Small Molecule HMS LINCS ID	Small Molecule Name	Protein HMS LINCS ID	Protein Name	Kd	Conc unit
10041-999-4	BI-2536	200001	AAK1	2800.0	nM
10041-999-4	BI-2536	200004	ABL1(E255K)-phosphorylated	5900.0	nM
10041-999-4	BI-2536	200006	ABL1(F317I)-nonphosphorylated		nM
10041-999-4	BI-2536	200007	ABL1(F317I)-phosphorylated		nM
10041-999-4	BI-2536	200009	ABL1(F317L)-nonphosphorylated		nM
10041-999-4	BI-2536	200010	ABL1(F317L)-phosphorylated	2400.0	nM
10041-999-4	BI-2536	200012	ABL1(H396P)-nonphosphorylated	2000.0	nM
10041-999-4	BI-2536	200013	ABL1(H396P)-phosphorylated	2600.0	nM
10041-999-4	BI-2536	200015	ABL1(M351T)-phosphorylated		nM
10041-999-4	BI-2536	200017	ABL1(Q252H)-nonphosphorylated		nM
10041-999-4	BI-2536	200018	ABL1(Q252H)-phosphorylated		nM
10041-999-4	BI-2536	200020	ABL1(T315I)-nonphosphorylated		nM
10041-999-4	BI-2536	200021	ABL1(T315I)-phosphorylated		nM
10041-999-4	BI-2536	200023	ABL1(Y253F)-phosphorylated		nM
10041-999-4	BI-2536	200024	ABL1-nonphosphorylated		nM
10041-999-4	BI-2536	200025	ABL1-phosphorylated	3500.0	nM
10041-999-4	BI-2536	200026	ABL2		nM
10041-999-4	BI-2536	200027	ACVR1		nM
10041-999-4	BI-2536	200028	ACVR1B		nM
10041-999-4	BI-2536	200029	ACVR2A		nM
10041-999-4	BI-2536	200030	ACVR2B		nM
10041-999-4	BI-2536	200031	ACVRL1		nM
10041-999-4	BI-2536	200032	ADCK3		nM
10041-999-4	BI-2536	200033	ADCK4		nM
10041-999-4	BI-2536	200034	AKT1		nM
10041-999-4	BI-2536	200035	AKT2		nM
10041-999-4	BI-2536	200036	AKT3		nM
10041-999-4	BI-2536	200037	ALK	160.0	nM
10041-999-4	BI-2536	200038	AMPK-alpha1		nM
10041-999-4	BI-2536	200039	AMPK-alpha2		nM
10041-999-4	BI-2536	200040	ANKK1		nM
10041-999-4	BI-2536	200041	NUAK1		nM
10041-999-4	BI-2536	200042	M3K5		nM
10041-999-4	BI-2536	200043	M3K6		nM
10041-999-4	BI-2536	200044	AURKA		nM
10041-999-4	BI-2536	200045	AURKB		nM
10041-999-4	BI-2536	200046	AURKC		nM
10041-999-4	BI-2536	200047	AXL		nM
10041-999-4	BI-2536	200048	BIKE		nM
10041-999-4	BI-2536	200049	BLK		nM
10041-999-4	BI-2536	200050	BMPR1A		nM
10041-999-4	BI-2536	200051	BMPR1B		nM
10041-999-4	BI-2536	200052	BMPR2		nM
10041-999-4	BI-2536	200053	BMX		nM
10041-999-4	BI-2536	200054	BRAF		nM
10041-999-4	BI-2536	200055	BRAF(V600E)		nM
10041-999-4	BI-2536	200056	PTK6		nM
10041-999-4	BI-2536	200057	BRSK1		nM
10041-999-4	BI-2536	200058	BRSK2		nM
10041-999-4	BI-2536	200059	BTK		nM
10041-999-4	BI-2536	200060	CAMK1		nM
10041-999-4	BI-2536	200061	CAMK1D	5400.0	nM
10041-999-4	BI-2536	200062	CAMK1G		nM
10041-999-4	BI-2536	200063	CAMK2A	1300.0	nM
10041-999-4	BI-2536	200064	CAMK2B	4200.0	nM
10041-999-4	BI-2536	200065	KCC2D	2400.0	nM
10041-999-4	BI-2536	200066	CAMK2G	1200.0	nM
10041-999-4	BI-2536	200067	KCC4		nM
10041-999-4	BI-2536	200068	KKCC1	22.0	nM
10041-999-4	BI-2536	200069	CAMKK2	23.0	nM
10041-999-4	BI-2536	200070	CASK		nM
10041-999-4	BI-2536	200071	CDC2L1		nM
10041-999-4	BI-2536	200072	CDC2L2		nM
10041-999-4	BI-2536	200073	CDC2L5		nM
10041-999-4	BI-2536	200074	CDK11		nM
10041-999-4	BI-2536	200075	CDK2		nM
10041-999-4	BI-2536	200076	CDK3		nM
10041-999-4	BI-2536	200077	CDK4-cyclinD1		nM
10041-999-4	BI-2536	200078	CDK4-cyclinD3	1900.0	nM
10041-999-4	BI-2536	200079	CDK5		nM
10041-999-4	BI-2536	200080	CDK7	3500.0	nM
10041-999-4	BI-2536	200081	CDK8		nM
10041-999-4	BI-2536	200082	CDK9		nM
10041-999-4	BI-2536	200083	CDKL1		nM
10041-999-4	BI-2536	200084	CDKL2		nM
10041-999-4	BI-2536	200085	CDKL3		nM
10041-999-4	BI-2536	200086	CDKL5		nM
10041-999-4	BI-2536	200087	CHEK1		nM
10041-999-4	BI-2536	200088	CHK2	7700.0	nM
10041-999-4	BI-2536	200089	CIT	5200.0	nM
10041-999-4	BI-2536	200090	CLK1	940.0	nM
10041-999-4	BI-2536	200091	CLK2	460.0	nM
10041-999-4	BI-2536	200092	CLK3	630.0	nM
10041-999-4	BI-2536	200093	CLK4		nM
10041-999-4	BI-2536	200094	CSF1R		nM
10041-999-4	BI-2536	200095	CSK		nM
10041-999-4	BI-2536	200096	CSNK1A1	3100.0	nM
10041-999-4	BI-2536	200097	CSNK1A1L		nM
10041-999-4	BI-2536	200098	CSNK1D	1500.0	nM
10041-999-4	BI-2536	200099	CSNK1E	380.0	nM
10041-999-4	BI-2536	200100	KC1G1	4500.0	nM
10041-999-4	BI-2536	200101	KC1G2	5700.0	nM
10041-999-4	BI-2536	200102	CSNK1G3	2400.0	nM
10041-999-4	BI-2536	200103	CSNK2A1		nM
10041-999-4	BI-2536	200104	CSNK2A2		nM
10041-999-4	BI-2536	200105	CTK		nM
10041-999-4	BI-2536	200106	DAPK1	540.0	nM
10041-999-4	BI-2536	200107	DAPK2	930.0	nM
10041-999-4	BI-2536	200108	DAPK3	130.0	nM
10041-999-4	BI-2536	200109	DCLK1	5900.0	nM
10041-999-4	BI-2536	200110	DCAMKL2		nM
10041-999-4	BI-2536	200111	DCAMKL3		nM
10041-999-4	BI-2536	200112	DDR1		nM
10041-999-4	BI-2536	200113	DDR2		nM
10041-999-4	BI-2536	200114	M3K12		nM
10041-999-4	BI-2536	200115	DMPK	2900.0	nM
10041-999-4	BI-2536	200116	DMPK2		nM
10041-999-4	BI-2536	200117	DRAK1		nM
10041-999-4	BI-2536	200118	DRAK2		nM
10041-999-4	BI-2536	200119	DYRK1A		nM
10041-999-4	BI-2536	200120	DYRK1B		nM
10041-999-4	BI-2536	200121	DYRK2		nM
10041-999-4	BI-2536	200122	EGFR	2200.0	nM
10041-999-4	BI-2536	200123	EGFR(E746-A750del)	1900.0	nM
10041-999-4	BI-2536	200124	EGFR(G719C)	630.0	nM
10041-999-4	BI-2536	200125	EGFR(G719S)	1300.0	nM
10041-999-4	BI-2536	200126	EGFR(L747-E749del, A750P)	1100.0	nM
10041-999-4	BI-2536	200127	EGFR(L747-S752del, P753S)	6300.0	nM
10041-999-4	BI-2536	200128	EGFR(L747-T751del,Sins)	4800.0	nM
10041-999-4	BI-2536	200129	EGFR(L858R)	1300.0	nM
10041-999-4	BI-2536	200130	EGFR(L858R,T790M)	240.0	nM
10041-999-4	BI-2536	200131	EGFR(L861Q)	2700.0	nM
10041-999-4	BI-2536	200132	EGFR(S752-I759del)	5300.0	nM
10041-999-4	BI-2536	200133	EGFR(T790M)	360.0	nM
10041-999-4	BI-2536	200134	EIF2AK1		nM
10041-999-4	BI-2536	200135	EPHA1		nM
10041-999-4	BI-2536	200136	EPHA2		nM
10041-999-4	BI-2536	200137	EPHA3		nM
10041-999-4	BI-2536	200138	EPHA4		nM
10041-999-4	BI-2536	200139	EPHA5		nM
10041-999-4	BI-2536	200140	EPHA6		nM
10041-999-4	BI-2536	200141	EPHA7		nM
10041-999-4	BI-2536	200142	EPHA8		nM
10041-999-4	BI-2536	200143	EPHB1		nM
10041-999-4	BI-2536	200144	EPHB2		nM
10041-999-4	BI-2536	200145	EPHB3		nM
10041-999-4	BI-2536	200146	EPHB4		nM
10041-999-4	BI-2536	200147	EPHB6		nM
10041-999-4	BI-2536	200148	ERBB2		nM
10041-999-4	BI-2536	200149	ERBB3		nM
10041-999-4	BI-2536	200150	ERBB4		nM
10041-999-4	BI-2536	200151	MK03		nM
10041-999-4	BI-2536	200152	MK01		nM
10041-999-4	BI-2536	200153	ERK3		nM
10041-999-4	BI-2536	200154	ERK4		nM
10041-999-4	BI-2536	200155	ERK5	3200.0	nM
10041-999-4	BI-2536	200156	ERK8		nM
10041-999-4	BI-2536	200157	ERN1		nM
10041-999-4	BI-2536	200158	FAK1	150.0	nM
10041-999-4	BI-2536	200159	FER		nM
10041-999-4	BI-2536	200160	FES	1900.0	nM
10041-999-4	BI-2536	200161	FGFR1		nM
10041-999-4	BI-2536	200162	FGFR2		nM
10041-999-4	BI-2536	200163	FGFR3		nM
10041-999-4	BI-2536	200164	FGFR3(G697C)		nM
10041-999-4	BI-2536	200165	FGFR4		nM
10041-999-4	BI-2536	200166	FGR		nM
10041-999-4	BI-2536	200167	VGFR1		nM
10041-999-4	BI-2536	200168	FLT3		nM
10041-999-4	BI-2536	200169	FLT3(D835H)		nM
10041-999-4	BI-2536	200170	FLT3(D835Y)	3000.0	nM
10041-999-4	BI-2536	200171	FLT3(ITD)		nM
10041-999-4	BI-2536	200172	FLT3(K663Q)		nM
10041-999-4	BI-2536	200173	FLT3(N841I)		nM
10041-999-4	BI-2536	200174	FLT3(R834Q)		nM
10041-999-4	BI-2536	200175	FLT4		nM
10041-999-4	BI-2536	200176	FRK		nM
10041-999-4	BI-2536	200177	FYN		nM
10041-999-4	BI-2536	200178	GAK	180.0	nM
10041-999-4	BI-2536	200179	GCN2(Kin.Dom.2,S808G)		nM
10041-999-4	BI-2536	200180	GRK1		nM
10041-999-4	BI-2536	200181	GRK4		nM
10041-999-4	BI-2536	200182	GRK7	850.0	nM
10041-999-4	BI-2536	200183	GSK3A		nM
10041-999-4	BI-2536	200184	GSK3B		nM
10041-999-4	BI-2536	200185	HCK		nM
10041-999-4	BI-2536	200186	HIPK1	4100.0	nM
10041-999-4	BI-2536	200187	HIPK2	2900.0	nM
10041-999-4	BI-2536	200188	HIPK3	3600.0	nM
10041-999-4	BI-2536	200189	HIPK4	2000.0	nM
10041-999-4	BI-2536	200190	M4K1		nM
10041-999-4	BI-2536	200191	HUNK	9700.0	nM
10041-999-4	BI-2536	200192	ICK		nM
10041-999-4	BI-2536	200193	IGF1R		nM
10041-999-4	BI-2536	200194	IKKA		nM
10041-999-4	BI-2536	200195	IKKB		nM
10041-999-4	BI-2536	200196	IKKE		nM
10041-999-4	BI-2536	200197	INSR		nM
10041-999-4	BI-2536	200198	INSRR		nM
10041-999-4	BI-2536	200199	IRAK1	1900.0	nM
10041-999-4	BI-2536	200200	IRAK3		nM
10041-999-4	BI-2536	200201	IRAK4	2100.0	nM
10041-999-4	BI-2536	200202	ITK		nM
10041-999-4	BI-2536	200203	JAK1(JH1domain-catalytic)		nM
10041-999-4	BI-2536	200204	JAK1(JH2domain-pseudokinase)		nM
10041-999-4	BI-2536	200207	JAK2(JH1domain-catalytic)		nM
10041-999-4	BI-2536	200209	JAK3(JH1domain-catalytic)		nM
10041-999-4	BI-2536	200211	JNK1		nM
10041-999-4	BI-2536	200212	MK09		nM
10041-999-4	BI-2536	200213	JNK3	1100.0	nM
10041-999-4	BI-2536	200214	KIT		nM
10041-999-4	BI-2536	200215	KIT(A829P)		nM
10041-999-4	BI-2536	200216	KIT(D816H)		nM
10041-999-4	BI-2536	200217	KIT(D816V)		nM
10041-999-4	BI-2536	200218	KIT(L576P)		nM
10041-999-4	BI-2536	200219	KIT(V559D)		nM
10041-999-4	BI-2536	200220	KIT(V559D,T670I)		nM
10041-999-4	BI-2536	200221	KIT(V559D,V654A)		nM
10041-999-4	BI-2536	200222	LATS1		nM
10041-999-4	BI-2536	200223	LATS2		nM
10041-999-4	BI-2536	200224	LCK		nM
10041-999-4	BI-2536	200225	LIMK1		nM
10041-999-4	BI-2536	200226	LIMK2		nM
10041-999-4	BI-2536	200227	LKB1		nM
10041-999-4	BI-2536	200228	LOK	4900.0	nM
10041-999-4	BI-2536	200229	LRRK2		nM
10041-999-4	BI-2536	200230	LRRK2(G2019S)		nM
10041-999-4	BI-2536	200231	LTK	1200.0	nM
10041-999-4	BI-2536	200232	LYN		nM
10041-999-4	BI-2536	200233	M3K13		nM
10041-999-4	BI-2536	200234	MAK		nM
10041-999-4	BI-2536	200235	MAP3K1		nM
10041-999-4	BI-2536	200236	MAP3K15		nM
10041-999-4	BI-2536	200237	M3K2		nM
10041-999-4	BI-2536	200238	MAP3K3		nM
10041-999-4	BI-2536	200239	MAP3K4		nM
10041-999-4	BI-2536	200240	MAP4K2		nM
10041-999-4	BI-2536	200241	M4K3		nM
10041-999-4	BI-2536	200242	MAP4K4		nM
10041-999-4	BI-2536	200243	MAP4K5		nM
10041-999-4	BI-2536	200244	MAPKAPK2		nM
10041-999-4	BI-2536	200245	MAPKAPK5		nM
10041-999-4	BI-2536	200246	MARK1		nM
10041-999-4	BI-2536	200247	MARK2		nM
10041-999-4	BI-2536	200248	MARK3		nM
10041-999-4	BI-2536	200249	MARK4		nM
10041-999-4	BI-2536	200250	MAST1		nM
10041-999-4	BI-2536	200251	MP2K1		nM
10041-999-4	BI-2536	200252	MP2K2		nM
10041-999-4	BI-2536	200253	MP2K3		nM
10041-999-4	BI-2536	200254	MP2K4		nM
10041-999-4	BI-2536	200255	MP2K5		nM
10041-999-4	BI-2536	200256	MP2K6		nM
10041-999-4	BI-2536	200257	MELK		nM
10041-999-4	BI-2536	200258	MERTK	3100.0	nM
10041-999-4	BI-2536	200259	MET	2400.0	nM
10041-999-4	BI-2536	200260	MET(M1250T)		nM
10041-999-4	BI-2536	200261	MET(Y1235D)		nM
10041-999-4	BI-2536	200262	MINK	1600.0	nM
10041-999-4	BI-2536	200263	MP2K7		nM
10041-999-4	BI-2536	200264	MKNK1		nM
10041-999-4	BI-2536	200265	MKNK2		nM
10041-999-4	BI-2536	200266	MLCK		nM
10041-999-4	BI-2536	200267	MLK1		nM
10041-999-4	BI-2536	200268	MLK2		nM
10041-999-4	BI-2536	200269	MLK3		nM
10041-999-4	BI-2536	200270	MRCKA		nM
10041-999-4	BI-2536	200271	MRCKB		nM
10041-999-4	BI-2536	200272	MST1		nM
10041-999-4	BI-2536	200273	MST1R		nM
10041-999-4	BI-2536	200274	MST2		nM
10041-999-4	BI-2536	200275	MST3		nM
10041-999-4	BI-2536	200276	MST4		nM
10041-999-4	BI-2536	200277	MTOR		nM
10041-999-4	BI-2536	200278	MUSK		nM
10041-999-4	BI-2536	200279	MYLK	97.0	nM
10041-999-4	BI-2536	200280	MYLK2		nM
10041-999-4	BI-2536	200281	MYLK4		nM
10041-999-4	BI-2536	200282	MYO3A	6300.0	nM
10041-999-4	BI-2536	200283	MYO3B	3500.0	nM
10041-999-4	BI-2536	200284	NDR1		nM
10041-999-4	BI-2536	200285	NDR2		nM
10041-999-4	BI-2536	200286	NEK1		nM
10041-999-4	BI-2536	200287	NEK11		nM
10041-999-4	BI-2536	200288	NEK2	2000.0	nM
10041-999-4	BI-2536	200289	NEK3	720.0	nM
10041-999-4	BI-2536	200290	NEK4		nM
10041-999-4	BI-2536	200291	NEK5		nM
10041-999-4	BI-2536	200292	NEK6		nM
10041-999-4	BI-2536	200293	NEK7	6100.0	nM
10041-999-4	BI-2536	200294	NEK9		nM
10041-999-4	BI-2536	200295	NIM1	770.0	nM
10041-999-4	BI-2536	200296	NLK		nM
10041-999-4	BI-2536	200297	OSR1		nM
10041-999-4	BI-2536	200298	MK14		nM
10041-999-4	BI-2536	200299	MK11		nM
10041-999-4	BI-2536	200300	MK13		nM
10041-999-4	BI-2536	200301	MK12		nM
10041-999-4	BI-2536	200302	PAK1		nM
10041-999-4	BI-2536	200303	PAK2		nM
10041-999-4	BI-2536	200304	PAK3		nM
10041-999-4	BI-2536	200305	PAK4		nM
10041-999-4	BI-2536	200306	PAK6		nM
10041-999-4	BI-2536	200307	PAK7		nM
10041-999-4	BI-2536	200309	CDK16		nM
10041-999-4	BI-2536	200310	PCTK2		nM
10041-999-4	BI-2536	200311	PCTK3		nM
10041-999-4	BI-2536	200312	PGFRA		nM
10041-999-4	BI-2536	200313	PGFRB		nM
10041-999-4	BI-2536	200314	PDPK1		nM
10041-999-4	BI-2536	200315	PFCDPK1(P.falciparum)		nM
10041-999-4	BI-2536	200316	PFPK5(P.falciparum)		nM
10041-999-4	BI-2536	200317	CDK15		nM
10041-999-4	BI-2536	200318	CDK14		nM
10041-999-4	BI-2536	200319	PHKG1		nM
10041-999-4	BI-2536	200320	PHKG2	1600.0	nM
10041-999-4	BI-2536	200321	PIK3C2B		nM
10041-999-4	BI-2536	200322	PIK3C2G		nM
10041-999-4	BI-2536	200323	PIK3CA		nM
10041-999-4	BI-2536	200324	PIK3CA(C420R)		nM
10041-999-4	BI-2536	200325	PIK3CA(E542K)		nM
10041-999-4	BI-2536	200326	PIK3CA(E545A)		nM
10041-999-4	BI-2536	200327	PIK3CA(E545K)		nM
10041-999-4	BI-2536	200328	PIK3CA(H1047L)		nM
10041-999-4	BI-2536	200329	PIK3CA(H1047Y)		nM
10041-999-4	BI-2536	200330	PIK3CA(I800L)		nM
10041-999-4	BI-2536	200331	PIK3CA(M1043I)		nM
10041-999-4	BI-2536	200332	PIK3CA(Q546K)		nM
10041-999-4	BI-2536	200333	PIK3CB		nM
10041-999-4	BI-2536	200334	PIK3CD	7600.0	nM
10041-999-4	BI-2536	200335	PIK3CG		nM
10041-999-4	BI-2536	200336	PIK4CB		nM
10041-999-4	BI-2536	200337	PIM1		nM
10041-999-4	BI-2536	200338	PIM2		nM
10041-999-4	BI-2536	200339	PIM3		nM
10041-999-4	BI-2536	200340	PIP5K1A		nM
10041-999-4	BI-2536	200341	PIP5K1C		nM
10041-999-4	BI-2536	200342	PIP5K2B		nM
10041-999-4	BI-2536	200343	PI42C	110.0	nM
10041-999-4	BI-2536	200344	PKAC-alpha		nM
10041-999-4	BI-2536	200345	PKAC-beta		nM
10041-999-4	BI-2536	200346	PKMYT1		nM
10041-999-4	BI-2536	200347	PKN1		nM
10041-999-4	BI-2536	200348	PKN2		nM
10041-999-4	BI-2536	200349	PKNB(M.tuberculosis)		nM
10041-999-4	BI-2536	200350	PLK1	0.2	nM
10041-999-4	BI-2536	200351	PLK2	0.8	nM
10041-999-4	BI-2536	200352	PLK3	4.0	nM
10041-999-4	BI-2536	200353	PLK4		nM
10041-999-4	BI-2536	200354	KPCD		nM
10041-999-4	BI-2536	200355	KPCE		nM
10041-999-4	BI-2536	200356	KPCL		nM
10041-999-4	BI-2536	200357	KPCI		nM
10041-999-4	BI-2536	200358	KPCT		nM
10041-999-4	BI-2536	200359	KPCD1	320.0	nM
10041-999-4	BI-2536	200360	KPCD2	510.0	nM
10041-999-4	BI-2536	200361	KPCD3	350.0	nM
10041-999-4	BI-2536	200362	KGP1		nM
10041-999-4	BI-2536	200363	KGP2		nM
10041-999-4	BI-2536	200364	PRKR	460.0	nM
10041-999-4	BI-2536	200365	PRKX		nM
10041-999-4	BI-2536	200366	PRP4		nM
10041-999-4	BI-2536	200367	FAK2	310.0	nM
10041-999-4	BI-2536	200368	SIK3		nM
10041-999-4	BI-2536	200369	RAF1		nM
10041-999-4	BI-2536	200370	RET		nM
10041-999-4	BI-2536	200371	RET(M918T)		nM
10041-999-4	BI-2536	200372	RET(V804L)		nM
10041-999-4	BI-2536	200373	RET(V804M)		nM
10041-999-4	BI-2536	200374	RIOK1	2200.0	nM
10041-999-4	BI-2536	200375	RIOK2		nM
10041-999-4	BI-2536	200376	RIOK3	4400.0	nM
10041-999-4	BI-2536	200377	RIPK1		nM
10041-999-4	BI-2536	200378	RIPK2		nM
10041-999-4	BI-2536	200379	RIPK4		nM
10041-999-4	BI-2536	200380	RIPK5		nM
10041-999-4	BI-2536	200381	ROCK1		nM
10041-999-4	BI-2536	200382	ROCK2		nM
10041-999-4	BI-2536	200383	ROS1		nM
10041-999-4	BI-2536	200390	RPS6KA4(Kin.Dom.1-N-terminal)		nM
10041-999-4	BI-2536	200392	RPS6KA4(Kin.Dom.2-C-terminal)	12.0	nM
10041-999-4	BI-2536	200394	RPS6KA5(Kin.Dom.1-N-terminal)		nM
10041-999-4	BI-2536	200396	RPS6KA5(Kin.Dom.2-C-terminal)	270.0	nM
10041-999-4	BI-2536	200399	RSK1(Kin.Dom.1-N-terminal)	5400.0	nM
10041-999-4	BI-2536	200400	RSK1(Kin.Dom.2-C-terminal)		nM
10041-999-4	BI-2536	200401	RSK2(Kin.Dom.1-N-terminal)		nM
10041-999-4	BI-2536	200402	RSK3(Kin.Dom.1-N-terminal)		nM
10041-999-4	BI-2536	200403	RSK3(Kin.Dom.2-C-terminal)	700.0	nM
10041-999-4	BI-2536	200404	RSK4(Kin.Dom.1-N-terminal)		nM
10041-999-4	BI-2536	200405	RSK4(Kin.Dom.2-C-terminal)	1300.0	nM
10041-999-4	BI-2536	200406	S6K1		nM
10041-999-4	BI-2536	200407	SBK1		nM
10041-999-4	BI-2536	200408	SgK110		nM
10041-999-4	BI-2536	200409	SGK3		nM
10041-999-4	BI-2536	200410	SIK1		nM
10041-999-4	BI-2536	200411	SIK2		nM
10041-999-4	BI-2536	200412	SLK	4100.0	nM
10041-999-4	BI-2536	200413	SNARK		nM
10041-999-4	BI-2536	200414	SNRK		nM
10041-999-4	BI-2536	200415	SRC		nM
10041-999-4	BI-2536	200416	SRMS		nM
10041-999-4	BI-2536	200417	SRPK1		nM
10041-999-4	BI-2536	200418	SRPK2		nM
10041-999-4	BI-2536	200419	SRPK3		nM
10041-999-4	BI-2536	200420	STK16	1100.0	nM
10041-999-4	BI-2536	200421	STK33	1100.0	nM
10041-999-4	BI-2536	200422	STK35		nM
10041-999-4	BI-2536	200423	STK36		nM
10041-999-4	BI-2536	200424	STK39		nM
10041-999-4	BI-2536	200425	SYK	4700.0	nM
10041-999-4	BI-2536	200426	TAK1		nM
10041-999-4	BI-2536	200427	TAOK1		nM
10041-999-4	BI-2536	200428	TAOK2		nM
10041-999-4	BI-2536	200429	TAOK3	1700.0	nM
10041-999-4	BI-2536	200430	TBK1		nM
10041-999-4	BI-2536	200431	TEC		nM
10041-999-4	BI-2536	200432	TESK1		nM
10041-999-4	BI-2536	200433	TGFBR1		nM
10041-999-4	BI-2536	200434	TGFBR2		nM
10041-999-4	BI-2536	200435	TIE1		nM
10041-999-4	BI-2536	200436	TIE2		nM
10041-999-4	BI-2536	200437	TLK1		nM
10041-999-4	BI-2536	200438	TLK2		nM
10041-999-4	BI-2536	200439	TNIK		nM
10041-999-4	BI-2536	200440	TNK1		nM
10041-999-4	BI-2536	200441	TNK2		nM
10041-999-4	BI-2536	200442	TNNI3K		nM
10041-999-4	BI-2536	200443	TRKA		nM
10041-999-4	BI-2536	200444	TRKB		nM
10041-999-4	BI-2536	200445	TRKC		nM
10041-999-4	BI-2536	200446	TRPM6		nM
10041-999-4	BI-2536	200447	TSSK1		nM
10041-999-4	BI-2536	200448	TTK	2500.0	nM
10041-999-4	BI-2536	200449	TXK		nM
10041-999-4	BI-2536	200450	TYK2(JH1domain-catalytic)		nM
10041-999-4	BI-2536	200451	TYK2(JH2domain-pseudokinase)		nM
10041-999-4	BI-2536	200454	TYRO3		nM
10041-999-4	BI-2536	200455	ULK1		nM
10041-999-4	BI-2536	200456	ULK2		nM
10041-999-4	BI-2536	200457	ULK3		nM
10041-999-4	BI-2536	200458	VGFR2		nM
10041-999-4	BI-2536	200459	VRK2		nM
10041-999-4	BI-2536	200460	WEE1		nM
10041-999-4	BI-2536	200461	WEE2		nM
10041-999-4	BI-2536	200462	YANK1		nM
10041-999-4	BI-2536	200463	YANK2		nM
10041-999-4	BI-2536	200464	YANK3		nM
10041-999-4	BI-2536	200465	YES		nM
10041-999-4	BI-2536	200466	YSK1		nM
10041-999-4	BI-2536	200467	YSK4	480.0	nM
10041-999-4	BI-2536	200468	MLTK		nM
10041-999-4	BI-2536	200469	ZAP70		nM
