Small Molecule HMS LINCS ID	Small Molecule Name	Protein HMS LINCS ID	Protein Name	Kd	Conc unit
10114-999-3	Pazopanib	200001	AAK1	2900.0	nM
10114-999-3	Pazopanib	200004	ABL1(E255K)-phosphorylated	800.0	nM
10114-999-3	Pazopanib	200006	ABL1(F317I)-nonphosphorylated		nM
10114-999-3	Pazopanib	200007	ABL1(F317I)-phosphorylated		nM
10114-999-3	Pazopanib	200009	ABL1(F317L)-nonphosphorylated	4400.0	nM
10114-999-3	Pazopanib	200010	ABL1(F317L)-phosphorylated	2700.0	nM
10114-999-3	Pazopanib	200012	ABL1(H396P)-nonphosphorylated	380.0	nM
10114-999-3	Pazopanib	200013	ABL1(H396P)-phosphorylated	700.0	nM
10114-999-3	Pazopanib	200015	ABL1(M351T)-phosphorylated	560.0	nM
10114-999-3	Pazopanib	200017	ABL1(Q252H)-nonphosphorylated	530.0	nM
10114-999-3	Pazopanib	200018	ABL1(Q252H)-phosphorylated	530.0	nM
10114-999-3	Pazopanib	200020	ABL1(T315I)-nonphosphorylated	3800.0	nM
10114-999-3	Pazopanib	200021	ABL1(T315I)-phosphorylated	2100.0	nM
10114-999-3	Pazopanib	200023	ABL1(Y253F)-phosphorylated	480.0	nM
10114-999-3	Pazopanib	200024	ABL1-nonphosphorylated	620.0	nM
10114-999-3	Pazopanib	200025	ABL1-phosphorylated	650.0	nM
10114-999-3	Pazopanib	200026	ABL2	3000.0	nM
10114-999-3	Pazopanib	200027	ACVR1		nM
10114-999-3	Pazopanib	200028	ACVR1B		nM
10114-999-3	Pazopanib	200029	ACVR2A		nM
10114-999-3	Pazopanib	200030	ACVR2B	2400.0	nM
10114-999-3	Pazopanib	200031	ACVRL1		nM
10114-999-3	Pazopanib	200032	ADCK3		nM
10114-999-3	Pazopanib	200033	ADCK4		nM
10114-999-3	Pazopanib	200034	AKT1		nM
10114-999-3	Pazopanib	200035	AKT2		nM
10114-999-3	Pazopanib	200036	AKT3		nM
10114-999-3	Pazopanib	200037	ALK	2200.0	nM
10114-999-3	Pazopanib	200038	AMPK-alpha1		nM
10114-999-3	Pazopanib	200039	AMPK-alpha2		nM
10114-999-3	Pazopanib	200040	ANKK1		nM
10114-999-3	Pazopanib	200041	NUAK1		nM
10114-999-3	Pazopanib	200042	M3K5		nM
10114-999-3	Pazopanib	200043	M3K6		nM
10114-999-3	Pazopanib	200044	AURKA	7100.0	nM
10114-999-3	Pazopanib	200045	AURKB		nM
10114-999-3	Pazopanib	200046	AURKC	750.0	nM
10114-999-3	Pazopanib	200047	AXL		nM
10114-999-3	Pazopanib	200048	BIKE	8800.0	nM
10114-999-3	Pazopanib	200049	BLK	2600.0	nM
10114-999-3	Pazopanib	200050	BMPR1A		nM
10114-999-3	Pazopanib	200051	BMPR1B	1000.0	nM
10114-999-3	Pazopanib	200052	BMPR2		nM
10114-999-3	Pazopanib	200053	BMX		nM
10114-999-3	Pazopanib	200054	BRAF	730.0	nM
10114-999-3	Pazopanib	200055	BRAF(V600E)	430.0	nM
10114-999-3	Pazopanib	200056	PTK6	2300.0	nM
10114-999-3	Pazopanib	200057	BRSK1		nM
10114-999-3	Pazopanib	200058	BRSK2		nM
10114-999-3	Pazopanib	200059	BTK		nM
10114-999-3	Pazopanib	200060	CAMK1	2100.0	nM
10114-999-3	Pazopanib	200061	CAMK1D		nM
10114-999-3	Pazopanib	200062	CAMK1G	3700.0	nM
10114-999-3	Pazopanib	200063	CAMK2A		nM
10114-999-3	Pazopanib	200064	CAMK2B		nM
10114-999-3	Pazopanib	200065	KCC2D		nM
10114-999-3	Pazopanib	200066	CAMK2G		nM
10114-999-3	Pazopanib	200067	KCC4		nM
10114-999-3	Pazopanib	200068	KKCC1		nM
10114-999-3	Pazopanib	200069	CAMKK2		nM
10114-999-3	Pazopanib	200070	CASK		nM
10114-999-3	Pazopanib	200071	CDC2L1	2100.0	nM
10114-999-3	Pazopanib	200072	CDC2L2	1300.0	nM
10114-999-3	Pazopanib	200073	CDC2L5		nM
10114-999-3	Pazopanib	200074	CDK11		nM
10114-999-3	Pazopanib	200075	CDK2		nM
10114-999-3	Pazopanib	200076	CDK3		nM
10114-999-3	Pazopanib	200077	CDK4-cyclinD1		nM
10114-999-3	Pazopanib	200078	CDK4-cyclinD3		nM
10114-999-3	Pazopanib	200079	CDK5		nM
10114-999-3	Pazopanib	200080	CDK7		nM
10114-999-3	Pazopanib	200081	CDK8		nM
10114-999-3	Pazopanib	200082	CDK9		nM
10114-999-3	Pazopanib	200083	CDKL1		nM
10114-999-3	Pazopanib	200084	CDKL2		nM
10114-999-3	Pazopanib	200085	CDKL3		nM
10114-999-3	Pazopanib	200086	CDKL5		nM
10114-999-3	Pazopanib	200087	CHEK1		nM
10114-999-3	Pazopanib	200088	CHK2		nM
10114-999-3	Pazopanib	200089	CIT		nM
10114-999-3	Pazopanib	200090	CLK1		nM
10114-999-3	Pazopanib	200091	CLK2		nM
10114-999-3	Pazopanib	200092	CLK3		nM
10114-999-3	Pazopanib	200093	CLK4		nM
10114-999-3	Pazopanib	200094	CSF1R	7.9	nM
10114-999-3	Pazopanib	200095	CSK		nM
10114-999-3	Pazopanib	200096	CSNK1A1		nM
10114-999-3	Pazopanib	200097	CSNK1A1L		nM
10114-999-3	Pazopanib	200098	CSNK1D		nM
10114-999-3	Pazopanib	200099	CSNK1E		nM
10114-999-3	Pazopanib	200100	KC1G1		nM
10114-999-3	Pazopanib	200101	KC1G2		nM
10114-999-3	Pazopanib	200102	CSNK1G3		nM
10114-999-3	Pazopanib	200103	CSNK2A1		nM
10114-999-3	Pazopanib	200104	CSNK2A2		nM
10114-999-3	Pazopanib	200105	CTK		nM
10114-999-3	Pazopanib	200106	DAPK1		nM
10114-999-3	Pazopanib	200107	DAPK2		nM
10114-999-3	Pazopanib	200108	DAPK3		nM
10114-999-3	Pazopanib	200109	DCLK1		nM
10114-999-3	Pazopanib	200110	DCAMKL2		nM
10114-999-3	Pazopanib	200111	DCAMKL3		nM
10114-999-3	Pazopanib	200112	DDR1	57.0	nM
10114-999-3	Pazopanib	200113	DDR2	98.0	nM
10114-999-3	Pazopanib	200114	M3K12		nM
10114-999-3	Pazopanib	200115	DMPK		nM
10114-999-3	Pazopanib	200116	DMPK2		nM
10114-999-3	Pazopanib	200117	DRAK1		nM
10114-999-3	Pazopanib	200118	DRAK2		nM
10114-999-3	Pazopanib	200119	DYRK1A		nM
10114-999-3	Pazopanib	200120	DYRK1B		nM
10114-999-3	Pazopanib	200121	DYRK2		nM
10114-999-3	Pazopanib	200122	EGFR		nM
10114-999-3	Pazopanib	200123	EGFR(E746-A750del)		nM
10114-999-3	Pazopanib	200124	EGFR(G719C)		nM
10114-999-3	Pazopanib	200125	EGFR(G719S)		nM
10114-999-3	Pazopanib	200126	EGFR(L747-E749del, A750P)		nM
10114-999-3	Pazopanib	200127	EGFR(L747-S752del, P753S)		nM
10114-999-3	Pazopanib	200128	EGFR(L747-T751del,Sins)		nM
10114-999-3	Pazopanib	200129	EGFR(L858R)		nM
10114-999-3	Pazopanib	200130	EGFR(L858R,T790M)		nM
10114-999-3	Pazopanib	200131	EGFR(L861Q)		nM
10114-999-3	Pazopanib	200132	EGFR(S752-I759del)		nM
10114-999-3	Pazopanib	200133	EGFR(T790M)		nM
10114-999-3	Pazopanib	200134	EIF2AK1		nM
10114-999-3	Pazopanib	200135	EPHA1		nM
10114-999-3	Pazopanib	200136	EPHA2		nM
10114-999-3	Pazopanib	200137	EPHA3		nM
10114-999-3	Pazopanib	200138	EPHA4		nM
10114-999-3	Pazopanib	200139	EPHA5		nM
10114-999-3	Pazopanib	200140	EPHA6		nM
10114-999-3	Pazopanib	200141	EPHA7		nM
10114-999-3	Pazopanib	200142	EPHA8		nM
10114-999-3	Pazopanib	200143	EPHB1		nM
10114-999-3	Pazopanib	200144	EPHB2		nM
10114-999-3	Pazopanib	200145	EPHB3		nM
10114-999-3	Pazopanib	200146	EPHB4		nM
10114-999-3	Pazopanib	200147	EPHB6	81.0	nM
10114-999-3	Pazopanib	200148	ERBB2		nM
10114-999-3	Pazopanib	200149	ERBB3		nM
10114-999-3	Pazopanib	200150	ERBB4		nM
10114-999-3	Pazopanib	200151	MK03		nM
10114-999-3	Pazopanib	200152	MK01		nM
10114-999-3	Pazopanib	200153	ERK3		nM
10114-999-3	Pazopanib	200154	ERK4		nM
10114-999-3	Pazopanib	200155	ERK5		nM
10114-999-3	Pazopanib	200156	ERK8		nM
10114-999-3	Pazopanib	200157	ERN1		nM
10114-999-3	Pazopanib	200158	FAK1		nM
10114-999-3	Pazopanib	200159	FER	2700.0	nM
10114-999-3	Pazopanib	200160	FES	1400.0	nM
10114-999-3	Pazopanib	200161	FGFR1	990.0	nM
10114-999-3	Pazopanib	200162	FGFR2	210.0	nM
10114-999-3	Pazopanib	200163	FGFR3	740.0	nM
10114-999-3	Pazopanib	200164	FGFR3(G697C)	620.0	nM
10114-999-3	Pazopanib	200165	FGFR4	2800.0	nM
10114-999-3	Pazopanib	200166	FGR	1600.0	nM
10114-999-3	Pazopanib	200167	VGFR1	14.0	nM
10114-999-3	Pazopanib	200168	FLT3	1100.0	nM
10114-999-3	Pazopanib	200169	FLT3(D835H)	1100.0	nM
10114-999-3	Pazopanib	200170	FLT3(D835Y)	810.0	nM
10114-999-3	Pazopanib	200171	FLT3(ITD)	2500.0	nM
10114-999-3	Pazopanib	200172	FLT3(K663Q)	740.0	nM
10114-999-3	Pazopanib	200173	FLT3(N841I)	1600.0	nM
10114-999-3	Pazopanib	200174	FLT3(R834Q)	9600.0	nM
10114-999-3	Pazopanib	200175	FLT4	27.0	nM
10114-999-3	Pazopanib	200176	FRK	750.0	nM
10114-999-3	Pazopanib	200177	FYN	2700.0	nM
10114-999-3	Pazopanib	200178	GAK	200.0	nM
10114-999-3	Pazopanib	200179	GCN2(Kin.Dom.2,S808G)		nM
10114-999-3	Pazopanib	200180	GRK1		nM
10114-999-3	Pazopanib	200181	GRK4		nM
10114-999-3	Pazopanib	200182	GRK7		nM
10114-999-3	Pazopanib	200183	GSK3A		nM
10114-999-3	Pazopanib	200184	GSK3B		nM
10114-999-3	Pazopanib	200185	HCK	5700.0	nM
10114-999-3	Pazopanib	200186	HIPK1		nM
10114-999-3	Pazopanib	200187	HIPK2		nM
10114-999-3	Pazopanib	200188	HIPK3		nM
10114-999-3	Pazopanib	200189	HIPK4		nM
10114-999-3	Pazopanib	200190	M4K1	750.0	nM
10114-999-3	Pazopanib	200191	HUNK		nM
10114-999-3	Pazopanib	200192	ICK		nM
10114-999-3	Pazopanib	200193	IGF1R		nM
10114-999-3	Pazopanib	200194	IKKA		nM
10114-999-3	Pazopanib	200195	IKKB		nM
10114-999-3	Pazopanib	200196	IKKE		nM
10114-999-3	Pazopanib	200197	INSR		nM
10114-999-3	Pazopanib	200198	INSRR		nM
10114-999-3	Pazopanib	200199	IRAK1	5900.0	nM
10114-999-3	Pazopanib	200200	IRAK3	800.0	nM
10114-999-3	Pazopanib	200201	IRAK4		nM
10114-999-3	Pazopanib	200202	ITK		nM
10114-999-3	Pazopanib	200203	JAK1(JH1domain-catalytic)		nM
10114-999-3	Pazopanib	200204	JAK1(JH2domain-pseudokinase)		nM
10114-999-3	Pazopanib	200207	JAK2(JH1domain-catalytic)	1700.0	nM
10114-999-3	Pazopanib	200209	JAK3(JH1domain-catalytic)	6900.0	nM
10114-999-3	Pazopanib	200211	JNK1	2000.0	nM
10114-999-3	Pazopanib	200212	MK09		nM
10114-999-3	Pazopanib	200213	JNK3	1900.0	nM
10114-999-3	Pazopanib	200214	KIT	2.8	nM
10114-999-3	Pazopanib	200215	KIT(A829P)	33.0	nM
10114-999-3	Pazopanib	200216	KIT(D816H)	1000.0	nM
10114-999-3	Pazopanib	200217	KIT(D816V)	500.0	nM
10114-999-3	Pazopanib	200218	KIT(L576P)	1.8	nM
10114-999-3	Pazopanib	200219	KIT(V559D)	2.3	nM
10114-999-3	Pazopanib	200220	KIT(V559D,T670I)	6.5	nM
10114-999-3	Pazopanib	200221	KIT(V559D,V654A)	30.0	nM
10114-999-3	Pazopanib	200222	LATS1		nM
10114-999-3	Pazopanib	200223	LATS2		nM
10114-999-3	Pazopanib	200224	LCK	1200.0	nM
10114-999-3	Pazopanib	200225	LIMK1	720.0	nM
10114-999-3	Pazopanib	200226	LIMK2	390.0	nM
10114-999-3	Pazopanib	200227	LKB1		nM
10114-999-3	Pazopanib	200228	LOK	84.0	nM
10114-999-3	Pazopanib	200229	LRRK2		nM
10114-999-3	Pazopanib	200230	LRRK2(G2019S)		nM
10114-999-3	Pazopanib	200231	LTK	6800.0	nM
10114-999-3	Pazopanib	200232	LYN	1100.0	nM
10114-999-3	Pazopanib	200233	M3K13		nM
10114-999-3	Pazopanib	200234	MAK		nM
10114-999-3	Pazopanib	200235	MAP3K1	2900.0	nM
10114-999-3	Pazopanib	200236	MAP3K15		nM
10114-999-3	Pazopanib	200237	M3K2	290.0	nM
10114-999-3	Pazopanib	200238	MAP3K3		nM
10114-999-3	Pazopanib	200239	MAP3K4		nM
10114-999-3	Pazopanib	200240	MAP4K2	2700.0	nM
10114-999-3	Pazopanib	200241	M4K3	1600.0	nM
10114-999-3	Pazopanib	200242	MAP4K4	2200.0	nM
10114-999-3	Pazopanib	200243	MAP4K5	3000.0	nM
10114-999-3	Pazopanib	200244	MAPKAPK2		nM
10114-999-3	Pazopanib	200245	MAPKAPK5		nM
10114-999-3	Pazopanib	200246	MARK1		nM
10114-999-3	Pazopanib	200247	MARK2		nM
10114-999-3	Pazopanib	200248	MARK3	4000.0	nM
10114-999-3	Pazopanib	200249	MARK4		nM
10114-999-3	Pazopanib	200250	MAST1		nM
10114-999-3	Pazopanib	200251	MP2K1		nM
10114-999-3	Pazopanib	200252	MP2K2		nM
10114-999-3	Pazopanib	200253	MP2K3		nM
10114-999-3	Pazopanib	200254	MP2K4	590.0	nM
10114-999-3	Pazopanib	200255	MP2K5	480.0	nM
10114-999-3	Pazopanib	200256	MP2K6	4100.0	nM
10114-999-3	Pazopanib	200257	MELK		nM
10114-999-3	Pazopanib	200258	MERTK	3300.0	nM
10114-999-3	Pazopanib	200259	MET	2000.0	nM
10114-999-3	Pazopanib	200260	MET(M1250T)	3400.0	nM
10114-999-3	Pazopanib	200261	MET(Y1235D)	2100.0	nM
10114-999-3	Pazopanib	200262	MINK		nM
10114-999-3	Pazopanib	200263	MP2K7		nM
10114-999-3	Pazopanib	200264	MKNK1		nM
10114-999-3	Pazopanib	200265	MKNK2		nM
10114-999-3	Pazopanib	200266	MLCK		nM
10114-999-3	Pazopanib	200267	MLK1	290.0	nM
10114-999-3	Pazopanib	200268	MLK2	2100.0	nM
10114-999-3	Pazopanib	200269	MLK3	740.0	nM
10114-999-3	Pazopanib	200270	MRCKA		nM
10114-999-3	Pazopanib	200271	MRCKB		nM
10114-999-3	Pazopanib	200272	MST1		nM
10114-999-3	Pazopanib	200273	MST1R		nM
10114-999-3	Pazopanib	200274	MST2		nM
10114-999-3	Pazopanib	200275	MST3		nM
10114-999-3	Pazopanib	200276	MST4		nM
10114-999-3	Pazopanib	200277	MTOR		nM
10114-999-3	Pazopanib	200278	MUSK		nM
10114-999-3	Pazopanib	200279	MYLK		nM
10114-999-3	Pazopanib	200280	MYLK2	2000.0	nM
10114-999-3	Pazopanib	200281	MYLK4		nM
10114-999-3	Pazopanib	200282	MYO3A		nM
10114-999-3	Pazopanib	200283	MYO3B		nM
10114-999-3	Pazopanib	200284	NDR1		nM
10114-999-3	Pazopanib	200285	NDR2		nM
10114-999-3	Pazopanib	200286	NEK1		nM
10114-999-3	Pazopanib	200287	NEK11		nM
10114-999-3	Pazopanib	200288	NEK2	980.0	nM
10114-999-3	Pazopanib	200289	NEK3		nM
10114-999-3	Pazopanib	200290	NEK4		nM
10114-999-3	Pazopanib	200291	NEK5	7300.0	nM
10114-999-3	Pazopanib	200292	NEK6		nM
10114-999-3	Pazopanib	200293	NEK7		nM
10114-999-3	Pazopanib	200294	NEK9		nM
10114-999-3	Pazopanib	200295	NIM1		nM
10114-999-3	Pazopanib	200296	NLK	4400.0	nM
10114-999-3	Pazopanib	200297	OSR1		nM
10114-999-3	Pazopanib	200298	MK14		nM
10114-999-3	Pazopanib	200299	MK11		nM
10114-999-3	Pazopanib	200300	MK13		nM
10114-999-3	Pazopanib	200301	MK12		nM
10114-999-3	Pazopanib	200302	PAK1		nM
10114-999-3	Pazopanib	200303	PAK2		nM
10114-999-3	Pazopanib	200304	PAK3		nM
10114-999-3	Pazopanib	200305	PAK4		nM
10114-999-3	Pazopanib	200306	PAK6		nM
10114-999-3	Pazopanib	200307	PAK7		nM
10114-999-3	Pazopanib	200309	CDK16	1200.0	nM
10114-999-3	Pazopanib	200310	PCTK2		nM
10114-999-3	Pazopanib	200311	PCTK3		nM
10114-999-3	Pazopanib	200312	PGFRA	4.9	nM
10114-999-3	Pazopanib	200313	PGFRB	2.0	nM
10114-999-3	Pazopanib	200314	PDPK1		nM
10114-999-3	Pazopanib	200315	PFCDPK1(P.falciparum)	370.0	nM
10114-999-3	Pazopanib	200316	PFPK5(P.falciparum)		nM
10114-999-3	Pazopanib	200317	CDK15		nM
10114-999-3	Pazopanib	200318	CDK14		nM
10114-999-3	Pazopanib	200319	PHKG1		nM
10114-999-3	Pazopanib	200320	PHKG2		nM
10114-999-3	Pazopanib	200321	PIK3C2B		nM
10114-999-3	Pazopanib	200322	PIK3C2G		nM
10114-999-3	Pazopanib	200323	PIK3CA		nM
10114-999-3	Pazopanib	200324	PIK3CA(C420R)		nM
10114-999-3	Pazopanib	200325	PIK3CA(E542K)		nM
10114-999-3	Pazopanib	200326	PIK3CA(E545A)		nM
10114-999-3	Pazopanib	200327	PIK3CA(E545K)		nM
10114-999-3	Pazopanib	200328	PIK3CA(H1047L)		nM
10114-999-3	Pazopanib	200329	PIK3CA(H1047Y)		nM
10114-999-3	Pazopanib	200330	PIK3CA(I800L)		nM
10114-999-3	Pazopanib	200331	PIK3CA(M1043I)		nM
10114-999-3	Pazopanib	200332	PIK3CA(Q546K)		nM
10114-999-3	Pazopanib	200333	PIK3CB		nM
10114-999-3	Pazopanib	200334	PIK3CD		nM
10114-999-3	Pazopanib	200335	PIK3CG		nM
10114-999-3	Pazopanib	200336	PIK4CB	960.0	nM
10114-999-3	Pazopanib	200337	PIM1		nM
10114-999-3	Pazopanib	200338	PIM2		nM
10114-999-3	Pazopanib	200339	PIM3		nM
10114-999-3	Pazopanib	200340	PIP5K1A		nM
10114-999-3	Pazopanib	200341	PIP5K1C	1900.0	nM
10114-999-3	Pazopanib	200342	PIP5K2B		nM
10114-999-3	Pazopanib	200343	PI42C	280.0	nM
10114-999-3	Pazopanib	200344	PKAC-alpha		nM
10114-999-3	Pazopanib	200345	PKAC-beta		nM
10114-999-3	Pazopanib	200346	PKMYT1		nM
10114-999-3	Pazopanib	200347	PKN1		nM
10114-999-3	Pazopanib	200348	PKN2		nM
10114-999-3	Pazopanib	200349	PKNB(M.tuberculosis)		nM
10114-999-3	Pazopanib	200350	PLK1		nM
10114-999-3	Pazopanib	200351	PLK2		nM
10114-999-3	Pazopanib	200352	PLK3		nM
10114-999-3	Pazopanib	200353	PLK4	290.0	nM
10114-999-3	Pazopanib	200354	KPCD		nM
10114-999-3	Pazopanib	200355	KPCE		nM
10114-999-3	Pazopanib	200356	KPCL		nM
10114-999-3	Pazopanib	200357	KPCI		nM
10114-999-3	Pazopanib	200358	KPCT		nM
10114-999-3	Pazopanib	200359	KPCD1		nM
10114-999-3	Pazopanib	200360	KPCD2		nM
10114-999-3	Pazopanib	200361	KPCD3		nM
10114-999-3	Pazopanib	200362	KGP1		nM
10114-999-3	Pazopanib	200363	KGP2		nM
10114-999-3	Pazopanib	200364	PRKR	1900.0	nM
10114-999-3	Pazopanib	200365	PRKX		nM
10114-999-3	Pazopanib	200366	PRP4		nM
10114-999-3	Pazopanib	200367	FAK2		nM
10114-999-3	Pazopanib	200368	SIK3		nM
10114-999-3	Pazopanib	200369	RAF1	900.0	nM
10114-999-3	Pazopanib	200370	RET	310.0	nM
10114-999-3	Pazopanib	200371	RET(M918T)	270.0	nM
10114-999-3	Pazopanib	200372	RET(V804L)	5900.0	nM
10114-999-3	Pazopanib	200373	RET(V804M)	2300.0	nM
10114-999-3	Pazopanib	200374	RIOK1		nM
10114-999-3	Pazopanib	200375	RIOK2	610.0	nM
10114-999-3	Pazopanib	200376	RIOK3		nM
10114-999-3	Pazopanib	200377	RIPK1	260.0	nM
10114-999-3	Pazopanib	200378	RIPK2	580.0	nM
10114-999-3	Pazopanib	200379	RIPK4		nM
10114-999-3	Pazopanib	200380	RIPK5		nM
10114-999-3	Pazopanib	200381	ROCK1		nM
10114-999-3	Pazopanib	200382	ROCK2		nM
10114-999-3	Pazopanib	200383	ROS1	920.0	nM
10114-999-3	Pazopanib	200390	RPS6KA4(Kin.Dom.1-N-terminal)		nM
10114-999-3	Pazopanib	200392	RPS6KA4(Kin.Dom.2-C-terminal)		nM
10114-999-3	Pazopanib	200394	RPS6KA5(Kin.Dom.1-N-terminal)		nM
10114-999-3	Pazopanib	200396	RPS6KA5(Kin.Dom.2-C-terminal)		nM
10114-999-3	Pazopanib	200399	RSK1(Kin.Dom.1-N-terminal)		nM
10114-999-3	Pazopanib	200400	RSK1(Kin.Dom.2-C-terminal)		nM
10114-999-3	Pazopanib	200401	RSK2(Kin.Dom.1-N-terminal)		nM
10114-999-3	Pazopanib	200402	RSK3(Kin.Dom.1-N-terminal)		nM
10114-999-3	Pazopanib	200403	RSK3(Kin.Dom.2-C-terminal)		nM
10114-999-3	Pazopanib	200404	RSK4(Kin.Dom.1-N-terminal)		nM
10114-999-3	Pazopanib	200405	RSK4(Kin.Dom.2-C-terminal)		nM
10114-999-3	Pazopanib	200406	S6K1		nM
10114-999-3	Pazopanib	200407	SBK1		nM
10114-999-3	Pazopanib	200408	SgK110		nM
10114-999-3	Pazopanib	200409	SGK3		nM
10114-999-3	Pazopanib	200410	SIK1	2200.0	nM
10114-999-3	Pazopanib	200411	SIK2	7300.0	nM
10114-999-3	Pazopanib	200412	SLK	240.0	nM
10114-999-3	Pazopanib	200413	SNARK		nM
10114-999-3	Pazopanib	200414	SNRK		nM
10114-999-3	Pazopanib	200415	SRC	2800.0	nM
10114-999-3	Pazopanib	200416	SRMS	2500.0	nM
10114-999-3	Pazopanib	200417	SRPK1		nM
10114-999-3	Pazopanib	200418	SRPK2		nM
10114-999-3	Pazopanib	200419	SRPK3		nM
10114-999-3	Pazopanib	200420	STK16	360.0	nM
10114-999-3	Pazopanib	200421	STK33		nM
10114-999-3	Pazopanib	200422	STK35		nM
10114-999-3	Pazopanib	200423	STK36	470.0	nM
10114-999-3	Pazopanib	200424	STK39		nM
10114-999-3	Pazopanib	200425	SYK	4700.0	nM
10114-999-3	Pazopanib	200426	TAK1		nM
10114-999-3	Pazopanib	200427	TAOK1	240.0	nM
10114-999-3	Pazopanib	200428	TAOK2	1800.0	nM
10114-999-3	Pazopanib	200429	TAOK3	45.0	nM
10114-999-3	Pazopanib	200430	TBK1		nM
10114-999-3	Pazopanib	200431	TEC		nM
10114-999-3	Pazopanib	200432	TESK1		nM
10114-999-3	Pazopanib	200433	TGFBR1		nM
10114-999-3	Pazopanib	200434	TGFBR2	3000.0	nM
10114-999-3	Pazopanib	200435	TIE1	700.0	nM
10114-999-3	Pazopanib	200436	TIE2	3300.0	nM
10114-999-3	Pazopanib	200437	TLK1		nM
10114-999-3	Pazopanib	200438	TLK2		nM
10114-999-3	Pazopanib	200439	TNIK	310.0	nM
10114-999-3	Pazopanib	200440	TNK1		nM
10114-999-3	Pazopanib	200441	TNK2		nM
10114-999-3	Pazopanib	200442	TNNI3K		nM
10114-999-3	Pazopanib	200443	TRKA		nM
10114-999-3	Pazopanib	200444	TRKB		nM
10114-999-3	Pazopanib	200445	TRKC		nM
10114-999-3	Pazopanib	200446	TRPM6		nM
10114-999-3	Pazopanib	200447	TSSK1		nM
10114-999-3	Pazopanib	200448	TTK	150.0	nM
10114-999-3	Pazopanib	200449	TXK	2600.0	nM
10114-999-3	Pazopanib	200450	TYK2(JH1domain-catalytic)	3400.0	nM
10114-999-3	Pazopanib	200451	TYK2(JH2domain-pseudokinase)		nM
10114-999-3	Pazopanib	200454	TYRO3		nM
10114-999-3	Pazopanib	200455	ULK1		nM
10114-999-3	Pazopanib	200456	ULK2		nM
10114-999-3	Pazopanib	200457	ULK3		nM
10114-999-3	Pazopanib	200458	VGFR2	14.0	nM
10114-999-3	Pazopanib	200459	VRK2		nM
10114-999-3	Pazopanib	200460	WEE1		nM
10114-999-3	Pazopanib	200461	WEE2		nM
10114-999-3	Pazopanib	200462	YANK1		nM
10114-999-3	Pazopanib	200463	YANK2		nM
10114-999-3	Pazopanib	200464	YANK3		nM
10114-999-3	Pazopanib	200465	YES	5000.0	nM
10114-999-3	Pazopanib	200466	YSK1		nM
10114-999-3	Pazopanib	200467	YSK4	940.0	nM
10114-999-3	Pazopanib	200468	MLTK		nM
10114-999-3	Pazopanib	200469	ZAP70		nM
