-2	Nintedanib	200032	ADCK3		nM
10151-999-2	Nintedanib	200033	ADCK4		nM
10151-999-2	Nintedanib	200034	AKT1		nM
10151-999-2	Nintedanib	200035	AKT2		nM
10151-999-2	Nintedanib	200036	AKT3		nM
10151-999-2	Nintedanib	200037	ALK	31.0	nM
10151-999-2	Nintedanib	200038	AMPK-alpha1	87.0	nM
10151-999-2	Nintedanib	200039	AMPK-alpha2	84.0	nM
10151-999-2	Nintedanib	200040	ANKK1		nM
10151-999-2	Nintedanib	200041	NUAK1	160.0	nM
10151-999-2	Nintedanib	200042	M3K5		nM
10151-999-2	Nintedanib	200043	M3K6		nM
10151-999-2	Nintedanib	200044	AURKA		nM
10151-999-2	Nintedanib	200045	AURKB	420.0	nM
10151-999-2	Nintedanib	200046	AURKC	190.0	nM
10151-999-2	Nintedanib	200047	AXL	12.0	nM
10151-999-2	Nintedanib	200048	BIKE	2.2	nM
10151-999-2	Nintedanib	200049	BLK	380.0	nM
10151-999-2	Nintedanib	200050	BMPR1A		nM
10151-999-2	Nintedanib	200051	BMPR1B		nM
10151-999-2	Nintedanib	200052	BMPR2	56.0	nM
10151-999-2	Nintedanib	200053	BMX		nM
10151-999-2	Nintedanib	200054	BRAF		nM
10151-999-2	Nintedanib	200055	BRAF(V600E)		nM
10151-999-2	Nintedanib	200056	PTK6		nM
10151-999-2	Nintedanib	200057	BRSK1		nM
10151-999-2	Nintedanib	200058	BRSK2		nM
10151-999-2	Nintedanib	200059	BTK	310.0	nM
10151-999-2	Nintedanib	200060	CAMK1	5900.0	nM
10151-999-2	Nintedanib	200061	CAMK1D	2200.0	nM
10151-999-2	Nintedanib	200062	CAMK1G	260.0	nM
10151-999-2	Nintedanib	200063	CAMK2A	3600.0	nM
10151-999-2	Nintedanib	200064	CAMK2B		nM
10151-999-2	Nintedanib	200065	KCC2D		nM
10151-999-2	Nintedanib	200066	CAMK2G		nM
10151-999-2	Nintedanib	200067	KCC4	3700.0	nM
10151-999-2	Nintedanib	200068	KKCC1	630.0	nM
10151-999-2	Nintedanib	200069	CAMKK2	920.0	nM
10151-999-2	Nintedanib	200070	CASK		nM
10151-999-2	Nintedanib	200071	CDC2L1		nM
10151-999-2	Nintedanib	200072	CDC2L2		nM
10151-999-2	Nintedanib	200073	CDC2L5		nM
10151-999-2	Nintedanib	200074	CDK11		nM
10151-999-2	Nintedanib	200075	CDK2	1400.0	nM
10151-999-2	Nintedanib	200076	CDK3		nM
10151-999-2	Nintedanib	200077	CDK4-cyclinD1	160.0	nM
10151-999-2	Nintedanib	200078	CDK4-cyclinD3	720.0	nM
10151-999-2	Nintedanib	200079	CDK5		nM
10151-999-2	Nintedanib	200080	CDK7	300.0	nM
10151-999-2	Nintedanib	200081	CDK8		nM
10151-999-2	Nintedanib	200082	CDK9		nM
10151-999-2	Nintedanib	200083	CDKL1		nM
10151-999-2	Nintedanib	200084	CDKL2	1300.0	nM
10151-999-2	Nintedanib	200085	CDKL3		nM
10151-999-2	Nintedanib	200086	CDKL5		nM
10151-999-2	Nintedanib	200087	CHEK1	290.0	nM
10151-999-2	Nintedanib	200088	CHK2		nM
10151-999-2	Nintedanib	200089	CIT		nM
10151-999-2	Nintedanib	200090	CLK1	8.8	nM
10151-999-2	Nintedanib	200091	CLK2	760.0	nM
10151-999-2	Nintedanib	200092	CLK3		nM
10151-999-2	Nintedanib	200093	CLK4	18.0	nM
10151-999-2	Nintedanib	200094	CSF1R	48.0	nM
10151-999-2	Nintedanib	200095	CSK		nM
10151-999-2	Nintedanib	200096	CSNK1A1		nM
10151-999-2	Nintedanib	200097	CSNK1A1L		nM
10151-999-2	Nintedanib	200098	CSNK1D	1300.0	nM
10151-999-2	Nintedanib	200099	CSNK1E	230.0	nM
10151-999-2	Nintedanib	200100	KC1G1		nM
10151-999-2	Nintedanib	200101	KC1G2		nM
10151-999-2	Nintedanib	200102	CSNK1G3		nM
10151-999-2	Nintedanib	200103	CSNK2A1	7500.0	nM
10151-999-2	Nintedanib	200104	CSNK2A2	890.0	nM
10151-999-2	Nintedanib	200105	CTK		nM
10151-999-2	Nintedanib	200106	DAPK1		nM
10151-999-2	Nintedanib	200107	DAPK2	3200.0	nM
10151-999-2	Nintedanib	200108	DAPK3	2100.0	nM
10151-999-2	Nintedanib	200109	DCLK1	540.0	nM
10151-999-2	Nintedanib	200110	DCAMKL2		nM
10151-999-2	Nintedanib	200111	DCAMKL3	770.0	nM
10151-999-2	Nintedanib	200112	DDR1	12.0	nM
10151-999-2	Nintedanib	200113	DDR2	42.0	nM
10151-999-2	Nintedanib	200114	M3K12	140.0	nM
10151-999-2	Nintedanib	200115	DMPK		nM
10151-999-2	Nintedanib	200116	DMPK2		nM
10151-999-2	Nintedanib	200117	DRAK1	110.0	nM
10151-999-2	Nintedanib	200118	DRAK2	670.0	nM
10151-999-2	Nintedanib	200119	DYRK1A		nM
10151-999-2	Nintedanib	200120	DYRK1B	1600.0	nM
10151-999-2	Nintedanib	200121	DYRK2		nM
10151-999-2	Nintedanib	200122	EGFR		nM
10151-999-2	Nintedanib	200123	EGFR(E746-A750del)		nM
10151-999-2	Nintedanib	200124	EGFR(G719C)		nM
10151-999-2	Nintedanib	200125	EGFR(G719S)		nM
10151-999-2	Nintedanib	200126	EGFR(L747-E749del, A750P)		nM
10151-999-2	Nintedanib	200127	EGFR(L747-S752del, P753S)		nM
10151-999-2	Nintedanib	200128	EGFR(L747-T751del,Sins)		nM
10151-999-2	Nintedanib	200129	EGFR(L858R)		nM
10151-999-2	Nintedanib	200130	EGFR(L858R,T790M)		nM
10151-999-2	Nintedanib	200131	EGFR(L861Q)		nM
10151-999-2	Nintedanib	200132	EGFR(S752-I759del)		nM
10151-999-2	Nintedanib	200133	EGFR(T790M)		nM
10151-999-2	Nintedanib	200134	EIF2AK1		nM
10151-999-2	Nintedanib	200135	EPHA1	1200.0	nM
10151-999-2	Nintedanib	200136	EPHA2	2900.0	nM
10151-999-2	Nintedanib	200137	EPHA3	8600.0	nM
10151-999-2	Nintedanib	200138	EPHA4		nM
10151-999-2	Nintedanib	200139	EPHA5		nM
10151-999-2	Nintedanib	200140	EPHA6	940.0	nM
10151-999-2	Nintedanib	200141	EPHA7		nM
10151-999-2	Nintedanib	200142	EPHA8		nM
10151-999-2	Nintedanib	200143	EPHB1	550.0	nM
10151-999-2	Nintedanib	200144	EPHB2		nM
10151-999-2	Nintedanib	200145	EPHB3		nM
10151-999-2	Nintedanib	200146	EPHB4	1100.0	nM
10151-999-2	Nintedanib	200147	EPHB6	140.0	nM
10151-999-2	Nintedanib	200148	ERBB2		nM
10151-999-2	Nintedanib	200149	ERBB3		nM
10151-999-2	Nintedanib	200150	ERBB4		nM
10151-999-2	Nintedanib	200151	MK03		nM
10151-999-2	Nintedanib	200152	MK01		nM
10151-999-2	Nintedanib	200153	ERK3		nM
10151-999-2	Nintedanib	200154	ERK4		nM
10151-999-2	Nintedanib	200155	ERK5	2500.0	nM
10151-999-2	Nintedanib	200156	ERK8		nM
10151-999-2	Nintedanib	200157	ERN1	2000.0	nM
10151-999-2	Nintedanib	200158	FAK1	210.0	nM
10151-999-2	Nintedanib	200159	FER	73.0	nM
10151-999-2	Nintedanib	200160	FES	1200.0	nM
10151-999-2	Nintedanib	200161	FGFR1	92.0	nM
10151-999-2	Nintedanib	200162	FGFR2	350.0	nM
10151-999-2	Nintedanib	200163	FGFR3	93.0	nM
10151-999-2	Nintedanib	200164	FGFR3(G697C)	140.0	nM
10151-999-2	Nintedanib	200165	FGFR4	1800.0	nM
10151-999-2	Nintedanib	200166	FGR	300.0	nM
10151-999-2	Nintedanib	200167	VGFR1	63.0	nM
10151-999-2	Nintedanib	200168	FLT3	3.8	nM
10151-999-2	Nintedanib	200169	FLT3(D835H)	0.7	nM
10151-999-2	Nintedanib	200170	FLT3(D835Y)	0.4	nM
10151-999-2	Nintedanib	200171	FLT3(ITD)	0.7	nM
10151-999-2	Nintedanib	200172	FLT3(K663Q)	4.5	nM
10151-999-2	Nintedanib	200173	FLT3(N841I)	2.6	nM
10151-999-2	Nintedanib	200174	FLT3(R834Q)	17.0	nM
10151-999-2	Nintedanib	200175	FLT4	95.0	nM
10151-999-2	Nintedanib	200176	FRK	2700.0	nM
10151-999-2	Nintedanib	200177	FYN	630.0	nM
10151-999-2	Nintedanib	200178	GAK		nM
10151-999-2	Nintedanib	200179	GCN2(Kin.Dom.2,S808G)	2000.0	nM
10151-999-2	Nintedanib	200180	GRK1	1000.0	nM
10151-999-2	Nintedanib	200181	GRK4	17.0	nM
10151-999-2	Nintedanib	200182	GRK7	1200.0	nM
10151-999-2	Nintedanib	200183	GSK3A	430.0	nM
10151-999-2	Nintedanib	200184	GSK3B	83.0	nM
10151-999-2	Nintedanib	200185	HCK	5300.0	nM
10151-999-2	Nintedanib	200186	HIPK1	1300.0	nM
10151-999-2	Nintedanib	200187	HIPK2	790.0	nM
10151-999-2	Nintedanib	200188	HIPK3	850.0	nM
10151-999-2	Nintedanib	200189	HIPK4	1200.0	nM
10151-999-2	Nintedanib	200190	M4K1	35.0	nM
10151-999-2	Nintedanib	200191	HUNK		nM
10151-999-2	Nintedanib	200192	ICK	1700.0	nM
10151-999-2	Nintedanib	200193	IGF1R	62.0	nM
10151-999-2	Nintedanib	200194	IKKA	4500.0	nM
10151-999-2	Nintedanib	200195	IKKB		nM
10151-999-2	Nintedanib	200196	IKKE	170.0	nM
10151-999-2	Nintedanib	200197	INSR	24.0	nM
10151-999-2	Nintedanib	200198	INSRR	21.0	nM
10151-999-2	Nintedanib	200199	IRAK1	120.0	nM
10151-999-2	Nintedanib	200200	IRAK3	5300.0	nM
10151-999-2	Nintedanib	200201	IRAK4	810.0	nM
10151-999-2	Nintedanib	200202	ITK	210.0	nM
10151-999-2	Nintedanib	200203	JAK1(JH1domain-catalytic)	2500.0	nM
10151-999-2	Nintedanib	200204	JAK1(JH2domain-pseudokinase)	4.8	nM
10151-999-2	Nintedanib	200207	JAK2(JH1domain-catalytic)	14.0	nM
10151-999-2	Nintedanib	200209	JAK3(JH1domain-catalytic)	8.2	nM
10151-999-2	Nintedanib	200211	JNK1	630.0	nM
10151-999-2	Nintedanib	200212	MK09		nM
10151-999-2	Nintedanib	200213	JNK3	270.0	nM
10151-999-2	Nintedanib	200214	KIT	5.7	nM
10151-999-2	Nintedanib	200215	KIT(A829P)	87.0	nM
10151-999-2	Nintedanib	200216	KIT(D816H)	310.0	nM
10151-999-2	Nintedanib	200217	KIT(D816V)	47.0	nM
10151-999-2	Nintedanib	200218	KIT(L576P)	2.7	nM
10151-999-2	Nintedanib	200219	KIT(V559D)	6.3	nM
10151-999-2	Nintedanib	200220	KIT(V559D,T670I)	2.9	nM
10151-999-2	Nintedanib	200221	KIT(V559D,V654A)	29.0	nM
10151-999-2	Nintedanib	200222	LATS1	420.0	nM
10151-999-2	Nintedanib	200223	LATS2	380.0	nM
10151-999-2	Nintedanib	200224	LCK	6.2	nM
10151-999-2	Nintedanib	200225	LIMK1		nM
10151-999-2	Nintedanib	200226	LIMK2		nM
10151-999-2	Nintedanib	200227	LKB1	18.0	nM
10151-999-2	Nintedanib	200228	LOK	87.0	nM
10151-999-2	Nintedanib	200229	LRRK2	46.0	nM
10151-999-2	Nintedanib	200230	LRRK2(G2019S)	37.0	nM
10151-999-2	Nintedanib	200231	LTK	150.0	nM
10151-999-2	Nintedanib	200232	LYN	940.0	nM
10151-999-2	Nintedanib	200233	M3K13	140.0	nM
10151-999-2	Nintedanib	200234	MAK		nM
10151-999-2	Nintedanib	200235	MAP3K1		nM
10151-999-2	Nintedanib	200236	MAP3K15	1400.0	nM
10151-999-2	Nintedanib	200237	M3K2	9.4	nM
10151-999-2	Nintedanib	200238	MAP3K3	34.0	nM
10151-999-2	Nintedanib	200239	MAP3K4		nM
10151-999-2	Nintedanib	200240	MAP4K2	290.0	nM
10151-999-2	Nintedanib	200241	M4K3	290.0	nM
10151-999-2	Nintedanib	200242	MAP4K4	150.0	nM
10151-999-2	Nintedanib	200243	MAP4K5	390.0	nM
10151-999-2	Nintedanib	200244	MAPKAPK2		nM
10151-999-2	Nintedanib	200245	MAPKAPK5		nM
10151-999-2	Nintedanib	200246	MARK1	1400.0	nM
10151-999-2	Nintedanib	200247	MARK2	1400.0	nM
10151-999-2	Nintedanib	200248	MARK3	770.0	nM
10151-999-2	Nintedanib	200249	MARK4	2000.0	nM
10151-999-2	Nintedanib	200250	MAST1	4600.0	nM
10151-999-2	Nintedanib	200251	MP2K1	10.0	nM
10151-999-2	Nintedanib	200252	MP2K2	42.0	nM
10151-999-2	Nintedanib	200253	MP2K3	2100.0	nM
10151-999-2	Nintedanib	200254	MP2K4	3700.0	nM
10151-999-2	Nintedanib	200255	MP2K5	1.8	nM
10151-999-2	Nintedanib	200256	MP2K6		nM
10151-999-2	Nintedanib	200257	MELK	4.9	nM
10151-999-2	Nintedanib	200258	MERTK	8.5	nM
10151-999-2	Nintedanib	200259	MET	200.0	nM
10151-999-2	Nintedanib	200260	MET(M1250T)	340.0	nM
10151-999-2	Nintedanib	200261	MET(Y1235D)	460.0	nM
10151-999-2	Nintedanib	200262	MINK	82.0	nM
10151-999-2	Nintedanib	200263	MP2K7		nM
10151-999-2	Nintedanib	200264	MKNK1		nM
10151-999-2	Nintedanib	200265	MKNK2		nM
10151-999-2	Nintedanib	200266	MLCK	110.0	nM
10151-999-2	Nintedanib	200267	MLK1	220.0	nM
10151-999-2	Nintedanib	200268	MLK2	2300.0	nM
10151-999-2	Nintedanib	200269	MLK3	700.0	nM
10151-999-2	Nintedanib	200270	MRCKA		nM
10151-999-2	Nintedanib	200271	MRCKB		nM
10151-999-2	Nintedanib	200272	MST1	9.0	nM
10151-999-2	Nintedanib	200273	MST1R		nM
10151-999-2	Nintedanib	200274	MST2	38.0	nM
10151-999-2	Nintedanib	200275	MST3	110.0	nM
10151-999-2	Nintedanib	200276	MST4	49.0	nM
10151-999-2	Nintedanib	200277	MTOR		nM
10151-999-2	Nintedanib	200278	MUSK	590.0	nM
10151-999-2	Nintedanib	200279	MYLK	290.0	nM
10151-999-2	Nintedanib	200280	MYLK2	4000.0	nM
10151-999-2	Nintedanib	200281	MYLK4	440.0	nM
10151-999-2	Nintedanib	200282	MYO3A		nM
10151-999-2	Nintedanib	200283	MYO3B	2700.0	nM
10151-999-2	Nintedanib	200284	NDR1		nM
10151-999-2	Nintedanib	200285	NDR2		nM
10151-999-2	Nintedanib	200286	NEK1		nM
10151-999-2	Nintedanib	200287	NEK11		nM
10151-999-2	Nintedanib	200288	NEK2		nM
10151-999-2	Nintedanib	200289	NEK3		nM
10151-999-2	Nintedanib	200290	NEK4		nM
10151-999-2	Nintedanib	200291	NEK5		nM
10151-999-2	Nintedanib	200292	NEK6		nM
10151-999-2	Nintedanib	200293	NEK7		nM
10151-999-2	Nintedanib	200294	NEK9		nM
10151-999-2	Nintedanib	200295	NIM1		nM
10151-999-2	Nintedanib	200296	NLK		nM
10151-999-2	Nintedanib	200297	OSR1	1300.0	nM
10151-999-2	Nintedanib	200298	MK14		nM
10151-999-2	Nintedanib	200299	MK11		nM
10151-999-2	Nintedanib	200300	MK13		nM
10151-999-2	Nintedanib	200301	MK12		nM
10151-999-2	Nintedanib	200302	PAK1		nM
10151-999-2	Nintedanib	200303	PAK2	3300.0	nM
10151-999-2	Nintedanib	200304	PAK3	210.0	nM
10151-999-2	Nintedanib	200305	PAK4	3000.0	nM
10151-999-2	Nintedanib	200306	PAK6		nM
10151-999-2	Nintedanib	200307	PAK7	1300.0	nM
10151-999-2	Nintedanib	200309	CDK16	21.0	nM
10151-999-2	Nintedanib	200310	PCTK2	93.0	nM
10151-999-2	Nintedanib	200311	PCTK3	510.0	nM
10151-999-2	Nintedanib	200312	PGFRA	16.0	nM
10151-999-2	Nintedanib	200313	PGFRB	15.0	nM
10151-999-2	Nintedanib	200314	PDPK1	2800.0	nM
10151-999-2	Nintedanib	200315	PFCDPK1(P.falciparum)	1200.0	nM
10151-999-2	Nintedanib	200316	PFPK5(P.falciparum)		nM
10151-999-2	Nintedanib	200317	CDK15		nM
10151-999-2	Nintedanib	200318	CDK14	470.0	nM
10151-999-2	Nintedanib	200319	PHKG1	140.0	nM
10151-999-2	Nintedanib	200320	PHKG2	260.0	nM
10151-999-2	Nintedanib	200321	PIK3C2B		nM
10151-999-2	Nintedanib	200322	PIK3C2G		nM
10151-999-2	Nintedanib	200323	PIK3CA		nM
10151-999-2	Nintedanib	200324	PIK3CA(C420R)		nM
10151-999-2	Nintedanib	200325	PIK3CA(E542K)		nM
10151-999-2	Nintedanib	200326	PIK3CA(E545A)		nM
10151-999-2	Nintedanib	200327	PIK3CA(E545K)		nM
10151-999-2	Nintedanib	200328	PIK3CA(H1047L)		nM
10151-999-2	Nintedanib	200329	PIK3CA(H1047Y)		nM
10151-999-2	Nintedanib	200330	PIK3CA(I800L)		nM
10151-999-2	Nintedanib	200331	PIK3CA(M1043I)		nM
10151-999-2	Nintedanib	200332	PIK3CA(Q546K)		nM
10151-999-2	Nintedanib	200333	PIK3CB		nM
10151-999-2	Nintedanib	200334	PIK3CD		nM
10151-999-2	Nintedanib	200335	PIK3CG		nM
10151-999-2	Nintedanib	200336	PIK4CB		nM
10151-999-2	Nintedanib	200337	PIM1		nM
10151-999-2	Nintedanib	200338	PIM2		nM
10151-999-2	Nintedanib	200339	PIM3		nM
10151-999-2	Nintedanib	200340	PIP5K1A	49.0	nM
10151-999-2	Nintedanib	200341	PIP5K1C		nM
10151-999-2	Nintedanib	200342	PIP5K2B	17.0	nM
10151-999-2	Nintedanib	200343	PI42C		nM
10151-999-2	Nintedanib	200344	PKAC-alpha		nM
10151-999-2	Nintedanib	200345	PKAC-beta		nM
10151-999-2	Nintedanib	200346	PKMYT1		nM
10151-999-2	Nintedanib	200347	PKN1	740.0	nM
10151-999-2	Nintedanib	200348	PKN2	1400.0	nM
10151-999-2	Nintedanib	200349	PKNB(M.tuberculosis)	3.6	nM
10151-999-2	Nintedanib	200350	PLK1		nM
10151-999-2	Nintedanib	200351	PLK2		nM
10151-999-2	Nintedanib	200352	PLK3		nM
10151-999-2	Nintedanib	200353	PLK4	53.0	nM
10151-999-2	Nintedanib	200354	KPCD		nM
10151-999-2	Nintedanib	200355	KPCE		nM
10151-999-2	Nintedanib	200356	KPCL		nM
10151-999-2	Nintedanib	200357	KPCI		nM
10151-999-2	Nintedanib	200358	KPCT	5500.0	nM
10151-999-2	Nintedanib	200359	KPCD1	990.0	nM
10151-999-2	Nintedanib	200360	KPCD2	720.0	nM
10151-999-2	Nintedanib	200361	KPCD3	640.0	nM
10151-999-2	Nintedanib	200362	KGP1	14.0	nM
10151-999-2	Nintedanib	200363	KGP2		nM
10151-999-2	Nintedanib	200364	PRKR		nM
10151-999-2	Nintedanib	200365	PRKX		nM
10151-999-2	Nintedanib	200366	PRP4	8.4	nM
10151-999-2	Nintedanib	200367	FAK2	81.0	nM
10151-999-2	Nintedanib	200368	SIK3		nM
10151-999-2	Nintedanib	200369	RAF1		nM
10151-999-2	Nintedanib	200370	RET	31.0	nM
10151-999-2	Nintedanib	200371	RET(M918T)	30.0	nM
10151-999-2	Nintedanib	200372	RET(V804L)	9.8	nM
10151-999-2	Nintedanib	200373	RET(V804M)	9.6	nM
10151-999-2	Nintedanib	200374	RIOK1	23.0	nM
10151-999-2	Nintedanib	200375	RIOK2		nM
10151-999-2	Nintedanib	200376	RIOK3	36.0	nM
10151-999-2	Nintedanib	200377	RIPK1	240.0	nM
10151-999-2	Nintedanib	200378	RIPK2		nM
10151-999-2	Nintedanib	200379	RIPK4	440.0	nM
10151-999-2	Nintedanib	200380	RIPK5		nM
10151-999-2	Nintedanib	200381	ROCK1		nM
10151-999-2	Nintedanib	200382	ROCK2		nM
10151-999-2	Nintedanib	200383	ROS1	3700.0	nM
10151-999-2	Nintedanib	200390	RPS6KA4(Kin.Dom.1-N-terminal)	620.0	nM
10151-999-2	Nintedanib	200392	RPS6KA4(Kin.Dom.2-C-terminal)		nM
10151-999-2	Nintedanib	200394	RPS6KA5(Kin.Dom.1-N-terminal)	200.0	nM
10151-999-2	Nintedanib	200396	RPS6KA5(Kin.Dom.2-C-terminal)		nM
10151-999-2	Nintedanib	200399	RSK1(Kin.Dom.1-N-terminal)	180.0	nM
10151-999-2	Nintedanib	200400	RSK1(Kin.Dom.2-C-terminal)		nM
10151-999-2	Nintedanib	200401	RSK2(Kin.Dom.1-N-terminal)	65.0	nM
10151-999-2	Nintedanib	200402	RSK3(Kin.Dom.1-N-terminal)	58.0	nM
10151-999-2	Nintedanib	200403	RSK3(Kin.Dom.2-C-terminal)		nM
10151-999-2	Nintedanib	200404	RSK4(Kin.Dom.1-N-terminal)	230.0	nM
10151-999-2	Nintedanib	200405	RSK4(Kin.Dom.2-C-terminal)		nM
10151-999-2	Nintedanib	200406	S6K1	190.0	nM
10151-999-2	Nintedanib	200407	SBK1	110.0	nM
10151-999-2	Nintedanib	200408	SgK110	2000.0	nM
10151-999-2	Nintedanib	200409	SGK3	1000.0	nM
10151-999-2	Nintedanib	200410	SIK1	670.0	nM
10151-999-2	Nintedanib	200411	SIK2	280.0	nM
10151-999-2	Nintedanib	200412	SLK	51.0	nM
10151-999-2	Nintedanib	200413	SNARK	21.0	nM
10151-999-2	Nintedanib	200414	SNRK		nM
10151-999-2	Nintedanib	200415	SRC	580.0	nM
10151-999-2	Nintedanib	200416	SRMS		nM
10151-999-2	Nintedanib	200417	SRPK1	37.0	nM
10151-999-2	Nintedanib	200418	SRPK2	36.0	nM
10151-999-2	Nintedanib	200419	SRPK3	12.0	nM
10151-999-2	Nintedanib	200420	STK16	18.0	nM
10151-999-2	Nintedanib	200421	STK33	1100.0	nM
10151-999-2	Nintedanib	200422	STK35	810.0	nM
10151-999-2	Nintedanib	200423	STK36		nM
10151-999-2	Nintedanib	200424	STK39	520.0	nM
10151-999-2	Nintedanib	200425	SYK		nM
10151-999-2	Nintedanib	200426	TAK1	4.1	nM
10151-999-2	Nintedanib	200427	TAOK1		nM
10151-999-2	Nintedanib	200428	TAOK2		nM
10151-999-2	Nintedanib	200429	TAOK3		nM
10151-999-2	Nintedanib	200430	TBK1	150.0	nM
10151-999-2	Nintedanib	200431	TEC		nM
10151-999-2	Nintedanib	200432	TESK1		nM
10151-999-2	Nintedanib	200433	TGFBR1	4200.0	nM
10151-999-2	Nintedanib	200434	TGFBR2		nM
10151-999-2	Nintedanib	200435	TIE1	2200.0	nM
10151-999-2	Nintedanib	200436	TIE2	1400.0	nM
10151-999-2	Nintedanib	200437	TLK1		nM
10151-999-2	Nintedanib	200438	TLK2		nM
10151-999-2	Nintedanib	200439	TNIK	53.0	nM
10151-999-2	Nintedanib	200440	TNK1	210.0	nM
10151-999-2	Nintedanib	200441	TNK2	1600.0	nM
10151-999-2	Nintedanib	200442	TNNI3K		nM
10151-999-2	Nintedanib	200443	TRKA	4.5	nM
10151-999-2	Nintedanib	200444	TRKB	19.0	nM
10151-999-2	Nintedanib	200445	TRKC	32.0	nM
10151-999-2	Nintedanib	200446	TRPM6		nM
10151-999-2	Nintedanib	200447	TSSK1	6100.0	nM
10151-999-2	Nintedanib	200448	TTK	22.0	nM
10151-999-2	Nintedanib	200449	TXK	860.0	nM
10151-999-2	Nintedanib	200450	TYK2(JH1domain-catalytic)	37.0	nM
10151-999-2	Nintedanib	200451	TYK2(JH2domain-pseudokinase)	500.0	nM
10151-999-2	Nintedanib	200454	TYRO3	4900.0	nM
10151-999-2	Nintedanib	200455	ULK1	340.0	nM
10151-999-2	Nintedanib	200456	ULK2	380.0	nM
10151-999-2	Nintedanib	200457	ULK3	60.0	nM
10151-999-2	Nintedanib	200458	VGFR2	2.9	nM
10151-999-2	Nintedanib	200459	VRK2		nM
10151-999-2	Nintedanib	200460	WEE1	2900.0	nM
10151-999-2	Nintedanib	200461	WEE2		nM
10151-999-2	Nintedanib	200462	YANK1		nM
10151-999-2	Nintedanib	200463	YANK2		nM
10151-999-2	Nintedanib	200464	YANK3		nM
10151-999-2	Nintedanib	200465	YES	80.0	nM
10151-999-2	Nintedanib	200466	YSK1		nM
10151-999-2	Nintedanib	200467	YSK4	5.2	nM
10151-999-2	Nintedanib	200468	MLTK		nM
10151-999-2	Nintedanib	200469	ZAP70	3500.0	nM
