Small Molecule HMS LINCS ID	Small Molecule Name	Protein HMS LINCS ID	Protein Name	Kd	Conc unit
10051-999-6	Lapatinib	200001	AAK1		nM
10051-999-6	Lapatinib	200004	ABL1(E255K)-phosphorylated		nM
10051-999-6	Lapatinib	200006	ABL1(F317I)-nonphosphorylated		nM
10051-999-6	Lapatinib	200007	ABL1(F317I)-phosphorylated		nM
10051-999-6	Lapatinib	200009	ABL1(F317L)-nonphosphorylated		nM
10051-999-6	Lapatinib	200010	ABL1(F317L)-phosphorylated		nM
10051-999-6	Lapatinib	200012	ABL1(H396P)-nonphosphorylated		nM
10051-999-6	Lapatinib	200013	ABL1(H396P)-phosphorylated		nM
10051-999-6	Lapatinib	200015	ABL1(M351T)-phosphorylated		nM
10051-999-6	Lapatinib	200017	ABL1(Q252H)-nonphosphorylated		nM
10051-999-6	Lapatinib	200018	ABL1(Q252H)-phosphorylated		nM
10051-999-6	Lapatinib	200020	ABL1(T315I)-nonphosphorylated		nM
10051-999-6	Lapatinib	200021	ABL1(T315I)-phosphorylated		nM
10051-999-6	Lapatinib	200023	ABL1(Y253F)-phosphorylated		nM
10051-999-6	Lapatinib	200024	ABL1-nonphosphorylated		nM
10051-999-6	Lapatinib	200025	ABL1-phosphorylated		nM
10051-999-6	Lapatinib	200026	ABL2		nM
10051-999-6	Lapatinib	200027	ACVR1		nM
10051-999-6	Lapatinib	200028	ACVR1B		nM
10051-999-6	Lapatinib	200029	ACVR2A		nM
10051-999-6	Lapatinib	200030	ACVR2B		nM
10051-999-6	Lapatinib	200031	ACVRL1		nM
10051-999-6	Lapatinib	200032	ADCK3		nM
10051-999-6	Lapatinib	200033	ADCK4		nM
10051-999-6	Lapatinib	200034	AKT1		nM
10051-999-6	Lapatinib	200035	AKT2		nM
10051-999-6	Lapatinib	200036	AKT3		nM
10051-999-6	Lapatinib	200037	ALK		nM
10051-999-6	Lapatinib	200038	AMPK-alpha1		nM
10051-999-6	Lapatinib	200039	AMPK-alpha2		nM
10051-999-6	Lapatinib	200040	ANKK1		nM
10051-999-6	Lapatinib	200041	NUAK1		nM
10051-999-6	Lapatinib	200042	M3K5		nM
10051-999-6	Lapatinib	200043	M3K6		nM
10051-999-6	Lapatinib	200044	AURKA		nM
10051-999-6	Lapatinib	200045	AURKB		nM
10051-999-6	Lapatinib	200046	AURKC		nM
10051-999-6	Lapatinib	200047	AXL		nM
10051-999-6	Lapatinib	200048	BIKE		nM
10051-999-6	Lapatinib	200049	BLK		nM
10051-999-6	Lapatinib	200050	BMPR1A		nM
10051-999-6	Lapatinib	200051	BMPR1B		nM
10051-999-6	Lapatinib	200052	BMPR2		nM
10051-999-6	Lapatinib	200053	BMX		nM
10051-999-6	Lapatinib	200054	BRAF		nM
10051-999-6	Lapatinib	200055	BRAF(V600E)		nM
10051-999-6	Lapatinib	200056	PTK6		nM
10051-999-6	Lapatinib	200057	BRSK1		nM
10051-999-6	Lapatinib	200058	BRSK2		nM
10051-999-6	Lapatinib	200059	BTK		nM
10051-999-6	Lapatinib	200060	CAMK1		nM
10051-999-6	Lapatinib	200061	CAMK1D		nM
10051-999-6	Lapatinib	200062	CAMK1G		nM
10051-999-6	Lapatinib	200063	CAMK2A		nM
10051-999-6	Lapatinib	200064	CAMK2B		nM
10051-999-6	Lapatinib	200065	KCC2D		nM
10051-999-6	Lapatinib	200066	CAMK2G		nM
10051-999-6	Lapatinib	200067	KCC4		nM
10051-999-6	Lapatinib	200068	KKCC1		nM
10051-999-6	Lapatinib	200069	CAMKK2		nM
10051-999-6	Lapatinib	200070	CASK		nM
10051-999-6	Lapatinib	200071	CDC2L1		nM
10051-999-6	Lapatinib	200072	CDC2L2		nM
10051-999-6	Lapatinib	200073	CDC2L5		nM
10051-999-6	Lapatinib	200074	CDK11		nM
10051-999-6	Lapatinib	200075	CDK2		nM
10051-999-6	Lapatinib	200076	CDK3		nM
10051-999-6	Lapatinib	200077	CDK4-cyclinD1		nM
10051-999-6	Lapatinib	200078	CDK4-cyclinD3		nM
10051-999-6	Lapatinib	200079	CDK5		nM
10051-999-6	Lapatinib	200080	CDK7		nM
10051-999-6	Lapatinib	200081	CDK8		nM
10051-999-6	Lapatinib	200082	CDK9		nM
10051-999-6	Lapatinib	200083	CDKL1		nM
10051-999-6	Lapatinib	200084	CDKL2		nM
10051-999-6	Lapatinib	200085	CDKL3		nM
10051-999-6	Lapatinib	200086	CDKL5		nM
10051-999-6	Lapatinib	200087	CHEK1		nM
10051-999-6	Lapatinib	200088	CHK2		nM
10051-999-6	Lapatinib	200089	CIT		nM
10051-999-6	Lapatinib	200090	CLK1		nM
10051-999-6	Lapatinib	200091	CLK2		nM
10051-999-6	Lapatinib	200092	CLK3		nM
10051-999-6	Lapatinib	200093	CLK4		nM
10051-999-6	Lapatinib	200094	CSF1R		nM
10051-999-6	Lapatinib	200095	CSK		nM
10051-999-6	Lapatinib	200096	CSNK1A1		nM
10051-999-6	Lapatinib	200097	CSNK1A1L		nM
10051-999-6	Lapatinib	200098	CSNK1D		nM
10051-999-6	Lapatinib	200099	CSNK1E		nM
10051-999-6	Lapatinib	200100	KC1G1		nM
10051-999-6	Lapatinib	200101	KC1G2		nM
10051-999-6	Lapatinib	200102	CSNK1G3		nM
10051-999-6	Lapatinib	200103	CSNK2A1		nM
10051-999-6	Lapatinib	200104	CSNK2A2		nM
10051-999-6	Lapatinib	200105	CTK		nM
10051-999-6	Lapatinib	200106	DAPK1		nM
10051-999-6	Lapatinib	200107	DAPK2		nM
10051-999-6	Lapatinib	200108	DAPK3		nM
10051-999-6	Lapatinib	200109	DCLK1		nM
10051-999-6	Lapatinib	200110	DCAMKL2		nM
10051-999-6	Lapatinib	200111	DCAMKL3		nM
10051-999-6	Lapatinib	200112	DDR1		nM
10051-999-6	Lapatinib	200113	DDR2		nM
10051-999-6	Lapatinib	200114	M3K12		nM
10051-999-6	Lapatinib	200115	DMPK		nM
10051-999-6	Lapatinib	200116	DMPK2		nM
10051-999-6	Lapatinib	200117	DRAK1		nM
10051-999-6	Lapatinib	200118	DRAK2		nM
10051-999-6	Lapatinib	200119	DYRK1A		nM
10051-999-6	Lapatinib	200120	DYRK1B		nM
10051-999-6	Lapatinib	200121	DYRK2		nM
10051-999-6	Lapatinib	200122	EGFR	2.4	nM
10051-999-6	Lapatinib	200123	EGFR(E746-A750del)	8.6	nM
10051-999-6	Lapatinib	200124	EGFR(G719C)	0.9	nM
10051-999-6	Lapatinib	200125	EGFR(G719S)	2.1	nM
10051-999-6	Lapatinib	200126	EGFR(L747-E749del, A750P)	2.2	nM
10051-999-6	Lapatinib	200127	EGFR(L747-S752del, P753S)	3.9	nM
10051-999-6	Lapatinib	200128	EGFR(L747-T751del,Sins)	3.5	nM
10051-999-6	Lapatinib	200129	EGFR(L858R)	2.8	nM
10051-999-6	Lapatinib	200130	EGFR(L858R,T790M)		nM
10051-999-6	Lapatinib	200131	EGFR(L861Q)	1.2	nM
10051-999-6	Lapatinib	200132	EGFR(S752-I759del)	4.2	nM
10051-999-6	Lapatinib	200133	EGFR(T790M)	860.0	nM
10051-999-6	Lapatinib	200134	EIF2AK1		nM
10051-999-6	Lapatinib	200135	EPHA1		nM
10051-999-6	Lapatinib	200136	EPHA2		nM
10051-999-6	Lapatinib	200137	EPHA3		nM
10051-999-6	Lapatinib	200138	EPHA4		nM
10051-999-6	Lapatinib	200139	EPHA5		nM
10051-999-6	Lapatinib	200140	EPHA6		nM
10051-999-6	Lapatinib	200141	EPHA7		nM
10051-999-6	Lapatinib	200142	EPHA8		nM
10051-999-6	Lapatinib	200143	EPHB1		nM
10051-999-6	Lapatinib	200144	EPHB2		nM
10051-999-6	Lapatinib	200145	EPHB3		nM
10051-999-6	Lapatinib	200146	EPHB4		nM
10051-999-6	Lapatinib	200147	EPHB6		nM
10051-999-6	Lapatinib	200148	ERBB2	7.0	nM
10051-999-6	Lapatinib	200149	ERBB3	5500.0	nM
10051-999-6	Lapatinib	200150	ERBB4	54.0	nM
10051-999-6	Lapatinib	200151	MK03		nM
10051-999-6	Lapatinib	200152	MK01		nM
10051-999-6	Lapatinib	200153	ERK3		nM
10051-999-6	Lapatinib	200154	ERK4		nM
10051-999-6	Lapatinib	200155	ERK5		nM
10051-999-6	Lapatinib	200156	ERK8		nM
10051-999-6	Lapatinib	200157	ERN1		nM
10051-999-6	Lapatinib	200158	FAK1		nM
10051-999-6	Lapatinib	200159	FER		nM
10051-999-6	Lapatinib	200160	FES		nM
10051-999-6	Lapatinib	200161	FGFR1		nM
10051-999-6	Lapatinib	200162	FGFR2		nM
10051-999-6	Lapatinib	200163	FGFR3		nM
10051-999-6	Lapatinib	200164	FGFR3(G697C)		nM
10051-999-6	Lapatinib	200165	FGFR4		nM
10051-999-6	Lapatinib	200166	FGR		nM
10051-999-6	Lapatinib	200167	VGFR1		nM
10051-999-6	Lapatinib	200168	FLT3		nM
10051-999-6	Lapatinib	200169	FLT3(D835H)		nM
10051-999-6	Lapatinib	200170	FLT3(D835Y)		nM
10051-999-6	Lapatinib	200171	FLT3(ITD)		nM
10051-999-6	Lapatinib	200172	FLT3(K663Q)		nM
10051-999-6	Lapatinib	200173	FLT3(N841I)		nM
10051-999-6	Lapatinib	200174	FLT3(R834Q)		nM
10051-999-6	Lapatinib	200175	FLT4		nM
10051-999-6	Lapatinib	200176	FRK		nM
10051-999-6	Lapatinib	200177	FYN		nM
10051-999-6	Lapatinib	200178	GAK		nM
10051-999-6	Lapatinib	200179	GCN2(Kin.Dom.2,S808G)		nM
10051-999-6	Lapatinib	200180	GRK1		nM
10051-999-6	Lapatinib	200181	GRK4		nM
10051-999-6	Lapatinib	200182	GRK7		nM
10051-999-6	Lapatinib	200183	GSK3A		nM
10051-999-6	Lapatinib	200184	GSK3B		nM
10051-999-6	Lapatinib	200185	HCK		nM
10051-999-6	Lapatinib	200186	HIPK1		nM
10051-999-6	Lapatinib	200187	HIPK2		nM
10051-999-6	Lapatinib	200188	HIPK3		nM
10051-999-6	Lapatinib	200189	HIPK4		nM
10051-999-6	Lapatinib	200190	M4K1		nM
10051-999-6	Lapatinib	200191	HUNK		nM
10051-999-6	Lapatinib	200192	ICK		nM
10051-999-6	Lapatinib	200193	IGF1R		nM
10051-999-6	Lapatinib	200194	IKKA		nM
10051-999-6	Lapatinib	200195	IKKB		nM
10051-999-6	Lapatinib	200196	IKKE		nM
10051-999-6	Lapatinib	200197	INSR		nM
10051-999-6	Lapatinib	200198	INSRR		nM
10051-999-6	Lapatinib	200199	IRAK1		nM
10051-999-6	Lapatinib	200200	IRAK3		nM
10051-999-6	Lapatinib	200201	IRAK4		nM
10051-999-6	Lapatinib	200202	ITK		nM
10051-999-6	Lapatinib	200203	JAK1(JH1domain-catalytic)		nM
10051-999-6	Lapatinib	200204	JAK1(JH2domain-pseudokinase)		nM
10051-999-6	Lapatinib	200207	JAK2(JH1domain-catalytic)		nM
10051-999-6	Lapatinib	200209	JAK3(JH1domain-catalytic)		nM
10051-999-6	Lapatinib	200211	JNK1		nM
10051-999-6	Lapatinib	200212	MK09		nM
10051-999-6	Lapatinib	200213	JNK3		nM
10051-999-6	Lapatinib	200214	KIT		nM
10051-999-6	Lapatinib	200215	KIT(A829P)		nM
10051-999-6	Lapatinib	200216	KIT(D816H)		nM
10051-999-6	Lapatinib	200217	KIT(D816V)		nM
10051-999-6	Lapatinib	200218	KIT(L576P)		nM
10051-999-6	Lapatinib	200219	KIT(V559D)		nM
10051-999-6	Lapatinib	200220	KIT(V559D,T670I)		nM
10051-999-6	Lapatinib	200221	KIT(V559D,V654A)		nM
10051-999-6	Lapatinib	200222	LATS1		nM
10051-999-6	Lapatinib	200223	LATS2		nM
10051-999-6	Lapatinib	200224	LCK		nM
10051-999-6	Lapatinib	200225	LIMK1		nM
10051-999-6	Lapatinib	200226	LIMK2		nM
10051-999-6	Lapatinib	200227	LKB1		nM
10051-999-6	Lapatinib	200228	LOK	4400.0	nM
10051-999-6	Lapatinib	200229	LRRK2		nM
10051-999-6	Lapatinib	200230	LRRK2(G2019S)		nM
10051-999-6	Lapatinib	200231	LTK		nM
10051-999-6	Lapatinib	200232	LYN		nM
10051-999-6	Lapatinib	200233	M3K13		nM
10051-999-6	Lapatinib	200234	MAK		nM
10051-999-6	Lapatinib	200235	MAP3K1		nM
10051-999-6	Lapatinib	200236	MAP3K15		nM
10051-999-6	Lapatinib	200237	M3K2		nM
10051-999-6	Lapatinib	200238	MAP3K3		nM
10051-999-6	Lapatinib	200239	MAP3K4		nM
10051-999-6	Lapatinib	200240	MAP4K2		nM
10051-999-6	Lapatinib	200241	M4K3		nM
10051-999-6	Lapatinib	200242	MAP4K4		nM
10051-999-6	Lapatinib	200243	MAP4K5		nM
10051-999-6	Lapatinib	200244	MAPKAPK2		nM
10051-999-6	Lapatinib	200245	MAPKAPK5		nM
10051-999-6	Lapatinib	200246	MARK1		nM
10051-999-6	Lapatinib	200247	MARK2		nM
10051-999-6	Lapatinib	200248	MARK3		nM
10051-999-6	Lapatinib	200249	MARK4		nM
10051-999-6	Lapatinib	200250	MAST1		nM
10051-999-6	Lapatinib	200251	MP2K1		nM
10051-999-6	Lapatinib	200252	MP2K2		nM
10051-999-6	Lapatinib	200253	MP2K3		nM
10051-999-6	Lapatinib	200254	MP2K4		nM
10051-999-6	Lapatinib	200255	MP2K5	1100.0	nM
10051-999-6	Lapatinib	200256	MP2K6		nM
10051-999-6	Lapatinib	200257	MELK		nM
10051-999-6	Lapatinib	200258	MERTK		nM
10051-999-6	Lapatinib	200259	MET		nM
10051-999-6	Lapatinib	200260	MET(M1250T)		nM
10051-999-6	Lapatinib	200261	MET(Y1235D)		nM
10051-999-6	Lapatinib	200262	MINK		nM
10051-999-6	Lapatinib	200263	MP2K7	4400.0	nM
10051-999-6	Lapatinib	200264	MKNK1		nM
10051-999-6	Lapatinib	200265	MKNK2		nM
10051-999-6	Lapatinib	200266	MLCK		nM
10051-999-6	Lapatinib	200267	MLK1		nM
10051-999-6	Lapatinib	200268	MLK2		nM
10051-999-6	Lapatinib	200269	MLK3		nM
10051-999-6	Lapatinib	200270	MRCKA		nM
10051-999-6	Lapatinib	200271	MRCKB		nM
10051-999-6	Lapatinib	200272	MST1		nM
10051-999-6	Lapatinib	200273	MST1R		nM
10051-999-6	Lapatinib	200274	MST2		nM
10051-999-6	Lapatinib	200275	MST3		nM
10051-999-6	Lapatinib	200276	MST4		nM
10051-999-6	Lapatinib	200277	MTOR		nM
10051-999-6	Lapatinib	200278	MUSK		nM
10051-999-6	Lapatinib	200279	MYLK		nM
10051-999-6	Lapatinib	200280	MYLK2		nM
10051-999-6	Lapatinib	200281	MYLK4		nM
10051-999-6	Lapatinib	200282	MYO3A		nM
10051-999-6	Lapatinib	200283	MYO3B		nM
10051-999-6	Lapatinib	200284	NDR1		nM
10051-999-6	Lapatinib	200285	NDR2		nM
10051-999-6	Lapatinib	200286	NEK1		nM
10051-999-6	Lapatinib	200287	NEK11		nM
10051-999-6	Lapatinib	200288	NEK2		nM
10051-999-6	Lapatinib	200289	NEK3		nM
10051-999-6	Lapatinib	200290	NEK4		nM
10051-999-6	Lapatinib	200291	NEK5		nM
10051-999-6	Lapatinib	200292	NEK6		nM
10051-999-6	Lapatinib	200293	NEK7		nM
10051-999-6	Lapatinib	200294	NEK9		nM
10051-999-6	Lapatinib	200295	NIM1		nM
10051-999-6	Lapatinib	200296	NLK		nM
10051-999-6	Lapatinib	200297	OSR1		nM
10051-999-6	Lapatinib	200298	MK14		nM
10051-999-6	Lapatinib	200299	MK11		nM
10051-999-6	Lapatinib	200300	MK13		nM
10051-999-6	Lapatinib	200301	MK12		nM
10051-999-6	Lapatinib	200302	PAK1		nM
10051-999-6	Lapatinib	200303	PAK2		nM
10051-999-6	Lapatinib	200304	PAK3		nM
10051-999-6	Lapatinib	200305	PAK4		nM
10051-999-6	Lapatinib	200306	PAK6		nM
10051-999-6	Lapatinib	200307	PAK7		nM
10051-999-6	Lapatinib	200309	CDK16		nM
10051-999-6	Lapatinib	200310	PCTK2		nM
10051-999-6	Lapatinib	200311	PCTK3		nM
10051-999-6	Lapatinib	200312	PGFRA		nM
10051-999-6	Lapatinib	200313	PGFRB		nM
10051-999-6	Lapatinib	200314	PDPK1		nM
10051-999-6	Lapatinib	200315	PFCDPK1(P.falciparum)		nM
10051-999-6	Lapatinib	200316	PFPK5(P.falciparum)		nM
10051-999-6	Lapatinib	200317	CDK15		nM
10051-999-6	Lapatinib	200318	CDK14		nM
10051-999-6	Lapatinib	200319	PHKG1		nM
10051-999-6	Lapatinib	200320	PHKG2		nM
10051-999-6	Lapatinib	200321	PIK3C2B	670.0	nM
10051-999-6	Lapatinib	200322	PIK3C2G	7500.0	nM
10051-999-6	Lapatinib	200323	PIK3CA		nM
10051-999-6	Lapatinib	200324	PIK3CA(C420R)		nM
10051-999-6	Lapatinib	200325	PIK3CA(E542K)		nM
10051-999-6	Lapatinib	200326	PIK3CA(E545A)		nM
10051-999-6	Lapatinib	200327	PIK3CA(E545K)		nM
10051-999-6	Lapatinib	200328	PIK3CA(H1047L)		nM
10051-999-6	Lapatinib	200329	PIK3CA(H1047Y)		nM
10051-999-6	Lapatinib	200330	PIK3CA(I800L)		nM
10051-999-6	Lapatinib	200331	PIK3CA(M1043I)		nM
10051-999-6	Lapatinib	200332	PIK3CA(Q546K)		nM
10051-999-6	Lapatinib	200333	PIK3CB		nM
10051-999-6	Lapatinib	200334	PIK3CD		nM
10051-999-6	Lapatinib	200335	PIK3CG		nM
10051-999-6	Lapatinib	200336	PIK4CB	940.0	nM
10051-999-6	Lapatinib	200337	PIM1		nM
10051-999-6	Lapatinib	200338	PIM2		nM
10051-999-6	Lapatinib	200339	PIM3		nM
10051-999-6	Lapatinib	200340	PIP5K1A		nM
10051-999-6	Lapatinib	200341	PIP5K1C		nM
10051-999-6	Lapatinib	200342	PIP5K2B		nM
10051-999-6	Lapatinib	200343	PI42C		nM
10051-999-6	Lapatinib	200344	PKAC-alpha		nM
10051-999-6	Lapatinib	200345	PKAC-beta		nM
10051-999-6	Lapatinib	200346	PKMYT1		nM
10051-999-6	Lapatinib	200347	PKN1		nM
10051-999-6	Lapatinib	200348	PKN2		nM
10051-999-6	Lapatinib	200349	PKNB(M.tuberculosis)		nM
10051-999-6	Lapatinib	200350	PLK1		nM
10051-999-6	Lapatinib	200351	PLK2		nM
10051-999-6	Lapatinib	200352	PLK3		nM
10051-999-6	Lapatinib	200353	PLK4		nM
10051-999-6	Lapatinib	200354	KPCD		nM
10051-999-6	Lapatinib	200355	KPCE		nM
10051-999-6	Lapatinib	200356	KPCL		nM
10051-999-6	Lapatinib	200357	KPCI		nM
10051-999-6	Lapatinib	200358	KPCT		nM
10051-999-6	Lapatinib	200359	KPCD1		nM
10051-999-6	Lapatinib	200360	KPCD2		nM
10051-999-6	Lapatinib	200361	KPCD3		nM
10051-999-6	Lapatinib	200362	KGP1		nM
10051-999-6	Lapatinib	200363	KGP2		nM
10051-999-6	Lapatinib	200364	PRKR		nM
10051-999-6	Lapatinib	200365	PRKX		nM
10051-999-6	Lapatinib	200366	PRP4		nM
10051-999-6	Lapatinib	200367	FAK2		nM
10051-999-6	Lapatinib	200368	SIK3		nM
10051-999-6	Lapatinib	200369	RAF1		nM
10051-999-6	Lapatinib	200370	RET		nM
10051-999-6	Lapatinib	200371	RET(M918T)		nM
10051-999-6	Lapatinib	200372	RET(V804L)		nM
10051-999-6	Lapatinib	200373	RET(V804M)		nM
10051-999-6	Lapatinib	200374	RIOK1		nM
10051-999-6	Lapatinib	200375	RIOK2		nM
10051-999-6	Lapatinib	200376	RIOK3		nM
10051-999-6	Lapatinib	200377	RIPK1		nM
10051-999-6	Lapatinib	200378	RIPK2	3600.0	nM
10051-999-6	Lapatinib	200379	RIPK4		nM
10051-999-6	Lapatinib	200380	RIPK5		nM
10051-999-6	Lapatinib	200381	ROCK1		nM
10051-999-6	Lapatinib	200382	ROCK2		nM
10051-999-6	Lapatinib	200383	ROS1		nM
10051-999-6	Lapatinib	200390	RPS6KA4(Kin.Dom.1-N-terminal)		nM
10051-999-6	Lapatinib	200392	RPS6KA4(Kin.Dom.2-C-terminal)		nM
10051-999-6	Lapatinib	200394	RPS6KA5(Kin.Dom.1-N-terminal)		nM
10051-999-6	Lapatinib	200396	RPS6KA5(Kin.Dom.2-C-terminal)		nM
10051-999-6	Lapatinib	200399	RSK1(Kin.Dom.1-N-terminal)		nM
10051-999-6	Lapatinib	200400	RSK1(Kin.Dom.2-C-terminal)		nM
10051-999-6	Lapatinib	200401	RSK2(Kin.Dom.1-N-terminal)		nM
10051-999-6	Lapatinib	200402	RSK3(Kin.Dom.1-N-terminal)		nM
10051-999-6	Lapatinib	200403	RSK3(Kin.Dom.2-C-terminal)		nM
10051-999-6	Lapatinib	200404	RSK4(Kin.Dom.1-N-terminal)		nM
10051-999-6	Lapatinib	200405	RSK4(Kin.Dom.2-C-terminal)		nM
10051-999-6	Lapatinib	200406	S6K1		nM
10051-999-6	Lapatinib	200407	SBK1		nM
10051-999-6	Lapatinib	200408	SgK110		nM
10051-999-6	Lapatinib	200409	SGK3		nM
10051-999-6	Lapatinib	200410	SIK1		nM
10051-999-6	Lapatinib	200411	SIK2		nM
10051-999-6	Lapatinib	200412	SLK	3300.0	nM
10051-999-6	Lapatinib	200413	SNARK		nM
10051-999-6	Lapatinib	200414	SNRK		nM
10051-999-6	Lapatinib	200415	SRC		nM
10051-999-6	Lapatinib	200416	SRMS		nM
10051-999-6	Lapatinib	200417	SRPK1		nM
10051-999-6	Lapatinib	200418	SRPK2		nM
10051-999-6	Lapatinib	200419	SRPK3		nM
10051-999-6	Lapatinib	200420	STK16		nM
10051-999-6	Lapatinib	200421	STK33		nM
10051-999-6	Lapatinib	200422	STK35		nM
10051-999-6	Lapatinib	200423	STK36		nM
10051-999-6	Lapatinib	200424	STK39		nM
10051-999-6	Lapatinib	200425	SYK		nM
10051-999-6	Lapatinib	200426	TAK1		nM
10051-999-6	Lapatinib	200427	TAOK1		nM
10051-999-6	Lapatinib	200428	TAOK2		nM
10051-999-6	Lapatinib	200429	TAOK3		nM
10051-999-6	Lapatinib	200430	TBK1		nM
10051-999-6	Lapatinib	200431	TEC		nM
10051-999-6	Lapatinib	200432	TESK1		nM
10051-999-6	Lapatinib	200433	TGFBR1		nM
10051-999-6	Lapatinib	200434	TGFBR2		nM
10051-999-6	Lapatinib	200435	TIE1		nM
10051-999-6	Lapatinib	200436	TIE2		nM
10051-999-6	Lapatinib	200437	TLK1		nM
10051-999-6	Lapatinib	200438	TLK2		nM
10051-999-6	Lapatinib	200439	TNIK		nM
10051-999-6	Lapatinib	200440	TNK1		nM
10051-999-6	Lapatinib	200441	TNK2		nM
10051-999-6	Lapatinib	200442	TNNI3K		nM
10051-999-6	Lapatinib	200443	TRKA		nM
10051-999-6	Lapatinib	200444	TRKB		nM
10051-999-6	Lapatinib	200445	TRKC		nM
10051-999-6	Lapatinib	200446	TRPM6		nM
10051-999-6	Lapatinib	200447	TSSK1		nM
10051-999-6	Lapatinib	200448	TTK		nM
10051-999-6	Lapatinib	200449	TXK		nM
10051-999-6	Lapatinib	200450	TYK2(JH1domain-catalytic)		nM
10051-999-6	Lapatinib	200451	TYK2(JH2domain-pseudokinase)		nM
10051-999-6	Lapatinib	200454	TYRO3		nM
10051-999-6	Lapatinib	200455	ULK1		nM
10051-999-6	Lapatinib	200456	ULK2		nM
10051-999-6	Lapatinib	200457	ULK3		nM
10051-999-6	Lapatinib	200458	VGFR2		nM
10051-999-6	Lapatinib	200459	VRK2		nM
10051-999-6	Lapatinib	200460	WEE1		nM
10051-999-6	Lapatinib	200461	WEE2		nM
10051-999-6	Lapatinib	200462	YANK1		nM
10051-999-6	Lapatinib	200463	YANK2		nM
10051-999-6	Lapatinib	200464	YANK3		nM
10051-999-6	Lapatinib	200465	YES		nM
10051-999-6	Lapatinib	200466	YSK1		nM
10051-999-6	Lapatinib	200467	YSK4		nM
10051-999-6	Lapatinib	200468	MLTK		nM
10051-999-6	Lapatinib	200469	ZAP70		nM
