Small Molecule HMS LINCS ID	Small Molecule Name	Protein HMS LINCS ID	Protein Name	Kd	Conc unit
10067-999-4	Barasertib	200001	AAK1	3000.0	nM
10067-999-4	Barasertib	200004	ABL1(E255K)-phosphorylated	9600.0	nM
10067-999-4	Barasertib	200006	ABL1(F317I)-nonphosphorylated	3800.0	nM
10067-999-4	Barasertib	200007	ABL1(F317I)-phosphorylated	4600.0	nM
10067-999-4	Barasertib	200009	ABL1(F317L)-nonphosphorylated	1400.0	nM
10067-999-4	Barasertib	200010	ABL1(F317L)-phosphorylated	2300.0	nM
10067-999-4	Barasertib	200012	ABL1(H396P)-nonphosphorylated	1200.0	nM
10067-999-4	Barasertib	200013	ABL1(H396P)-phosphorylated		nM
10067-999-4	Barasertib	200015	ABL1(M351T)-phosphorylated	2200.0	nM
10067-999-4	Barasertib	200017	ABL1(Q252H)-nonphosphorylated	860.0	nM
10067-999-4	Barasertib	200018	ABL1(Q252H)-phosphorylated	6800.0	nM
10067-999-4	Barasertib	200020	ABL1(T315I)-nonphosphorylated	1100.0	nM
10067-999-4	Barasertib	200021	ABL1(T315I)-phosphorylated	4800.0	nM
10067-999-4	Barasertib	200023	ABL1(Y253F)-phosphorylated	3800.0	nM
10067-999-4	Barasertib	200024	ABL1-nonphosphorylated	1500.0	nM
10067-999-4	Barasertib	200025	ABL1-phosphorylated	5500.0	nM
10067-999-4	Barasertib	200026	ABL2		nM
10067-999-4	Barasertib	200027	ACVR1		nM
10067-999-4	Barasertib	200028	ACVR1B		nM
10067-999-4	Barasertib	200029	ACVR2A		nM
10067-999-4	Barasertib	200030	ACVR2B		nM
10067-999-4	Barasertib	200031	ACVRL1		nM
10067-999-4	Barasertib	200032	ADCK3		nM
10067-999-4	Barasertib	200033	ADCK4		nM
10067-999-4	Barasertib	200034	AKT1		nM
10067-999-4	Barasertib	200035	AKT2		nM
10067-999-4	Barasertib	200036	AKT3		nM
10067-999-4	Barasertib	200037	ALK		nM
10067-999-4	Barasertib	200038	AMPK-alpha1		nM
10067-999-4	Barasertib	200039	AMPK-alpha2		nM
10067-999-4	Barasertib	200040	ANKK1	1500.0	nM
10067-999-4	Barasertib	200041	NUAK1		nM
10067-999-4	Barasertib	200042	M3K5		nM
10067-999-4	Barasertib	200043	M3K6		nM
10067-999-4	Barasertib	200044	AURKA	400.0	nM
10067-999-4	Barasertib	200045	AURKB	4.6	nM
10067-999-4	Barasertib	200046	AURKC	4.4	nM
10067-999-4	Barasertib	200047	AXL	390.0	nM
10067-999-4	Barasertib	200048	BIKE		nM
10067-999-4	Barasertib	200049	BLK	1500.0	nM
10067-999-4	Barasertib	200050	BMPR1A		nM
10067-999-4	Barasertib	200051	BMPR1B		nM
10067-999-4	Barasertib	200052	BMPR2		nM
10067-999-4	Barasertib	200053	BMX		nM
10067-999-4	Barasertib	200054	BRAF		nM
10067-999-4	Barasertib	200055	BRAF(V600E)		nM
10067-999-4	Barasertib	200056	PTK6		nM
10067-999-4	Barasertib	200057	BRSK1		nM
10067-999-4	Barasertib	200058	BRSK2		nM
10067-999-4	Barasertib	200059	BTK	1200.0	nM
10067-999-4	Barasertib	200060	CAMK1		nM
10067-999-4	Barasertib	200061	CAMK1D		nM
10067-999-4	Barasertib	200062	CAMK1G		nM
10067-999-4	Barasertib	200063	CAMK2A		nM
10067-999-4	Barasertib	200064	CAMK2B		nM
10067-999-4	Barasertib	200065	KCC2D		nM
10067-999-4	Barasertib	200066	CAMK2G		nM
10067-999-4	Barasertib	200067	KCC4		nM
10067-999-4	Barasertib	200068	KKCC1		nM
10067-999-4	Barasertib	200069	CAMKK2		nM
10067-999-4	Barasertib	200070	CASK		nM
10067-999-4	Barasertib	200071	CDC2L1	1200.0	nM
10067-999-4	Barasertib	200072	CDC2L2	1000.0	nM
10067-999-4	Barasertib	200073	CDC2L5	1100.0	nM
10067-999-4	Barasertib	200074	CDK11		nM
10067-999-4	Barasertib	200075	CDK2		nM
10067-999-4	Barasertib	200076	CDK3		nM
10067-999-4	Barasertib	200077	CDK4-cyclinD1		nM
10067-999-4	Barasertib	200078	CDK4-cyclinD3		nM
10067-999-4	Barasertib	200079	CDK5		nM
10067-999-4	Barasertib	200080	CDK7	6200.0	nM
10067-999-4	Barasertib	200081	CDK8		nM
10067-999-4	Barasertib	200082	CDK9		nM
10067-999-4	Barasertib	200083	CDKL1		nM
10067-999-4	Barasertib	200084	CDKL2	1200.0	nM
10067-999-4	Barasertib	200085	CDKL3		nM
10067-999-4	Barasertib	200086	CDKL5		nM
10067-999-4	Barasertib	200087	CHEK1		nM
10067-999-4	Barasertib	200088	CHK2	1400.0	nM
10067-999-4	Barasertib	200089	CIT	5700.0	nM
10067-999-4	Barasertib	200090	CLK1		nM
10067-999-4	Barasertib	200091	CLK2		nM
10067-999-4	Barasertib	200092	CLK3		nM
10067-999-4	Barasertib	200093	CLK4		nM
10067-999-4	Barasertib	200094	CSF1R	1400.0	nM
10067-999-4	Barasertib	200095	CSK	3800.0	nM
10067-999-4	Barasertib	200096	CSNK1A1		nM
10067-999-4	Barasertib	200097	CSNK1A1L		nM
10067-999-4	Barasertib	200098	CSNK1D		nM
10067-999-4	Barasertib	200099	CSNK1E		nM
10067-999-4	Barasertib	200100	KC1G1		nM
10067-999-4	Barasertib	200101	KC1G2		nM
10067-999-4	Barasertib	200102	CSNK1G3		nM
10067-999-4	Barasertib	200103	CSNK2A1		nM
10067-999-4	Barasertib	200104	CSNK2A2		nM
10067-999-4	Barasertib	200105	CTK		nM
10067-999-4	Barasertib	200106	DAPK1		nM
10067-999-4	Barasertib	200107	DAPK2		nM
10067-999-4	Barasertib	200108	DAPK3		nM
10067-999-4	Barasertib	200109	DCLK1		nM
10067-999-4	Barasertib	200110	DCAMKL2		nM
10067-999-4	Barasertib	200111	DCAMKL3		nM
10067-999-4	Barasertib	200112	DDR1	1800.0	nM
10067-999-4	Barasertib	200113	DDR2	6600.0	nM
10067-999-4	Barasertib	200114	M3K12		nM
10067-999-4	Barasertib	200115	DMPK		nM
10067-999-4	Barasertib	200116	DMPK2		nM
10067-999-4	Barasertib	200117	DRAK1		nM
10067-999-4	Barasertib	200118	DRAK2		nM
10067-999-4	Barasertib	200119	DYRK1A		nM
10067-999-4	Barasertib	200120	DYRK1B		nM
10067-999-4	Barasertib	200121	DYRK2		nM
10067-999-4	Barasertib	200122	EGFR	450.0	nM
10067-999-4	Barasertib	200123	EGFR(E746-A750del)		nM
10067-999-4	Barasertib	200124	EGFR(G719C)	120.0	nM
10067-999-4	Barasertib	200125	EGFR(G719S)	170.0	nM
10067-999-4	Barasertib	200126	EGFR(L747-E749del, A750P)	2900.0	nM
10067-999-4	Barasertib	200127	EGFR(L747-S752del, P753S)	8800.0	nM
10067-999-4	Barasertib	200128	EGFR(L747-T751del,Sins)	3500.0	nM
10067-999-4	Barasertib	200129	EGFR(L858R)	980.0	nM
10067-999-4	Barasertib	200130	EGFR(L858R,T790M)		nM
10067-999-4	Barasertib	200131	EGFR(L861Q)	510.0	nM
10067-999-4	Barasertib	200132	EGFR(S752-I759del)	5200.0	nM
10067-999-4	Barasertib	200133	EGFR(T790M)	1500.0	nM
10067-999-4	Barasertib	200134	EIF2AK1	1500.0	nM
10067-999-4	Barasertib	200135	EPHA1		nM
10067-999-4	Barasertib	200136	EPHA2		nM
10067-999-4	Barasertib	200137	EPHA3		nM
10067-999-4	Barasertib	200138	EPHA4		nM
10067-999-4	Barasertib	200139	EPHA5		nM
10067-999-4	Barasertib	200140	EPHA6		nM
10067-999-4	Barasertib	200141	EPHA7		nM
10067-999-4	Barasertib	200142	EPHA8		nM
10067-999-4	Barasertib	200143	EPHB1		nM
10067-999-4	Barasertib	200144	EPHB2		nM
10067-999-4	Barasertib	200145	EPHB3		nM
10067-999-4	Barasertib	200146	EPHB4		nM
10067-999-4	Barasertib	200147	EPHB6	50.0	nM
10067-999-4	Barasertib	200148	ERBB2	4300.0	nM
10067-999-4	Barasertib	200149	ERBB3		nM
10067-999-4	Barasertib	200150	ERBB4	470.0	nM
10067-999-4	Barasertib	200151	MK03		nM
10067-999-4	Barasertib	200152	MK01		nM
10067-999-4	Barasertib	200153	ERK3		nM
10067-999-4	Barasertib	200154	ERK4		nM
10067-999-4	Barasertib	200155	ERK5		nM
10067-999-4	Barasertib	200156	ERK8		nM
10067-999-4	Barasertib	200157	ERN1		nM
10067-999-4	Barasertib	200158	FAK1		nM
10067-999-4	Barasertib	200159	FER		nM
10067-999-4	Barasertib	200160	FES		nM
10067-999-4	Barasertib	200161	FGFR1		nM
10067-999-4	Barasertib	200162	FGFR2		nM
10067-999-4	Barasertib	200163	FGFR3		nM
10067-999-4	Barasertib	200164	FGFR3(G697C)		nM
10067-999-4	Barasertib	200165	FGFR4		nM
10067-999-4	Barasertib	200166	FGR		nM
10067-999-4	Barasertib	200167	VGFR1	110.0	nM
10067-999-4	Barasertib	200168	FLT3	8.2	nM
10067-999-4	Barasertib	200169	FLT3(D835H)	210.0	nM
10067-999-4	Barasertib	200170	FLT3(D835Y)	670.0	nM
10067-999-4	Barasertib	200171	FLT3(ITD)	140.0	nM
10067-999-4	Barasertib	200172	FLT3(K663Q)	3.9	nM
10067-999-4	Barasertib	200173	FLT3(N841I)	43.0	nM
10067-999-4	Barasertib	200174	FLT3(R834Q)	130.0	nM
10067-999-4	Barasertib	200175	FLT4	2900.0	nM
10067-999-4	Barasertib	200176	FRK		nM
10067-999-4	Barasertib	200177	FYN		nM
10067-999-4	Barasertib	200178	GAK		nM
10067-999-4	Barasertib	200179	GCN2(Kin.Dom.2,S808G)		nM
10067-999-4	Barasertib	200180	GRK1		nM
10067-999-4	Barasertib	200181	GRK4		nM
10067-999-4	Barasertib	200182	GRK7		nM
10067-999-4	Barasertib	200183	GSK3A		nM
10067-999-4	Barasertib	200184	GSK3B		nM
10067-999-4	Barasertib	200185	HCK	3900.0	nM
10067-999-4	Barasertib	200186	HIPK1		nM
10067-999-4	Barasertib	200187	HIPK2	3700.0	nM
10067-999-4	Barasertib	200188	HIPK3	2500.0	nM
10067-999-4	Barasertib	200189	HIPK4	97.0	nM
10067-999-4	Barasertib	200190	M4K1		nM
10067-999-4	Barasertib	200191	HUNK		nM
10067-999-4	Barasertib	200192	ICK		nM
10067-999-4	Barasertib	200193	IGF1R		nM
10067-999-4	Barasertib	200194	IKKA		nM
10067-999-4	Barasertib	200195	IKKB		nM
10067-999-4	Barasertib	200196	IKKE		nM
10067-999-4	Barasertib	200197	INSR		nM
10067-999-4	Barasertib	200198	INSRR		nM
10067-999-4	Barasertib	200199	IRAK1		nM
10067-999-4	Barasertib	200200	IRAK3	7900.0	nM
10067-999-4	Barasertib	200201	IRAK4		nM
10067-999-4	Barasertib	200202	ITK		nM
10067-999-4	Barasertib	200203	JAK1(JH1domain-catalytic)		nM
10067-999-4	Barasertib	200204	JAK1(JH2domain-pseudokinase)		nM
10067-999-4	Barasertib	200207	JAK2(JH1domain-catalytic)		nM
10067-999-4	Barasertib	200209	JAK3(JH1domain-catalytic)		nM
10067-999-4	Barasertib	200211	JNK1		nM
10067-999-4	Barasertib	200212	MK09		nM
10067-999-4	Barasertib	200213	JNK3		nM
10067-999-4	Barasertib	200214	KIT	17.0	nM
10067-999-4	Barasertib	200215	KIT(A829P)	600.0	nM
10067-999-4	Barasertib	200216	KIT(D816H)	2900.0	nM
10067-999-4	Barasertib	200217	KIT(D816V)	4600.0	nM
10067-999-4	Barasertib	200218	KIT(L576P)	34.0	nM
10067-999-4	Barasertib	200219	KIT(V559D)	15.0	nM
10067-999-4	Barasertib	200220	KIT(V559D,T670I)	7.9	nM
10067-999-4	Barasertib	200221	KIT(V559D,V654A)	480.0	nM
10067-999-4	Barasertib	200222	LATS1		nM
10067-999-4	Barasertib	200223	LATS2		nM
10067-999-4	Barasertib	200224	LCK	380.0	nM
10067-999-4	Barasertib	200225	LIMK1		nM
10067-999-4	Barasertib	200226	LIMK2		nM
10067-999-4	Barasertib	200227	LKB1		nM
10067-999-4	Barasertib	200228	LOK	2800.0	nM
10067-999-4	Barasertib	200229	LRRK2		nM
10067-999-4	Barasertib	200230	LRRK2(G2019S)		nM
10067-999-4	Barasertib	200231	LTK	3200.0	nM
10067-999-4	Barasertib	200232	LYN	1600.0	nM
10067-999-4	Barasertib	200233	M3K13		nM
10067-999-4	Barasertib	200234	MAK		nM
10067-999-4	Barasertib	200235	MAP3K1		nM
10067-999-4	Barasertib	200236	MAP3K15		nM
10067-999-4	Barasertib	200237	M3K2		nM
10067-999-4	Barasertib	200238	MAP3K3		nM
10067-999-4	Barasertib	200239	MAP3K4		nM
10067-999-4	Barasertib	200240	MAP4K2		nM
10067-999-4	Barasertib	200241	M4K3		nM
10067-999-4	Barasertib	200242	MAP4K4		nM
10067-999-4	Barasertib	200243	MAP4K5	160.0	nM
10067-999-4	Barasertib	200244	MAPKAPK2		nM
10067-999-4	Barasertib	200245	MAPKAPK5		nM
10067-999-4	Barasertib	200246	MARK1		nM
10067-999-4	Barasertib	200247	MARK2		nM
10067-999-4	Barasertib	200248	MARK3		nM
10067-999-4	Barasertib	200249	MARK4		nM
10067-999-4	Barasertib	200250	MAST1		nM
10067-999-4	Barasertib	200251	MP2K1	1900.0	nM
10067-999-4	Barasertib	200252	MP2K2	4200.0	nM
10067-999-4	Barasertib	200253	MP2K3		nM
10067-999-4	Barasertib	200254	MP2K4		nM
10067-999-4	Barasertib	200255	MP2K5	2.8	nM
10067-999-4	Barasertib	200256	MP2K6		nM
10067-999-4	Barasertib	200257	MELK		nM
10067-999-4	Barasertib	200258	MERTK		nM
10067-999-4	Barasertib	200259	MET		nM
10067-999-4	Barasertib	200260	MET(M1250T)		nM
10067-999-4	Barasertib	200261	MET(Y1235D)	5700.0	nM
10067-999-4	Barasertib	200262	MINK		nM
10067-999-4	Barasertib	200263	MP2K7		nM
10067-999-4	Barasertib	200264	MKNK1		nM
10067-999-4	Barasertib	200265	MKNK2	1200.0	nM
10067-999-4	Barasertib	200266	MLCK		nM
10067-999-4	Barasertib	200267	MLK1		nM
10067-999-4	Barasertib	200268	MLK2		nM
10067-999-4	Barasertib	200269	MLK3		nM
10067-999-4	Barasertib	200270	MRCKA		nM
10067-999-4	Barasertib	200271	MRCKB		nM
10067-999-4	Barasertib	200272	MST1		nM
10067-999-4	Barasertib	200273	MST1R		nM
10067-999-4	Barasertib	200274	MST2		nM
10067-999-4	Barasertib	200275	MST3		nM
10067-999-4	Barasertib	200276	MST4		nM
10067-999-4	Barasertib	200277	MTOR		nM
10067-999-4	Barasertib	200278	MUSK	1500.0	nM
10067-999-4	Barasertib	200279	MYLK		nM
10067-999-4	Barasertib	200280	MYLK2		nM
10067-999-4	Barasertib	200281	MYLK4		nM
10067-999-4	Barasertib	200282	MYO3A		nM
10067-999-4	Barasertib	200283	MYO3B		nM
10067-999-4	Barasertib	200284	NDR1		nM
10067-999-4	Barasertib	200285	NDR2		nM
10067-999-4	Barasertib	200286	NEK1		nM
10067-999-4	Barasertib	200287	NEK11		nM
10067-999-4	Barasertib	200288	NEK2		nM
10067-999-4	Barasertib	200289	NEK3		nM
10067-999-4	Barasertib	200290	NEK4		nM
10067-999-4	Barasertib	200291	NEK5		nM
10067-999-4	Barasertib	200292	NEK6		nM
10067-999-4	Barasertib	200293	NEK7		nM
10067-999-4	Barasertib	200294	NEK9		nM
10067-999-4	Barasertib	200295	NIM1		nM
10067-999-4	Barasertib	200296	NLK		nM
10067-999-4	Barasertib	200297	OSR1		nM
10067-999-4	Barasertib	200298	MK14		nM
10067-999-4	Barasertib	200299	MK11		nM
10067-999-4	Barasertib	200300	MK13		nM
10067-999-4	Barasertib	200301	MK12		nM
10067-999-4	Barasertib	200302	PAK1		nM
10067-999-4	Barasertib	200303	PAK2		nM
10067-999-4	Barasertib	200304	PAK3		nM
10067-999-4	Barasertib	200305	PAK4		nM
10067-999-4	Barasertib	200306	PAK6		nM
10067-999-4	Barasertib	200307	PAK7		nM
10067-999-4	Barasertib	200309	CDK16	6300.0	nM
10067-999-4	Barasertib	200310	PCTK2		nM
10067-999-4	Barasertib	200311	PCTK3		nM
10067-999-4	Barasertib	200312	PGFRA	38.0	nM
10067-999-4	Barasertib	200313	PGFRB	41.0	nM
10067-999-4	Barasertib	200314	PDPK1		nM
10067-999-4	Barasertib	200315	PFCDPK1(P.falciparum)		nM
10067-999-4	Barasertib	200316	PFPK5(P.falciparum)		nM
10067-999-4	Barasertib	200317	CDK15		nM
10067-999-4	Barasertib	200318	CDK14		nM
10067-999-4	Barasertib	200319	PHKG1		nM
10067-999-4	Barasertib	200320	PHKG2		nM
10067-999-4	Barasertib	200321	PIK3C2B		nM
10067-999-4	Barasertib	200322	PIK3C2G		nM
10067-999-4	Barasertib	200323	PIK3CA		nM
10067-999-4	Barasertib	200324	PIK3CA(C420R)		nM
10067-999-4	Barasertib	200325	PIK3CA(E542K)		nM
10067-999-4	Barasertib	200326	PIK3CA(E545A)		nM
10067-999-4	Barasertib	200327	PIK3CA(E545K)		nM
10067-999-4	Barasertib	200328	PIK3CA(H1047L)		nM
10067-999-4	Barasertib	200329	PIK3CA(H1047Y)		nM
10067-999-4	Barasertib	200330	PIK3CA(I800L)		nM
10067-999-4	Barasertib	200331	PIK3CA(M1043I)		nM
10067-999-4	Barasertib	200332	PIK3CA(Q546K)		nM
10067-999-4	Barasertib	200333	PIK3CB		nM
10067-999-4	Barasertib	200334	PIK3CD		nM
10067-999-4	Barasertib	200335	PIK3CG		nM
10067-999-4	Barasertib	200336	PIK4CB		nM
10067-999-4	Barasertib	200337	PIM1		nM
10067-999-4	Barasertib	200338	PIM2		nM
10067-999-4	Barasertib	200339	PIM3		nM
10067-999-4	Barasertib	200340	PIP5K1A		nM
10067-999-4	Barasertib	200341	PIP5K1C		nM
10067-999-4	Barasertib	200342	PIP5K2B		nM
10067-999-4	Barasertib	200343	PI42C		nM
10067-999-4	Barasertib	200344	PKAC-alpha		nM
10067-999-4	Barasertib	200345	PKAC-beta		nM
10067-999-4	Barasertib	200346	PKMYT1		nM
10067-999-4	Barasertib	200347	PKN1		nM
10067-999-4	Barasertib	200348	PKN2		nM
10067-999-4	Barasertib	200349	PKNB(M.tuberculosis)		nM
10067-999-4	Barasertib	200350	PLK1		nM
10067-999-4	Barasertib	200351	PLK2		nM
10067-999-4	Barasertib	200352	PLK3		nM
10067-999-4	Barasertib	200353	PLK4	4700.0	nM
10067-999-4	Barasertib	200354	KPCD		nM
10067-999-4	Barasertib	200355	KPCE		nM
10067-999-4	Barasertib	200356	KPCL		nM
10067-999-4	Barasertib	200357	KPCI		nM
10067-999-4	Barasertib	200358	KPCT		nM
10067-999-4	Barasertib	200359	KPCD1		nM
10067-999-4	Barasertib	200360	KPCD2		nM
10067-999-4	Barasertib	200361	KPCD3		nM
10067-999-4	Barasertib	200362	KGP1		nM
10067-999-4	Barasertib	200363	KGP2		nM
10067-999-4	Barasertib	200364	PRKR		nM
10067-999-4	Barasertib	200365	PRKX		nM
10067-999-4	Barasertib	200366	PRP4		nM
10067-999-4	Barasertib	200367	FAK2		nM
10067-999-4	Barasertib	200368	SIK3		nM
10067-999-4	Barasertib	200369	RAF1		nM
10067-999-4	Barasertib	200370	RET	80.0	nM
10067-999-4	Barasertib	200371	RET(M918T)	120.0	nM
10067-999-4	Barasertib	200372	RET(V804L)	140.0	nM
10067-999-4	Barasertib	200373	RET(V804M)	240.0	nM
10067-999-4	Barasertib	200374	RIOK1		nM
10067-999-4	Barasertib	200375	RIOK2		nM
10067-999-4	Barasertib	200376	RIOK3		nM
10067-999-4	Barasertib	200377	RIPK1		nM
10067-999-4	Barasertib	200378	RIPK2	1800.0	nM
10067-999-4	Barasertib	200379	RIPK4		nM
10067-999-4	Barasertib	200380	RIPK5	3000.0	nM
10067-999-4	Barasertib	200381	ROCK1		nM
10067-999-4	Barasertib	200382	ROCK2		nM
10067-999-4	Barasertib	200383	ROS1		nM
10067-999-4	Barasertib	200390	RPS6KA4(Kin.Dom.1-N-terminal)		nM
10067-999-4	Barasertib	200392	RPS6KA4(Kin.Dom.2-C-terminal)		nM
10067-999-4	Barasertib	200394	RPS6KA5(Kin.Dom.1-N-terminal)		nM
10067-999-4	Barasertib	200396	RPS6KA5(Kin.Dom.2-C-terminal)		nM
10067-999-4	Barasertib	200399	RSK1(Kin.Dom.1-N-terminal)		nM
10067-999-4	Barasertib	200400	RSK1(Kin.Dom.2-C-terminal)		nM
10067-999-4	Barasertib	200401	RSK2(Kin.Dom.1-N-terminal)		nM
10067-999-4	Barasertib	200402	RSK3(Kin.Dom.1-N-terminal)		nM
10067-999-4	Barasertib	200403	RSK3(Kin.Dom.2-C-terminal)		nM
10067-999-4	Barasertib	200404	RSK4(Kin.Dom.1-N-terminal)		nM
10067-999-4	Barasertib	200405	RSK4(Kin.Dom.2-C-terminal)		nM
10067-999-4	Barasertib	200406	S6K1	2800.0	nM
10067-999-4	Barasertib	200407	SBK1		nM
10067-999-4	Barasertib	200408	SgK110		nM
10067-999-4	Barasertib	200409	SGK3		nM
10067-999-4	Barasertib	200410	SIK1		nM
10067-999-4	Barasertib	200411	SIK2		nM
10067-999-4	Barasertib	200412	SLK		nM
10067-999-4	Barasertib	200413	SNARK		nM
10067-999-4	Barasertib	200414	SNRK		nM
10067-999-4	Barasertib	200415	SRC		nM
10067-999-4	Barasertib	200416	SRMS	7900.0	nM
10067-999-4	Barasertib	200417	SRPK1		nM
10067-999-4	Barasertib	200418	SRPK2		nM
10067-999-4	Barasertib	200419	SRPK3		nM
10067-999-4	Barasertib	200420	STK16		nM
10067-999-4	Barasertib	200421	STK33		nM
10067-999-4	Barasertib	200422	STK35		nM
10067-999-4	Barasertib	200423	STK36	4600.0	nM
10067-999-4	Barasertib	200424	STK39		nM
10067-999-4	Barasertib	200425	SYK		nM
10067-999-4	Barasertib	200426	TAK1	650.0	nM
10067-999-4	Barasertib	200427	TAOK1		nM
10067-999-4	Barasertib	200428	TAOK2		nM
10067-999-4	Barasertib	200429	TAOK3		nM
10067-999-4	Barasertib	200430	TBK1		nM
10067-999-4	Barasertib	200431	TEC		nM
10067-999-4	Barasertib	200432	TESK1		nM
10067-999-4	Barasertib	200433	TGFBR1		nM
10067-999-4	Barasertib	200434	TGFBR2		nM
10067-999-4	Barasertib	200435	TIE1	350.0	nM
10067-999-4	Barasertib	200436	TIE2	1900.0	nM
10067-999-4	Barasertib	200437	TLK1		nM
10067-999-4	Barasertib	200438	TLK2		nM
10067-999-4	Barasertib	200439	TNIK	8500.0	nM
10067-999-4	Barasertib	200440	TNK1		nM
10067-999-4	Barasertib	200441	TNK2		nM
10067-999-4	Barasertib	200442	TNNI3K		nM
10067-999-4	Barasertib	200443	TRKA		nM
10067-999-4	Barasertib	200444	TRKB		nM
10067-999-4	Barasertib	200445	TRKC		nM
10067-999-4	Barasertib	200446	TRPM6		nM
10067-999-4	Barasertib	200447	TSSK1		nM
10067-999-4	Barasertib	200448	TTK	8500.0	nM
10067-999-4	Barasertib	200449	TXK		nM
10067-999-4	Barasertib	200450	TYK2(JH1domain-catalytic)		nM
10067-999-4	Barasertib	200451	TYK2(JH2domain-pseudokinase)		nM
10067-999-4	Barasertib	200454	TYRO3		nM
10067-999-4	Barasertib	200455	ULK1		nM
10067-999-4	Barasertib	200456	ULK2		nM
10067-999-4	Barasertib	200457	ULK3		nM
10067-999-4	Barasertib	200458	VGFR2	500.0	nM
10067-999-4	Barasertib	200459	VRK2		nM
10067-999-4	Barasertib	200460	WEE1		nM
10067-999-4	Barasertib	200461	WEE2		nM
10067-999-4	Barasertib	200462	YANK1		nM
10067-999-4	Barasertib	200463	YANK2		nM
10067-999-4	Barasertib	200464	YANK3		nM
10067-999-4	Barasertib	200465	YES	3800.0	nM
10067-999-4	Barasertib	200466	YSK1		nM
10067-999-4	Barasertib	200467	YSK4	2400.0	nM
10067-999-4	Barasertib	200468	MLTK	1700.0	nM
10067-999-4	Barasertib	200469	ZAP70		nM
